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Volumn 85, Issue 4, 1996, Pages 655-661

Effect of the novel high-affinity glycine-site N-methyl-D-aspartate antagonist ACEA- 1021 on 125I-MK-801 binding after subdural hematoma in the rat: An in vivo autoradiographic study

Author keywords

ACEA 1021; acute subdural hematoma; head injury; in vivo autoradiography; MK 801; N methyl D aspartate ion channel activation

Indexed keywords

6,7 DICHLORO 5 NITRO 2,3 QUINOXALINEDIONE; DIZOCILPINE; IODINE 125; N METHYL DEXTRO ASPARTIC ACID RECEPTOR; N METHYL DEXTRO ASPARTIC ACID RECEPTOR BLOCKING AGENT;

EID: 0029791376     PISSN: 00223085     EISSN: None     Source Type: Journal    
DOI: 10.3171/jns.1996.85.4.0655     Document Type: Article
Times cited : (27)

References (34)
  • 1
    • 0026674622 scopus 로고
    • Enhanced calcium uptake by CA1 pyramidal cell dendrites in the postischemic phase despite subnormal evoked field potentials: Excitatory amino acid receptor dependency and relationship to neuronal damage
    • Andiné P, Jacobson I, Hagberg H: Enhanced calcium uptake by CA1 pyramidal cell dendrites in the postischemic phase despite subnormal evoked field potentials: excitatory amino acid receptor dependency and relationship to neuronal damage. J Cereb Blood Flow Metab 12:773-783, 1992
    • (1992) J Cereb Blood Flow Metab , vol.12 , pp. 773-783
    • Andiné, P.1    Jacobson, I.2    Hagberg, H.3
  • 2
    • 0027295901 scopus 로고
    • Excitatory amino acids in cerebrospinal fluid following traumatic brain injury in humans
    • Baker AJ, Moulton RJ, MacMillan VH, et al: Excitatory amino acids in cerebrospinal fluid following traumatic brain injury in humans. J Neurosurg 79:369-372, 1993
    • (1993) J Neurosurg , vol.79 , pp. 369-372
    • Baker, A.J.1    Moulton, R.J.2    MacMillan, V.H.3
  • 4
    • 0025036657 scopus 로고
    • Comparison of phenytoin with noncompetitive N-methyl-D-aspartate antagonists in a model of focal brain ischemia in rat
    • Boxer PA, Cordon JJ, Mann ME, et al: Comparison of phenytoin with noncompetitive N-methyl-D-aspartate antagonists in a model of focal brain ischemia in rat. Stroke 21 (Suppl): III47-I1I51, 1990
    • (1990) Stroke , vol.21 , Issue.SUPPL.
    • Boxer, P.A.1    Cordon, J.J.2    Mann, M.E.3
  • 5
    • 0025653345 scopus 로고
    • Changes in extracellular glutamate concentration after acute subdural haematoma in the rat - Evidence for an "excitotoxic" mechanism?
    • Bullock R, Butcher S, McCulloch J: Changes in extracellular glutamate concentration after acute subdural haematoma in the rat - evidence for an "excitotoxic" mechanism? Acta Neurochir Suppl 51:274-276, 1990
    • (1990) Acta Neurochir Suppl , vol.51 , pp. 274-276
    • Bullock, R.1    Butcher, S.2    McCulloch, J.3
  • 6
    • 0025783089 scopus 로고
    • Correlation of the extracellular glutamate concentration with extent of blood flow reduction after subdural hematoma in the rat
    • Bullock R, Butcher SP, Chen MH, et al: Correlation of the extracellular glutamate concentration with extent of blood flow reduction after subdural hematoma in the rat. J Neurosurg 74: 794-802, 1991
    • (1991) J Neurosurg , vol.74 , pp. 794-802
    • Bullock, R.1    Butcher, S.P.2    Chen, M.H.3
  • 7
    • 0025142948 scopus 로고
    • Focal cerebral ischemia in the cat: Pretreatment with a competitive NMDA receptor antagonist, D-CPP-ene
    • Bullock R, Graham DI, Chen MH, et al: Focal cerebral ischemia in the cat: pretreatment with a competitive NMDA receptor antagonist, D-CPP-ene. J Cereb Blood Flow Metab 10: 668-674, 1990
    • (1990) J Cereb Blood Flow Metab , vol.10 , pp. 668-674
    • Bullock, R.1    Graham, D.I.2    Chen, M.H.3
  • 8
    • 0025811662 scopus 로고
    • Glial swelling following human cerebral contusion: An ultrastructural study
