Identification of ligand binding determinants in the somatostatin receptor subtypes 1 and 2

Journal of Biological Chemistry

Volumn 271, Issue 34, 1996, Pages 20331-20339

  Liapakis, George ^a   Fitzpatrick, Daniel ^b   Hoeger, Carl ^c   Rivier, Jean ^c   Vandlen, Richard ^b   Reisine, Terry ^a  

^a UNIVERSITY OF PENNSYLVANIA   (United States)

^b GENENTECH INC   (United States)

^c SALK INSTITUTE FOR BIOLOGICAL STUDIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

RECEPTOR SUBTYPE; SOMATOSTATIN RECEPTOR;

AMINO ACID SUBSTITUTION; ANIMAL CELL; ARTICLE; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN DOMAIN; RECEPTOR AFFINITY; RECEPTOR BINDING;

AMINO ACID SEQUENCE; ANIMALS; BINDING, COMPETITIVE; CERCOPITHECUS AETHIOPS; LIGANDS; MEMBRANE GLYCOPROTEINS; MICE; MOLECULAR SEQUENCE DATA; PEPTIDES; RECEPTORS, SOMATOSTATIN; RECOMBINANT FUSION PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP;

ANIMALIA; MATTES; MURINAE;

EID: 0029812686     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.271.34.20331     Document Type: Article

References (38)

1. Bell, G. I., and Reisine T (1993) Trends Neurosci. 16, 34-38
2. Bloom, S., Ralphs, D., Besser, G., Hall, R., Coy, D., Kastin, A., and Schally, A. (1975) Gut 16, 834
3. Brazeau, P., Vale, W., Burgus, R., Ling, N., Rivier, J., and Guillemin, R. (1972) Science 129, 77-79
4. Brown, J. (1990) Am. J. Med. Sci. 300, 267-273
5. Brown, M., Rivier, J., and Vale, W. (1977) Science 196, 1467-1469
6. Bruno, J. F., Xu, Y., Song, J., and Berelowitz, M. (1992) Proc. Natl. Acad. Sci. U. S. A. 89, 11151-11155
7. Buscail, L., Delesque, N., Esteve, J.-P., Saint-Laurent, N., Prats, H., Clerc, P., Robberecht, D., Bell, G. I., Liebow, C., Schally, A. V., Vaysse, N., and Susini, C. (1994) Proc. Natl. Acad. Sci. U. S. A. 91, 2315-2319
8. Buscail, L., Esteve, J. P., Saint-Laurent, N., Bertrand V., Reisine, T., O'Carroll, A. M., Bell, G. I., Schally, A., Vaysse, N., and Susini, C. (1995) Proc. Natl. Acad. Sci. U. S. A. 92, 1580-1584
9. tzpatrick, V., and Vandlen, R. (1994) J. Biol. Chem. 269, 24621-24626
10. Fong, T. M., Anderson, S. A., Yu, H., Huang, R. R. C., and Strader, C. D. (1991) Mol. Pharmacol. 41, 24-30
11. Gomez-Pan, A., Reed, J., Albinus, M., Shaw, B., Hall, R., Besser, G., Coy, D., Kastin, A., and Schally, A. (1975) Lancet 1, 888-890
12. Hellman, B., and Lernmark, A. (1969) Endocrinology 84, 1484-1488
13. Huang, Z., He, Y., Raynor, K., Tallent, M., Reisine, T., and Goodman, M. (1992) J. Am. Chem. Soc. 114, 9390-9401
14. Imai, Y., Matsushima, Y., Sugimura, T., and Terada, M. (1991) Nucleic Acids Res. 19, 2785
15. Kaupmann, K., Brans, C., Raulf, F., Weber, H., Mattes, H., and Lubbert, H. (1995) EMBO J. 14, 727-735
16. Kong, H., Raynor, K., Yano, H., Takeda, J., Bell, G. I., and Reisine, T. (1994) Proc. Natl. Acad. Sci. U. S. A. 91, 8042-8046
17. Kubota, A., Yamada, Y., Kagimoto, S., Shimatsu, A., Imamura, M., Tsuda, K., Imura, H., Seino, S., and Seino, Y. (1994) J. Clin. Invest. 93, 1321-1325
18. Kunkel, T. A. (1985) Proc. Natl. Acad. Sci. U. S. A. 82, 488-492
19. Lamberts, S., Krenning, E., Reubi, J.-C. (1991) Endocr. Rev. 12, 450-482
20. Liapakis, G., Hoeger, C., Rivier, J., and Reisine, T. (1996) J. Pharmacol. Exp. Ther. 276, 1089-1094
21. Liebow, C., Reilly, C., Serrano, M., and Schally, A. (1989) Proc. Natl. Acad. Sci. U. S. A. 86, 2003-2007
22. Mandarino, L., Stenner, D., Blanchard, W., Nissen, S., Gerich, J., Ling, N., Brazeau, P., Bohlen, P., Esch, F., and Guillemin, R. (1981) Nature 291, 76-77
23. O'Carroll, A.-M., Lolait, S. J., Konig, M., and Mahan, L. C. (1992) Mol. Pharmacol. 42, 939-946
24. O'Carroll, A.-M., Raynor, K., Lolait, S. J., and Reisine, T. (1994) Mol. Pharmacol. 48, 291-298
25. Raynor, K., and Reisine, T. (1992) Crit. Rev. Neurobiol. 16, 273-289
26. Raynor, K., Murphy, W., Coy, D., Taylor, J., Moreau, J.-P., Yasuda, K., Bell, G. I., and Reisine, T. (1993a) Mol. Pharmacol. 43, 838-844
27. Raynor, K., O'Carroll, A.-M., Kong, H., Yasuda, K., Mahan, L., Bell, G. I., and Reisine, T. (1993b) Mol. Pharmacol. 44, 385-392
28. Reichlin, S. (1983) N. Engl. J. Med. 309, 1495-1563
29. Reisine, T., and Bell, G. I. (1995) Endocr. Rev. 16, 427-442
30. Rens-Domiano, S., Law, S. F., Yamada, Y., Seino, S., Bell, G. I., and Reisine, T. (1992) Mol. Pharmacol. 42, 28-34
31. Rossowski, W., and Coy, D. (1994) Biochem. Biophys. Res. Commun. 205, 341-346
32. Rossowski, W., Gu, Z., Akarca, U., Jensen, R., and Coy, D. H. (1994) Peptides (Tarryt.) 15, 1421-1424
33. Taylor, J., Theveniau, M., Bashirzadeh, R., Reisine, T., and Eden, P. (1994) Peptides (Tarryt.) 15, 1229-1236
34. Wang, J., Johnson, P., Wu, J., Wang F., and Uhl, G. (1994) J. Biol. Chem. 269, 25966-25969
35. Xue, J., Chen, C., Zhu, J., Kunapuli, S., DeRiel, K., Yu, L., and Liu-Chem, L. (1994) J. Biol. Chem. 269, 30195-30199
36. Yamada, Y., Post, S. R., Wang, K., Tager, H. S., Bell, G. I., and Seino, S. (1992) Proc. Natl. Acad. Sci U. S. A. 89, 251-255
37. Yamada, Y., Reisine, T., Law, S. F., Ihara, Y., Kubota, A., Kagimoto, S., Seino, M., Seino, Y., Bell, G. I., and Seino, S. (1993) Mol. Endocrinol. 6, 2136-2142
38. Yasuda, K., Rens-Domiano, S., Breder, C. D., Law, S. F., Saper, C. B., Reisine, T., and Bell, G. I. (1992) J. Biol. Chem. 267, 20422-20428