메뉴 건너뛰기




Volumn 34, Issue 8, 1996, Pages 329-334

Zidovudine glucuronidation in human liver: Interindividual variability

Author keywords

Antivirals; Glucuronosyl transferase; Liver; Variability; Zidovudine

Indexed keywords

BILIRUBIN; GLUCURONIC ACID; GLUCURONOSYLTRANSFERASE; ZIDOVUDINE; ZIDOVUDINE GLUCURONIDE;

EID: 0029782873     PISSN: 09461965     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (26)

References (36)
  • 1
    • 0023680670 scopus 로고
    • Pharmacokinetic and bioavailability of zidovudine in humans
    • Blum MR, Liao SHT, Good SS, De Miranda P 1988 Pharmacokinetic and bioavailability of zidovudine in humans. Am J Med 85 (Suppl 2A): 189-194
    • (1988) Am J Med , vol.85 , Issue.SUPPL. 2A , pp. 189-194
    • Blum, M.R.1    Liao, S.H.T.2    Good, S.S.3    De Miranda, P.4
  • 2
    • 0028018821 scopus 로고
    • The influence of environmental and genetic factors on CYP2D6, CYP1A2 and UDP-glucuronosyltransferase in man using sparteine, caffeine and paracetamol as probes
    • Bock KW, Scherenk D, Foster A, Griese E-U, Morike K, Brockmeier D, Eichelbaum M 1994 The influence of environmental and genetic factors on CYP2D6, CYP1A2 and UDP-glucuronosyltransferase in man using sparteine, caffeine and paracetamol as probes. Pharmacogenetics 4: 209-218
    • (1994) Pharmacogenetics , vol.4 , pp. 209-218
    • Bock, K.W.1    Scherenk, D.2    Foster, A.3    Griese, E.-U.4    Morike, K.5    Brockmeier, D.6    Eichelbaum, M.7
  • 3
    • 0018145527 scopus 로고
    • Determination of microsomal UDP-glucuronosyltransferase in needle-biopsy specimens of human liver
    • Bock KW, Brunner G, Hoensch H, Huber E, Jostin D 1978 Determination of microsomal UDP-glucuronosyltransferase in needle-biopsy specimens of human liver. Eur J Clin Pharmacol 14: 367-373
    • (1978) Eur J Clin Pharmacol , vol.14 , pp. 367-373
    • Bock, K.W.1    Brunner, G.2    Hoensch, H.3    Huber, E.4    Jostin, D.5
  • 7
    • 0025944627 scopus 로고
    • Distribution of UDP-glucuronosyltransferase and its endogenous substrate uridine 5′-diphosphoglucuronic acid in human tissues
    • Cappiello M, Giuliani L, Pacifici GM 1991 Distribution of UDP-glucuronosyltransferase and its endogenous substrate uridine 5′-diphosphoglucuronic acid in human tissues. Eur J Clin Pharmacol 41: 345-350
    • (1991) Eur J Clin Pharmacol , vol.41 , pp. 345-350
    • Cappiello, M.1    Giuliani, L.2    Pacifici, G.M.3
  • 8
    • 0024505497 scopus 로고
    • A review of the pharmacokinetics of zidovudine in man
    • Cload PA 1989 A review of the pharmacokinetics of zidovudine in man. J Infection 18 (Suppl 1): 15-21
    • (1989) J Infection , vol.18 , Issue.1 SUPPL. , pp. 15-21
    • Cload, P.A.1
  • 9
    • 0025866909 scopus 로고
    • Modulation of 3′-azido-3′-deoxythymidine catabolism by probenecid and acetaminofen in freshly isolated rat hepatocytes
    • Cretton EM, Sommadossi J-P 1991 Modulation of 3′-azido-3′-deoxythymidine catabolism by probenecid and acetaminofen in freshly isolated rat hepatocytes. Biochem Pharmacol 42: 1475-1480
    • (1991) Biochem Pharmacol , vol.42 , pp. 1475-1480
    • Cretton, E.M.1    Sommadossi, J.-P.2
  • 10
    • 0025286491 scopus 로고
    • Glucuronidation of 3′-azido-3′-deoxythymidine by rat and human liver microsomes
    • Cretton EM, Waterhous DV, Bevan R, Somadossi JP 1990 Glucuronidation of 3′-azido-3′-deoxythymidine by rat and human liver microsomes. Drug Metab Dispos 18: 369-372
    • (1990) Drug Metab Dispos , vol.18 , pp. 369-372
    • Cretton, E.M.1    Waterhous, D.V.2    Bevan, R.3    Somadossi, J.P.4
  • 12