    • Bullock R, Maxwell WL, Graham DI, et al: Glial swelling following human cerebral contusion: an ultrastructural study. J Neurol Neurosurg Psychiatry 54:427-434, 1991
    • (1991) J Neurol Neurosurg Psychiatry , vol.54 , pp. 427-434
    • Bullock, R.1    Maxwell, W.L.2    Graham, D.I.3
  • 9
    • 0343612488 scopus 로고
    • Experience with the glutamate antagonist CGS19755 in severe human head injury: Evidence for ICP lowering effect
    • Nagai H, Kamiya K, Ishii S (eds): Tokyo: Springer-Verlag
    • Bullock R, Teasdale GM, Kotake A, et al: Experience with the glutamate antagonist CGS19755 in severe human head injury: evidence for ICP lowering effect, in Nagai H, Kamiya K, Ishii S (eds): Intracranial Pressure IX. Tokyo: Springer-Verlag, 1994, pp 238-241
    • (1994) Intracranial Pressure , vol.9 , pp. 238-241
    • Bullock, R.1    Teasdale, G.M.2    Kotake, A.3
  • 11
    • 0025763921 scopus 로고
    • Evaluation of a competitive NMDA antagonist (D-CPPene) in feline focal cerebral ischemia
    • Chen M, Bullock R, Graham DI, et al: Evaluation of a competitive NMDA antagonist (D-CPPene) in feline focal cerebral ischemia. Ann Neurol 30:62-70, 1991
    • (1991) Ann Neurol , vol.30 , pp. 62-70
    • Chen, M.1    Bullock, R.2    Graham, D.I.3
  • 12
    • 0025809541 scopus 로고
    • Ischemic neuronal damage after acute subdural hematoma in the rat: Effects of pretreatment with a glutamate antagonist
    • Chen MH, Bullock R, Graham DI, et al: Ischemic neuronal damage after acute subdural hematoma in the rat: effects of pretreatment with a glutamate antagonist. J Neurosurg 74: 944-950, 1991
    • (1991) J Neurosurg , vol.74 , pp. 944-950
    • Chen, M.H.1    Bullock, R.2    Graham, D.I.3
  • 13
    • 0023870521 scopus 로고
    • Pharmacology of glutamate neuroloxicity in cortical cell culture: Attenuation by NMDA antagonists
    • Choi DW, Koh J, Peters S: Pharmacology of glutamate neuroloxicity in cortical cell culture: attenuation by NMDA antagonists. J Neurosci 8:185-196, 1988
    • (1988) J Neurosci , vol.8 , pp. 185-196
    • Choi, D.W.1    Koh, J.2    Peters, S.3
  • 14
    • 0024405516 scopus 로고
    • Selective vulnerability of the brain: New insights into the pathophysiology of stroke
    • Collins RC, Dobkin BH, Choi DW: Selective vulnerability of the brain: new insights into the pathophysiology of stroke. Ann Intern Med 110:992-1000, 1989
    • (1989) Ann Intern Med , vol.110 , pp. 992-1000
    • Collins, R.C.1    Dobkin, B.H.2    Choi, D.W.3
  • 15
    • 0023778442 scopus 로고
    • Effect of ischemia and intra-amygdaloid kainate injection on the density of NMDA binding sites in the hippocampal CA1 region
    • Crepel V, Represa A, Ben-Ari Y: Effect of ischemia and intra-amygdaloid kainate injection on the density of NMDA binding sites in the hippocampal CA1 region. Eur J Pharmacol 151: 355-356, 1988
    • (1988) Eur J Pharmacol , vol.151 , pp. 355-356
    • Crepel, V.1    Represa, A.2    Ben-Ari, Y.3
  • 16
    • 0028189686 scopus 로고
    • Focal microvascular occlusion after acute subdural haematoma in the rat: A mechanism for ischaemic damage and brain swelling?
    • Fujisawa H, Maxwell WL, Graham DI, et al: Focal microvascular occlusion after acute subdural haematoma in the rat: a mechanism for ischaemic damage and brain swelling? Acta Neurochir Suppl 60:193-196, 1994
    • (1994) Acta Neurochir Suppl , vol.60 , pp. 193-196
    • Fujisawa, H.1    Maxwell, W.L.2    Graham, D.I.3
  • 17
    • 0026794490 scopus 로고
    • Glucose hypermetabolism after acute subdural hematoma is ameliorated by a competitive NMDA antagonist
    • Inglis F, Kuroda Y, Bullock R: Glucose hypermetabolism after acute subdural hematoma is ameliorated by a competitive NMDA antagonist. J Neurotrauma 9:75-84, 1992
