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Volumn 31, Issue 4, 1996, Pages 246-256

Clinical pharmacokinetics of bambuterol

Author keywords

[No Author keywords available]

Indexed keywords

BAMBUTEROL; CHOLINESTERASE; PRODRUG; SALBUTAMOL; SUXAMETHONIUM; TERBUTALINE;

EID: 0029797109     PISSN: 03125963     EISSN: None     Source Type: Journal    
DOI: 10.2165/00003088-199631040-00002     Document Type: Review
Times cited : (52)

References (48)
  • 1
    • 0027511935 scopus 로고
    • A placebo-controlled dose-finding study with bambuterol in elderly patients with asthma
    • Sitar DS, Aoki FY, Warren CP, et al. A placebo-controlled dose-finding study with bambuterol in elderly patients with asthma. Chest 1993; 103: 771-6
    • (1993) Chest , vol.103 , pp. 771-776
    • Sitar, D.S.1    Aoki, F.Y.2    Warren, C.P.3
  • 2
    • 0024166436 scopus 로고
    • The design and bioactivation of pre-systemically stable prodrugs
    • Svennson L-Å, Tunek A. The design and bioactivation of pre-systemically stable prodrugs. Drug Metab Rev 1988; 19: 165-94
    • (1988) Drug Metab Rev , vol.19 , pp. 165-194
    • Svennson, L.-Å.1    Tunek, A.2
  • 3
    • 0023724238 scopus 로고
    • Bambuterol, a carbamate ester prodrug of terbutaline, as inhibitor of cholinesterases in human blood
    • Tunek A, Svennson L-Å. Bambuterol, a carbamate ester prodrug of terbutaline, as inhibitor of cholinesterases in human blood. Drug Metab Dispos 1988; 16: 759-64
    • (1988) Drug Metab Dispos , vol.16 , pp. 759-764
    • Tunek, A.1    Svennson, L.-Å.2
  • 4
    • 0023820851 scopus 로고
    • 3H-bambuterol, a carbamate prodrug of terbutaline, in blood from humans and laboratory animals in vitro
    • 3H-bambuterol, a carbamate prodrug of terbutaline, in blood from humans and laboratory animals in vitro. Biochem Pharmacol 1988; 37: 3867-76
    • (1988) Biochem Pharmacol , vol.37 , pp. 3867-3876
    • Tunek, A.1    Levin, E.2    Svennson, L.-Å.3
  • 6
    • 0014907857 scopus 로고
    • Some pharmacological properties of terbutaline (INN), 1-(3,5-dihydroxyphenyl)-2-(t-butylamino)-ethanol. A new sympathomimetic β-receptor-stimulating agent
    • Persson H, Olsson T. Some pharmacological properties of terbutaline (INN), 1-(3,5-dihydroxyphenyl)-2-(t-butylamino)-ethanol. A new sympathomimetic β-receptor-stimulating agent. Acta Med Scand 1979; Suppl. 512: 11-9
    • (1979) Acta Med Scand , Issue.512 SUPPL. , pp. 11-19
    • Persson, H.1    Olsson, T.2
  • 7
    • 0015715187 scopus 로고
    • Terbutaline: A preliminary report of its pharmacological properties and therapeutic efficacy in asthma
    • Brogden RN, Speight TM, Avery GS. Terbutaline: a preliminary report of its pharmacological properties and therapeutic efficacy in asthma. Drugs 1973; 6: 324-32
    • (1973) Drugs , vol.6 , pp. 324-332
    • Brogden, R.N.1    Speight, T.M.2    Avery, G.S.3
  • 9
    • 0017383946 scopus 로고
    • Quantitative analysis of terbutaline in serum and urine at therapeutic levels using gas chromatography-mass spectrometry
    • Lefrink JG, Wagemaker-Engels I, Maees RAA, et al. Quantitative analysis of terbutaline in serum and urine at therapeutic levels using gas chromatography-mass spectrometry. J Chromatogr 1977; 143: 299-305
    • (1977) J Chromatogr , vol.143 , pp. 299-305
    • Lefrink, J.G.1    Wagemaker-Engels, I.2    Maees, R.A.A.3
  • 10
    • 0018417292 scopus 로고
    • The analysis of terbutaline in biological fluids by gas chromatography electron impact mass spectrometry
    • Clare RA, Davies DS, Baillie TA. The analysis of terbutaline in biological fluids by gas chromatography electron impact mass spectrometry. Biomed Mass Spectrum 1979; 6: 31-7
    • (1979) Biomed Mass Spectrum , vol.6 , pp. 31-37