    • 0027279427 scopus 로고
    • Pharmacokinetics of zidovudine after the initial single dose and during chronic-dose therapy in HIV-infected patients
    • Gallicano K, Sahai J, Ormsby E, Cameron DW, Pakuts A, McGilveray I 1993 Pharmacokinetics of zidovudine after the initial single dose and during chronic-dose therapy in HIV-infected patients. Br J Clin Pharmacol 36: 128-131
    • (1993) Br J Clin Pharmacol , vol.36 , pp. 128-131
    • Gallicano, K.1    Sahai, J.2    Ormsby, E.3    Cameron, D.W.4    Pakuts, A.5    McGilveray, I.6
  • 15
    • 0024997543 scopus 로고
    • Phenobarbital inducible UDP-glucuronosyltransferase is responsible for glucuronidation of 3′-azido-3′-deoxythymidine: Characterization of the enzyme in human and rat liver microsomes
    • Haumont M, Magdalou J, Lafaurie C, Ziegler J-M, Siest G, Colin J-N 1990 Phenobarbital inducible UDP-glucuronosyltransferase is responsible for glucuronidation of 3′-azido-3′-deoxythymidine: Characterization of the enzyme in human and rat liver microsomes. Arch Biochem Biophys 281: 264-270
    • (1990) Arch Biochem Biophys , vol.281 , pp. 264-270
    • Haumont, M.1    Magdalou, J.2    Lafaurie, C.3    Ziegler, J.-M.4    Siest, G.5    Colin, J.-N.6
  • 20
    • 0026586239 scopus 로고
    • In vitro inhibition studies of the glucuronidation of 3′-azido-3′-deoxythymidine catalysed by human liver UDP-glucuronosyl transferase
    • Macleod R, Eagling VA, Sim SM, Back DJ 1992 In vitro inhibition studies of the glucuronidation of 3′-azido-3′-deoxythymidine catalysed by human liver UDP-glucuronosyl transferase. Biochem Pharmacol 43: 382-386
    • (1992) Biochem Pharmacol , vol.43 , pp. 382-386
    • Macleod, R.1    Eagling, V.A.2    Sim, S.M.3    Back, D.J.4
  • 21
    • 0028960240 scopus 로고
    • Comparative metabolism of 3′-azido-3′-deoxythymidine in culturated hepatocytes from rats, dog, monkey and humans
    • Nicolas F, De Sousa G, Thomas P, Placidi M, Lorenzon G, Rahmani R 1995 Comparative metabolism of 3′-azido-3′-deoxythymidine in culturated hepatocytes from rats, dog, monkey and humans. Drug Metab Dis 23: 308-313
    • (1995) Drug Metab Dis , vol.23 , pp. 308-313
    • Nicolas, F.1    De Sousa, G.2    Thomas, P.3    Placidi, M.4    Lorenzon, G.5    Rahmani, R.6
  • 22
    • 9444292854 scopus 로고
    • Infectious disorders
    • Melmon KL, Morelli HF, Hoffman BB, Nierenberg DW (eds) McGraw-Hill, New York
    • O'Hanley PD, Tam JY, Holodniy M 1992 Infectious disorders. In: Melmon KL, Morelli HF, Hoffman BB, Nierenberg DW (eds) Clinical Pharmacology. 3rd edn., McGraw-Hill, New York, p 687
    • (1992) Clinical Pharmacology. 3rd Edn. , pp. 687
    • O'Hanley, P.D.1    Tam, J.Y.2    Holodniy, M.3
  • 23
    • 0025008823 scopus 로고
    • Development of the glucuronosyltransferase and sulphotransferase towards 2-naphthol in human fetus
    • Pacifici GM, Franchi M, Giuliani L, Rane A 1990a Development of the glucuronosyltransferase and sulphotransferase towards 2-naphthol in human fetus. Dev Pharmacol Ther 14: 108-114
    • (1990) Dev Pharmacol Ther , vol.14 , pp. 108-114
    • Pacifici, G.M.1    Franchi, M.2    Giuliani, L.3    Rane, A.4
  • 26
    • 0025871397 scopus 로고
    • Glucuronidation of 3′-azido-3′-deoxythymidine catalysed by human liver UDP-glucuronosyltransferase
    • Resetar A, Minick D, Spector T 1991 Glucuronidation of 3′-azido-3′-deoxythymidine catalysed by human liver UDP-glucuronosyltransferase. Biochem Pharmacol 42: 559-568
    • (1991) Biochem Pharmacol , vol.42 , pp. 559-568
    • Resetar, A.1    Minick, D.2    Spector, T.3
  • 27
    • 0024577652 scopus 로고