    • (1992) J Neurotrauma , vol.9 , pp. 75-84
    • Inglis, F.1    Kuroda, Y.2    Bullock, R.3
  • 18
    • 0026761089 scopus 로고
    • Local cerebral blood flow mapping before and after removal of acute subdural hematoma in the rat
    • Kuroda Y, Bullock R: Local cerebral blood flow mapping before and after removal of acute subdural hematoma in the rat. Neurosurgery 30:687-691, 1992
    • (1992) Neurosurgery , vol.30 , pp. 687-691
    • Kuroda, Y.1    Bullock, R.2
  • 19
    • 0027301088 scopus 로고
    • Early changes in second messenger but not receptor binding sites after acute subdural hematoma: An in vitro autoradiographic study
    • Kuroda Y, Dewar D, Bullock R: Early changes in second messenger but not receptor binding sites after acute subdural hematoma: an in vitro autoradiographic study. J Neurotrauma 10:47-55, 1993
    • (1993) J Neurotrauma , vol.10 , pp. 47-55
    • Kuroda, Y.1    Dewar, D.2    Bullock, R.3
  • 20
    • 0026535412 scopus 로고
    • Transient glucose hyper-metabolism after acute subdural hematoma in the rat
    • Kuroda Y, Inglis FM, Miller JD, et al: Transient glucose hyper-metabolism after acute subdural hematoma in the rat. J Neurosurg 76:471-477, 1992
    • (1992) J Neurosurg , vol.76 , pp. 471-477
    • Kuroda, Y.1    Inglis, F.M.2    Miller, J.D.3
  • 21
    • 0026488921 scopus 로고
    • NMDA receptor-mediated arachidonic acid release in neurons: Role in signal transduction and pathological aspects
    • Lazarewicz JW, Salinska E, Wroblewski JT: NMDA receptor-mediated arachidonic acid release in neurons: role in signal transduction and pathological aspects. Adv Exp Med Biol 318: 73-89, 1992
    • (1992) Adv Exp Med Biol , vol.318 , pp. 73-89
    • Lazarewicz, J.W.1    Salinska, E.2    Wroblewski, J.T.3
  • 22
    • 0026697498 scopus 로고
    • Protective effect of synaptic inhibition during cerebral ischemia in rats and rabbits
    • Lyden PD, Hedges B: Protective effect of synaptic inhibition during cerebral ischemia in rats and rabbits. Stroke 23: 1463-1469, 1992
    • (1992) Stroke , vol.23 , pp. 1463-1469
    • Lyden, P.D.1    Hedges, B.2
  • 23
    • 0028132189 scopus 로고
    • Effects of glycine receptor antagonism on spreading depression in the rat
    • Martin H, Warner DS, Todd MM: Effects of glycine receptor antagonism on spreading depression in the rat. Neurosci Lett 180:285-289, 1994
    • (1994) Neurosci Lett , vol.180 , pp. 285-289
    • Martin, H.1    Warner, D.S.2    Todd, M.M.3
  • 24
    • 0028949633 scopus 로고
    • Glycine receptor antagonism. Effects of ACEA-1021 on the minimum alveolar concentration for halothane in the rat
    • McFarlane C, Warner DS, Nader A, et al: Glycine receptor antagonism. Effects of ACEA-1021 on the minimum alveolar concentration for halothane in the rat. Anesthesiology 82: 963-968, 1995
    • (1995) Anesthesiology , vol.82 , pp. 963-968
    • McFarlane, C.1    Warner, D.S.2    Nader, A.3
  • 25
    • 0025130511 scopus 로고
    • Ischemic brain damage in a model of acute subdural hematoma
    • Miller JD, Bullock R, Graham DI, et al: Ischemic brain damage in a model of acute subdural hematoma. Neurosurgery 27: 433-439, 1990
    • (1990) Neurosurgery , vol.27 , pp. 433-439
    • Miller, J.D.1    Bullock, R.2    Graham, D.I.3
  • 26
    • 0026531063 scopus 로고
    • Chemical monitoring of neurosurgical intensive care patients using intracerebral microdialysis
    • Persson L, Hillered L: Chemical monitoring of neurosurgical intensive care patients using intracerebral microdialysis. J Neurosurg 76:72-80, 1992
    • (1992) J Neurosurg , vol.76 , pp. 72-80
    • Persson, L.1    Hillered, L.2
  • 27
    • 0025090064 scopus 로고