    • Clare, R.A.1    Davies, D.S.2    Baillie, T.A.3
  • 11
    • 0019274642 scopus 로고
    • Determination of terbutaline in plasma by gas chromatography chemical ionization mass spectrometry
    • Jacobsson S-E, Jönsson S, Lindberg C, et al. Determination of terbutaline in plasma by gas chromatography chemical ionization mass spectrometry. Biomed Mass Spectrom 1980; 7: 265-8
    • (1980) Biomed Mass Spectrom , vol.7 , pp. 265-268
    • Jacobsson, S.-E.1    Jönsson, S.2    Lindberg, C.3
  • 12
    • 0020359905 scopus 로고
    • Automated analysis of terbutaline (Bricanyl®) in human plasma with liquid chromatography and electrochemical detection using column switching (multidimensional chromatography)
    • Edholm L-E, Kennedy B-M, Bergquist S. Automated analysis of terbutaline (Bricanyl®) in human plasma with liquid chromatography and electrochemical detection using column switching (multidimensional chromatography). Chromatographia 1982; 16: 341-4
    • (1982) Chromatographia , vol.16 , pp. 341-344
    • Edholm, L.-E.1    Kennedy, B.-M.2    Bergquist, S.3
  • 13
    • 0021319691 scopus 로고
    • Multidimensional column liquid chromatography with electrochemical detection for the analysis of terbutaline in human plasma
    • Edholm L-E, Kennedy B-M, Bergquist S. Multidimensional column liquid chromatography with electrochemical detection for the analysis of terbutaline in human plasma. Eur J Resp Dis 1984; 65 Suppl. 134: 33-40
    • (1984) Eur J Resp Dis , vol.65 , Issue.134 SUPPL. , pp. 33-40
    • Edholm, L.-E.1    Kennedy, B.-M.2    Bergquist, S.3
  • 14
    • 0001666249 scopus 로고
    • Quantitative determination of terbutaline in human plasma after administration of bambuterol using coupled columns and electrochemical detection
    • Kennedy B-M, Blomgren A, Deholm L-E, et al. Quantitative determination of terbutaline in human plasma after administration of bambuterol using coupled columns and electrochemical detection. Chromatographia 1987; 24: 895-9
    • (1987) Chromatographia , vol.24 , pp. 895-899
    • Kennedy, B.-M.1    Blomgren, A.2    Deholm, L.-E.3
  • 15
    • 0017254117 scopus 로고
    • The relative bioavailability of terbutaline (Bricanyl®) elixir and tablet formulations
    • Sitar DS, Piafsky KM, Ogilvie RI. The relative bioavailability of terbutaline (Bricanyl®) elixir and tablet formulations. Curr Ther Res 1976; 19: 266-73
    • (1976) Curr Ther Res , vol.19 , pp. 266-273
    • Sitar, D.S.1    Piafsky, K.M.2    Ogilvie, R.I.3
  • 16
    • 0021327011 scopus 로고
    • Pharmacokinetic parameters of terbutaline in healthy man: An overview
    • Nyberg L. Pharmacokinetic parameters of terbutaline in healthy man: an overview. Eur J Respir Dis 1984; 65 Suppl. 134: 149-60
    • (1984) Eur J Respir Dis , vol.65 , Issue.134 SUPPL. , pp. 149-160
    • Nyberg, L.1
  • 18
    • 0025756009 scopus 로고
    • Bambuterol: A new long acting bronchodilating prodrug
    • Vilsvik JS, Langaker O, Persson G, et al. Bambuterol: a new long acting bronchodilating prodrug. Ann Allergy 1991; 66: 315-9
    • (1991) Ann Allergy , vol.66 , pp. 315-319
    • Vilsvik, J.S.1    Langaker, O.2    Persson, G.3
  • 19
    • 0023900866 scopus 로고
    • Bambuterol: Clinical effects of different doses of a long-acting bronchodilator prodrug
    • Sandström T, Åsander L, Clemmensen IH, et al. Bambuterol: clinical effects of different doses of a long-acting bronchodilator prodrug. Respiration 1988; 53: 31-6
    • (1988) Respiration , vol.53 , pp. 31-36
    • Sandström, T.1    Åsander, L.2    Clemmensen, I.H.3
  • 20
    • 0022647011 scopus 로고
    • Bambuterol: Dose response study of a new terbutaline prodrug in asthma