    • Glucuronidation of 3′-azido-3′-deoxythymidine: Human and rat enzyme specificity
    • Resetar A, Spector T 1989 Glucuronidation of 3′-azido-3′-deoxythymidine: human and rat enzyme specificity. Biochem Pharmacol 38: 1389-1393
    • (1989) Biochem Pharmacol , vol.38 , pp. 1389-1393
    • Resetar, A.1    Spector, T.2
  • 28
    • 0027364453 scopus 로고
    • Zidovudine response relationships in early human immunodeficiency virus infection
    • Sale M, Sheiner LB, Volberding P, Blaschke TF 1993 Zidovudine response relationships in early human immunodeficiency virus infection. Clin Pharmacol Ther 54: 556-566
    • (1993) Clin Pharmacol Ther , vol.54 , pp. 556-566
    • Sale, M.1    Sheiner, L.B.2    Volberding, P.3    Blaschke, T.F.4
  • 29
    • 0025850455 scopus 로고
    • The effect of various drugs on the glucuronidation of zidovudine azidothymidine; AZT by human liver microsomes
    • Sim SM, Back DJ, Brekenridge AM 1991 The effect of various drugs on the glucuronidation of zidovudine azidothymidine; AZT by human liver microsomes. Br J Clin Pharmacol 32: 17-21
    • (1991) Br J Clin Pharmacol , vol.32 , pp. 17-21
    • Sim, S.M.1    Back, D.J.2    Brekenridge, A.M.3
  • 30
    • 0025831505 scopus 로고
    • Interindividual variability in the glucuronidation and sulphation of ethinyloestradiol in human liver
    • Temellini A, Giuliani L, Pacifici GM 1991 Interindividual variability in the glucuronidation and sulphation of ethinyloestradiol in human liver. Br J Clin Pharmacol 31: 661-664
    • (1991) Br J Clin Pharmacol , vol.31 , pp. 661-664
    • Temellini, A.1    Giuliani, L.2    Pacifici, G.M.3
  • 31
    • 0024419214 scopus 로고
    • UDP-glucuronosyltransferases in the metabolic disposition of xenobiotics
    • Tephly TR, Townsend M, Green M 1989 UDP-glucuronosyltransferases in the metabolic disposition of xenobiotics. Drug Metab Dispos 20: 689-695
    • (1989) Drug Metab Dispos , vol.20 , pp. 689-695
    • Tephly, T.R.1    Townsend, M.2    Green, M.3
  • 32
    • 9444268674 scopus 로고
    • Topology and regulation in sealed native microsomes from rat liver
    • Van Roy P, Heirwegh KPM 1968 Topology and regulation in sealed native microsomes from rat liver. Arch Biochem Biophys 263: 216-225
    • (1968) Arch Biochem Biophys , vol.263 , pp. 216-225
    • Van Roy, P.1    Heirwegh, K.P.M.2
  • 34
    • 0014578362 scopus 로고
    • A rapid microdiazo technique for measuring total bilirubin
    • Winsten S, Cehelyk B 1969 A rapid microdiazo technique for measuring total bilirubin. Clin Chim Acta 25: 441-446
    • (1969) Clin Chim Acta , vol.25 , pp. 441-446
    • Winsten, S.1    Cehelyk, B.2
  • 35
    • 0024436217 scopus 로고
    • Clinical pharmacology of 3′-azido-2′,3′-dideoxythymidine zidovudine and related dideoxynucleosides
    • Yarchoan R, Mitsuya H, Myers CE, Broder S 1989 Clinical pharmacology of 3′-azido-2′,3′-dideoxythymidine zidovudine and related dideoxynucleosides. N Engl J Med 321: 726-738
    • (1989) N Engl J Med , vol.321 , pp. 726-738
    • Yarchoan, R.1    Mitsuya, H.2    Myers, C.E.3    Broder, S.4
  • 36
    • 0024355675 scopus 로고
    • Interindividual and interethnic differences in the demethylation and glucuronidation of codeine
    • Yue QY, Svensson J-O, Alam C, Sjoqvist F, Sawe J 1989 Interindividual and interethnic differences in the demethylation and glucuronidation of codeine. Br J Clin Pharmacol 28: 629-637
    • (1989) Br J Clin Pharmacol , vol.28 , pp. 629-637
    • Yue, Q.Y.1    Svensson, J.-O.2    Alam, C.3    Sjoqvist, F.4    Sawe, J.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.