Buspirone analogues as ligands of the 5-HT(1A) receptor. II: Capacity factors as chromatographic parameter of lipophilicity evaluation in a series of 5-HT(1A) and 5-HT(2A) receptor ligands

Pharmazie

Volumn 51, Issue 12, 1996, Pages 924-927

  Chilmonczyk, Z ^a   Ksycinska H ^a   Cybulski, J ^a   Wozniakowska Szelejewska A ^a  

^a INDUSTRIAL CHEMISTRY RESEARCH INSTITUTE   (Poland)

Author keywords

[No Author keywords available]

Indexed keywords

BUSPIRONE; BUSPIRONE DERIVATIVE; SEROTONIN AGONIST; UNCLASSIFIED DRUG;

ARTICLE; LIPOPHILICITY; REVERSED PHASE HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; TECHNIQUE; THEORY;

BUSPIRONE; CALIBRATION; CHEMISTRY, PHYSICAL; HYDROGEN-ION CONCENTRATION; INDICATORS AND REAGENTS; LIGANDS; RECEPTORS, SEROTONIN; SEROTONIN ANTAGONISTS;

EID: 0029802449     PISSN: 00317144     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (22)

1. Maj, J.; Lewandowska, A.: Pol. J. Pharmacol. Pharm. 32, 495 (1980)
2. Simansky, K. J.; Schechter, L. E.: J. Pharmacol. Exp. Ther. 247, 1073 (1988)
3. Glennon, R. A.; Naiman, N. A.; Prieson, M. E.; Titeler, M.; Lyon, R. A.; Herndon, J. L.: Drug Dev. Res. 16, 335 (1989)
4. Tatarczyńska, E.; Pawłowski, L.; Chojnacka-Wójcik, E.; Maj, J.: Pol. J. Pharmacol. Pharm. 41, 51 (1989)
5. Romero, A. G.; McCall, R. B.; in: Bristol, J. A. (Ed.): Advances in Medicinal Chemistry, vol. 27. Ch. 3, Academic Press, New York 1991
6. Murphy, D. L.; Leach, K. P.; Aulakh, C. S.; Pigott, T. A.: Pharmacol. Rev. 43, 527 (1991)
7. Goa, K.; Ward, A.: Drugs 32, 114 (1986)
8. Cybulski, J.; Chilmonczyk, Z.; Szelejewski, W.; Wojtasiewicz, K.; Wróbel, J. T.: Arch. Pharm. (Weinheim) 325, 313 (1992)
9. Chilmonczyk, Z.; Woźniakowska, A.; Cybulski, J.: To be published
10. Kuchar, M.; Jelínková, M.; in: Kuchar, M. (Ed.): QSAR in Design of Bioactive Compounds, p. 65, J. R. Prous Science Publishers, S. A./ Barcelona 1992
11. Tomlinson, E.: J. Chromatogr. 113, 1 (1975)
12. Kuchar, M.; Rejholec, V.: Cesk. Farm. 28, 212 (1979)
13. Carney, C. F.: J. Liquid Chromatogr. 8, 2781 (1985)
14. Kaliszan, R.: Quantitative Structure-Chromatographic Retention Relationships, Wiley, New York 1987
15. McCall, J. M.: J. Med. Chem. 18, 549 (1975)
16. Unger, S. H.; Cook, J. R.; Hollenberg, J. S.: J. Pharm. Sci. 67, 1364 (1978)
17. Tsantili-Kakoulidou, A.; Filippatos, E.; Todoulou, O.; Papadali-Valiraki, A.: J. Chromatogr. 654, 43 (1993)
18. Bechalany, A.; Tsantili-Kakoulidou, A.; El Tayar, N.; Testa, B.: J. Chromatogr. 541, 221 (1991)
19. Chen, N.; Zhang, Y.; Lu, P.: J. Chromatogr. 633, 31 (1993)
20. Valko, K.: J. Liq. Chromatogr. 10, 1663 (1987)
21. Schere, R. A.; Howard, S. M.: J. Med. Chem. 20, 53 (1977)
22. Leo, A.; Hansch, C.; Elkins, D.: Chem. Rev. 71, 525 (1971)