    • Holstein-Rathlou N-H, Laursen LC, Madsen F, et al. Bambuterol: dose response study of a new terbutaline prodrug in asthma. Eur J Clin Pharmacol 1986; 30: 7-11
    • (1986) Eur J Clin Pharmacol , vol.30 , pp. 7-11
    • Holstein-Rathlou, N.-H.1    Laursen, L.C.2    Madsen, F.3
  • 21
    • 0026737843 scopus 로고
    • Pharmacokinetics and pharmacodynamics of bambuterol, a long-acting bronchodilator prodrug of terbutaline, in young and elderly patients with asthma
    • Sitar DS, Warren CP, Aoki FY. Pharmacokinetics and pharmacodynamics of bambuterol, a long-acting bronchodilator prodrug of terbutaline, in young and elderly patients with asthma. Clin Pharmacol Ther 1992; 52: 297-306
    • (1992) Clin Pharmacol Ther , vol.52 , pp. 297-306
    • Sitar, D.S.1    Warren, C.P.2    Aoki, F.Y.3
  • 22
    • 0028854625 scopus 로고
    • Bambuterol in the treatment of asthma: A placebo-controlled comparison of once-daily morning vs evening administration
    • D'Alonzo GE, Smolensky MH, Feldman S, et al. Bambuterol in the treatment of asthma: a placebo-controlled comparison of once-daily morning vs evening administration. Chest 1995; 107: 406-12
    • (1995) Chest , vol.107 , pp. 406-412
    • D'Alonzo, G.E.1    Smolensky, M.H.2    Feldman, S.3
  • 23
    • 0021317659 scopus 로고
    • Pharmacokinetics of terbutaline after parenteral administration
    • Fagerström P-O. Pharmacokinetics of terbutaline after parenteral administration. Eur J Resp Dis 1984; 65 Suppl. 134: 101-10
    • (1984) Eur J Resp Dis , vol.65 , Issue.134 SUPPL. , pp. 101-110
    • Fagerström, P.-O.1
  • 24
    • 0023882809 scopus 로고
    • Bambuterol: Uptake and metabolism in guinea pig isolated lungs
    • Ryrfeldt Å, Nilsson E, Tunek A, et al. Bambuterol: uptake and metabolism in guinea pig isolated lungs. Pharm Res 1988; 5: 151-5
    • (1988) Pharm Res , vol.5 , pp. 151-155
    • Ryrfeldt, Å.1    Nilsson, E.2    Tunek, A.3
  • 25
    • 0015266111 scopus 로고
    • The tissue distribution of 3H-terbutaline (Bricanyl®) in mice
    • Bodin NO, Hansson E, Ramsay CH, et al. The tissue distribution of 3H-terbutaline (Bricanyl®) in mice. Acta Physiol Scand 1972; 84: 40-7
    • (1972) Acta Physiol Scand , vol.84 , pp. 40-47
    • Bodin, N.O.1    Hansson, E.2    Ramsay, C.H.3
  • 26
    • 0021306989 scopus 로고
    • Distribution of terbutaline
    • Ryrfeldt Å, Ramsay CH. Distribution of terbutaline. Eur J Resp Dis 1984; 65 Suppl. 134: 63-72
    • (1984) Eur J Resp Dis , vol.65 , Issue.134 SUPPL. , pp. 63-72
    • Ryrfeldt, Å.1    Ramsay, C.H.2
  • 27
    • 0024321858 scopus 로고
    • Metabolism of bambuterol in rat liver microsomes: Identification of hydroxylated and demethylated products by liquid chromatography mass spectrometry
    • Lindberg C, Roos C, Tunek A, et al. Metabolism of bambuterol in rat liver microsomes: identification of hydroxylated and demethylated products by liquid chromatography mass spectrometry. Drug Metab Dispos 1989; 17: 311-22
    • (1989) Drug Metab Dispos , vol.17 , pp. 311-322
    • Lindberg, C.1    Roos, C.2    Tunek, A.3
  • 28
    • 10244249572 scopus 로고
    • Pharmacokinetic properties of bambuterol in solution and tablets-basis for once daily dosage in asthma
    • Nyberg L. Pharmacokinetic properties of bambuterol in solution and tablets-basis for once daily dosage in asthma. Acta Pharmacol Toxicologica 1986; 59 Suppl. V: 229
    • (1986) Acta Pharmacol Toxicologica , vol.59 , Issue.SUPPL. V , pp. 229
    • Nyberg, L.1
  • 30
    • 0018382383 scopus 로고
    • Asthma in the elderly: An epidemiological survey
    • Burr ML, Charles TJ, Roy K, et al. Asthma in the elderly: an epidemiological survey. BMJ 1979; 1: 1041-7
    • (1979) BMJ , vol.1 , pp. 1041-1047
    • Burr, M.L.1    Charles, T.J.2    Roy, K.3
  • 31