    • Systematic studies on the effects of the NMDA receptor antagonist MK-801 on cerebral blood flow and responsivity, EEC, and blood-brain barrier following complete reversible cerebral ischemia
    • Stevens MK, Yaksh TL: Systematic studies on the effects of the NMDA receptor antagonist MK-801 on cerebral blood flow and responsivity, EEC, and blood-brain barrier following complete reversible cerebral ischemia. J Cereb Blood Flow Metab 10:77-88, 1990
    • (1990) J Cereb Blood Flow Metab , vol.10 , pp. 77-88
    • Stevens, M.K.1    Yaksh, T.L.2
  • 28
    • 0025334268 scopus 로고
    • Mechanistic distinctions between excitotoxic and acidotic hippocampal damage in an in vitro model of ischemia
    • Tombaugh GC, Sapolsky RM: Mechanistic distinctions between excitotoxic and acidotic hippocampal damage in an in vitro model of ischemia. J Cereb Blood Flow Metab 10: 527-535, 1990
    • (1990) J Cereb Blood Flow Metab , vol.10 , pp. 527-535
    • Tombaugh, G.C.1    Sapolsky, R.M.2
  • 29
    • 0029132006 scopus 로고
    • The effect of the glycine site-specific N-methyl-D-aspartate antagonist ACEA 1021 on ischemic brain damage caused by acute subdural hematoma in the rat
    • Tsuchida E, Bullock R: The effect of the glycine site-specific N-methyl-D-aspartate antagonist ACEA 1021 on ischemic brain damage caused by acute subdural hematoma in the rat. J Neurotrauma 12:279-288, 1995
    • (1995) J Neurotrauma , vol.12 , pp. 279-288
    • Tsuchida, E.1    Bullock, R.2
  • 30
    • 0026610369 scopus 로고
    • 3H-MK-801 (dizocilpine) in vivo uptake and in vitro binding after focal cerebral ischemia in the rat
    • 3H-MK-801 (dizocilpine) in vivo uptake and in vitro binding after focal cerebral ischemia in the rat. J Neurosurg 76:127-133, 1992
    • (1992) J Neurosurg , vol.76 , pp. 127-133
    • Wallace, M.C.1    Teasdale, G.M.2    McCulloch, J.3
  • 31
    • 0028834171 scopus 로고
    • In vivo models of cerebral ischemia: Effects of parenterally administered NMDA receptor glycine site antagonists
    • Warner DS, Martin H, Ludwig P, et al: In vivo models of cerebral ischemia: effects of parenterally administered NMDA receptor glycine site antagonists. J Cereb Blood Flow Metab 15: 188-196, 1995
    • (1995) J Cereb Blood Flow Metab , vol.15 , pp. 188-196
    • Warner, D.S.1    Martin, H.2    Ludwig, P.3
  • 32
    • 0025739645 scopus 로고
    • Regionally selective effects of NMDA receptor antagonists against ischemic brain damage in the gerbil
    • Warner MA, Neill KH, Nadler JV, et al: Regionally selective effects of NMDA receptor antagonists against ischemic brain damage in the gerbil. J Cereb Blood Flow Metab 11:600-610, 1991
    • (1991) J Cereb Blood Flow Metab , vol.11 , pp. 600-610
    • Warner, M.A.1    Neill, K.H.2    Nadler, J.V.3
  • 33
    • 0024511427 scopus 로고
    • Dynamic changes of excitatory amino acid receptors in the rat hippo-campus following transient cerebral ischemia
    • Westerberg E, Monaghan DT, Kalimo H, et al: Dynamic changes of excitatory amino acid receptors in the rat hippo-campus following transient cerebral ischemia. J Neurosci 9: 798-805, 1989
    • (1989) J Neurosci , vol.9 , pp. 798-805
    • Westerberg, E.1    Monaghan, D.T.2    Kalimo, H.3
  • 34
    • 0028916586 scopus 로고
    • In vitro pharmacology of ACEA-1021 and ACEA-1031: Systemically active quinoxalinediones with high affinity and selectivity for N-methyl-D-aspartate receptor glycine sites
    • Woodward RM, Huettner JE, Guastella J, et al: In vitro pharmacology of ACEA-1021 and ACEA-1031: systemically active quinoxalinediones with high affinity and selectivity for N-methyl-D-aspartate receptor glycine sites. Mol Pharmacol 47: 568-581, 1995
    • (1995) Mol Pharmacol , vol.47 , pp. 568-581
    • Woodward, R.M.1    Huettner, J.E.2    Guastella, J.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.