Molecular and functional properties of somatostatin receptor subtypes

Metabolism: Clinical and Experimental

Volumn 45, Issue SUPPL.1, 1996, Pages 12-13

  Liapakis, George ^a   Tallent, Melanie ^a   Reisine, Terry ^a  

^a UNIVERSITY OF PENNSYLVANIA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ADENYLATE CYCLASE; BIM 23027; CALCIUM CHANNEL; DEXTRO PHENYLALANYLPHENYLALANYLPHENYLALANYL DEXTRO TRYPTOPHYLLYSYLTHREONYLPHENYLALANYLTHREONINAMIDE; GUANINE NUCLEOTIDE BINDING PROTEIN; HYPOTHALAMUS RELEASE INHIBITING FACTOR; L 362855; OCTREOTIDE; PERTUSSIS TOXIN; RECEPTOR SUBTYPE; SEGLITIDE; SOMATOSTATIN RECEPTOR;

AMINO ACID SEQUENCE; ANIMAL CELL; ARTICLE; BINDING AFFINITY; BINDING SITE; CHO CELL; LIGAND BINDING; MOUSE; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR BINDING; RECEPTOR DOWN REGULATION; SITE DIRECTED MUTAGENESIS;

AMINO ACID SEQUENCE; ANIMALS; CALCIUM CHANNELS; GTP-BINDING PROTEINS; HUMANS; LIGANDS; RECEPTORS, SOMATOSTATIN;

EID: 0029786419     PISSN: 00260495     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0026-0495(96)90070-0     Document Type: Article

References (11)

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3. Raynor K, O'Carroll A-M, Kong H, et al: Characterisation of cloned somatostatin receptors SSTR-4 and SSTR-5. Mol Pharmacol 44:385-392, 1993
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7. Law S, Yasuda K, Bell GI, et al: Gia3 and Goa selectively associate with the cloned somatostatin receptor subtype SSTR2. J Biol Chem 268:10721-10727, 1993
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9. Law S, Zaina S, Sweet R, et al: Gial selectively couples the somatostatin receptor subtype SSTR-3 to adenylyl cyclase: Identification of the functional domains of this alpha subunit necessary for mediating somatostatin's inhibition of cAMP formation. Mol Pharmacol 45:587-590, 1994
10. O'Carroll A-M, Lolait S, Konig M, et al: Molecular cloning and expression of a pituitary somatostatin receptor with preferential affinity for somatostatin-28. Mol Pharmacol 42:939-946, 1992
11. 2+ current in the pituitary cell line AtT-20. Neuroscience 71:1073-1081, 1996