    • 0027501242 scopus 로고
    • Bambuterol: Effective in nocturnal asthma
    • Petrie GR, Chookang JY, Hassan WU, et al. Bambuterol: effective in nocturnal asthma. Respir Med 1993; 87: 581-5
    • (1993) Respir Med , vol.87 , pp. 581-585
    • Petrie, G.R.1    Chookang, J.Y.2    Hassan, W.U.3
  • 32
    • 0023771614 scopus 로고
    • Bambuterol: Clinical effects of three doses of bambuterol once daily in asthmatic patients
    • Clemmensen IH, Pedersen BK, Ravn S, et al. Bambuterol: clinical effects of three doses of bambuterol once daily in asthmatic patients. Allergy 1988; 43: 573-6
    • (1988) Allergy , vol.43 , pp. 573-576
    • Clemmensen, I.H.1    Pedersen, B.K.2    Ravn, S.3
  • 33
    • 0023896309 scopus 로고
    • Comparison between a new once-daily, bronchodilating drug, bambuterol, and terbutaline sustained-release, twice daily
    • Persson G, Gnosspelius Y, Anehus S. Comparison between a new once-daily, bronchodilating drug, bambuterol, and terbutaline sustained-release, twice daily. Eur Respir J 1988; 1: 223-6
    • (1988) Eur Respir J , vol.1 , pp. 223-226
    • Persson, G.1    Gnosspelius, Y.2    Anehus, S.3
  • 34
    • 0027140146 scopus 로고
    • Therapeutic equivalence between bambuterol, 10mg once daily, and terbutaline controlled release, 5mg twice daily, in mild to moderate asthma
    • Fugleholm AM, Ibsen TB, Laxmyr L, et al. Therapeutic equivalence between bambuterol, 10mg once daily, and terbutaline controlled release, 5mg twice daily, in mild to moderate asthma. Eur Respir J 1993; 6: 1474-8
    • (1993) Eur Respir J , vol.6 , pp. 1474-1478
    • Fugleholm, A.M.1    Ibsen, T.B.2    Laxmyr, L.3
  • 35
    • 0029029678 scopus 로고
    • Oral bambuterol versus terbutaline in patients with asthma
    • Persson G, Pahlm O, Gnosspelius Y. Oral bambuterol versus terbutaline in patients with asthma. Curr Ther Res 1995; 56: 457-65
    • (1995) Curr Ther Res , vol.56 , pp. 457-465
    • Persson, G.1    Pahlm, O.2    Gnosspelius, Y.3
  • 36
    • 0026783304 scopus 로고
    • Effects of budesonide and bambuterol on circadian variation of airway responsiveness and nocturnal symptoms of asthma
    • Wempe JB, Tammeling EP, Postma DS, et al. Effects of budesonide and bambuterol on circadian variation of airway responsiveness and nocturnal symptoms of asthma. J Allergy Clin Immunol 1992; 90: 349-57
    • (1992) J Allergy Clin Immunol , vol.90 , pp. 349-357
    • Wempe, J.B.1    Tammeling, E.P.2    Postma, D.S.3
  • 37
    • 0028918942 scopus 로고
    • Comparison of the efficacy, tolerability and patient acceptability of once-daily bambuterol tablets against twice-daily controlled release salbutamol in nocturnal asthma
    • Gunn SD, Ayres JG, McConchie SM, et al. Comparison of the efficacy, tolerability and patient acceptability of once-daily bambuterol tablets against twice-daily controlled release salbutamol in nocturnal asthma. Eur J Clin Pharmacol 1995; 48: 23-8
    • (1995) Eur J Clin Pharmacol , vol.48 , pp. 23-28
    • Gunn, S.D.1    Ayres, J.G.2    McConchie, S.M.3
  • 38
    • 0027379684 scopus 로고
    • Tremor in healthy volunteers after bambuterol and terbutaline CR-tablets
    • Larsén K, Schmekel B. Tremor in healthy volunteers after bambuterol and terbutaline CR-tablets. Eur J Clin Pharmacol 1993; 45: 303-5
    • (1993) Eur J Clin Pharmacol , vol.45 , pp. 303-305
    • Larsén, K.1    Schmekel, B.2
  • 39
    • 0017067925 scopus 로고
    • Salbutamol and hypokalemia
    • Deacon SP. Salbutamol and hypokalemia. Lancet 1976; I: 1302
    • (1976) Lancet , vol.1 , pp. 1302
    • Deacon, S.P.1
  • 40
    • 0017258354 scopus 로고
    • Effect of intravenous infusion of salbutamol on ventilatory response to carbon dioxide and hypoxia and on heart rate and plasma potassium in normal men
