A novel series of [2-[methyl(2-phenethyl)amino]-2-oxoethyl]benzene- containing leukotriene B4 antagonists: Initial structure-activity relationships

Journal of Medicinal Chemistry

Volumn 39, Issue 19, 1996, Pages 3748-3755

  Huang, Fu Chih ^c   Chan, Wan Kit ^a   Moriarty, Kevin J ^a   Poli, Gregory ^a   Morrissette, Matthew M ^a   Galemmo, Robert A ^b   Warus, James D ^a   Dankulich, William P ^a   Sutherland, Charles A ^a  

^a SANOFI   (France)

^b DUPONT COMPANY   (United States)

^c NONE

Author keywords

[No Author keywords available]

Indexed keywords

5 [2 [METHYL(2 PHENYLETHYL)AMINO] 2 OXOETHYL] 2 (BENZYLOXY)CINNAMIC ACID; LEUKOTRIENE B4; LEUKOTRIENE B4 RECEPTOR; LEUKOTRIENE RECEPTOR BLOCKING AGENT; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; GUINEA PIG; HUMAN; HUMAN CELL; NEUTROPHIL; NONHUMAN; SPLEEN CELL; STRUCTURE ACTIVITY RELATION;

ANIMALS; CELL MEMBRANE; CINNAMATES; GUINEA PIGS; HUMANS; LEUKOTRIENE B4; MOLECULAR STRUCTURE; NEUTROPHILS; RECEPTORS, LEUKOTRIENE B4; SPLEEN; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0029816607     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm9506985     Document Type: Article

References (9)

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