Benzylidene-substituted imidazo-thiazole-thiazine and -thiazepine derivatives: A new class of ligands for the benzodiazepine binding site of GABA(A) receptors

Scientia Pharmaceutica

Volumn 64, Issue 3-4, 1996, Pages 383-390

  Geis, Uli ^a   Kiec Kononowicz, Katarzyna ^b   Müller, Christa E ^a  

^a UNIVERSITY OF WÜRZBURG   (Germany)

^b JAGIELLONIAN UNIVERSITY MEDICAL COLLEGE   (Poland)

Author keywords

benzodiazepine; benzylidene 6,7 dihydro 5H imidazo 2,1 b 1,3 thiazin 3(2H) ones; GABA shift; GABA(A) receptor; structure activity relationship

Indexed keywords

4 AMINOBUTYRIC ACID RECEPTOR; BENZODIAZEPINE DERIVATIVE; BENZYLIDENE DERIVATIVE; DIAZEPAM; IMIDAZOLE DERIVATIVE; THIAZEPINE DERIVATIVE; THIAZINE DERIVATIVE;

ANIMAL TISSUE; ARTICLE; BRAIN CORTEX; CHEMICAL REACTION; CHEMICAL STRUCTURE; DRUG RECEPTOR BINDING; ISOTOPE LABELING; NONHUMAN; RAT; SYNTHESIS;

EID: 0029786024     PISSN: 00368709     EISSN: 22180532     Source Type: Journal    
DOI: None     Document Type: Article

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