    • Leitch AG, Clancy LJ, Costello JF, et al. Effect of intravenous infusion of salbutamol on ventilatory response to carbon dioxide and hypoxia and on heart rate and plasma potassium in normal men. BMJ 1976; 1: 365-7
    • (1976) BMJ , vol.1 , pp. 365-367
    • Leitch, A.G.1    Clancy, L.J.2    Costello, J.F.3
  • 41
    • 0026476530 scopus 로고
    • Blood eosinophil numbers and activity during 24 hours: Effects of treatment with budesonide and bambuterol
    • Wempe JB, Tammeling EP, Koëter GH, et al. Blood eosinophil numbers and activity during 24 hours: effects of treatment with budesonide and bambuterol. J Allergy Clin Immunol 1992; 90: 757-65
    • (1992) J Allergy Clin Immunol , vol.90 , pp. 757-765
    • Wempe, J.B.1    Tammeling, E.P.2    Koëter, G.H.3
  • 42
    • 0023811801 scopus 로고
    • The influence of bambuterol (carbamylated terbutaline) on the duration of action of succinylcholine-induced paralysis in humans
    • Fisher DM, Caldwell JE, Sharma M, et al. The influence of bambuterol (carbamylated terbutaline) on the duration of action of succinylcholine-induced paralysis in humans. Anesthesiology 1988; 69: 757-9
    • (1988) Anesthesiology , vol.69 , pp. 757-759
    • Fisher, D.M.1    Caldwell, J.E.2    Sharma, M.3
  • 43
    • 0025160867 scopus 로고
    • The influence of 10mg and 20mg of bambuterol on the duration of succinylcholine-induced neuromuscular blockade
    • Staun P, Lennmarken C, Eriksson LI, et al. The influence of 10mg and 20mg of bambuterol on the duration of succinylcholine-induced neuromuscular blockade. Acta Anaesthesiol Scand 1990; 34: 498-500
    • (1990) Acta Anaesthesiol Scand , vol.34 , pp. 498-500
    • Staun, P.1    Lennmarken, C.2    Eriksson, L.I.3
  • 44
    • 0025144977 scopus 로고
    • The effect of bambuterol (carbamylated terbutaline) on plasma cholinesterase activity and suxamethonium-induced neuromuscular blockade in genotypically normal patients
    • Bang U, Viby-Mogensen J, Wirén JE, et al. The effect of bambuterol (carbamylated terbutaline) on plasma cholinesterase activity and suxamethonium-induced neuromuscular blockade in genotypically normal patients. Acta Anaesthesiol Scand 1990; 34: 596-9
    • (1990) Acta Anaesthesiol Scand , vol.34 , pp. 596-599
    • Bang, U.1    Viby-Mogensen, J.2    Wirén, J.E.3
  • 45
    • 0025130933 scopus 로고
    • The effect of bambuterol on plasma cholinesterase activity and suxamethonium-induced neuromuscular blockade in subjects heterozygous for abnormal plasma cholinesterase
    • Hang U, Viby-Mogensen J, Wirén JE. The effect of bambuterol on plasma cholinesterase activity and suxamethonium-induced neuromuscular blockade in subjects heterozygous for abnormal plasma cholinesterase. Acta Anaesthesiol Scand 1990; 34: 600-4
    • (1990) Acta Anaesthesiol Scand , vol.34 , pp. 600-604
    • Hang, U.1    Viby-Mogensen, J.2    Wirén, J.E.3
  • 46
    • 0021114613 scopus 로고
    • Asthma at night
    • Asthma at night [editorial]. Lancet 1983; I: 220-2
    • (1983) Lancet , vol.1 , pp. 220-222
  • 47
    • 0028817898 scopus 로고
    • Long-acting inhaled beta agonists
    • Tilles SA, Nelson HS. Long-acting inhaled beta agonists. J Asthma 1995; 32: 397-404
    • (1995) J Asthma , vol.32 , pp. 397-404
    • Tilles, S.A.1    Nelson, H.S.2
  • 48
    • 0028823060 scopus 로고
    • Rapid onset of tolerance to the bronchoprotective effect of salmeterol
    • Bhagat R, Kalra S, Swystun VA, et al. Rapid onset of tolerance to the bronchoprotective effect of salmeterol. Chest 1995; 108: 1235-39
    • (1995) Chest , vol.108 , pp. 1235-1239
    • Bhagat, R.1    Kalra, S.2    Swystun, V.A.3


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