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Volumn 13, Issue 7, 1996, Pages 1078-1082

Suitability of enalapril as a probe of the dipeptide transporter system: In vitro and in vivo studies

Author keywords

Absorption; Caco 2; Dogs; Enalapril; rats

Indexed keywords

AMOXICILLIN; BETA LACTAM ANTIBIOTIC; CEFACLOR; CEFALEXIN; CEFAZOLIN; CEFOXITIN; CEFRADINE; CERANAPRIL; DIPEPTIDYL CARBOXYPEPTIDASE INHIBITOR; ENALAPRIL; GLYCYLPROLINE;

EID: 0029781995     PISSN: 07248741     EISSN: None     Source Type: Journal    
DOI: 10.1023/A:1016071027177     Document Type: Article
Times cited : (20)

References (17)
  • 1
    • 0024891564 scopus 로고
    • Passive and carrier-mediated intestinal absorption components of two angiotensin converting enzyme (ACE) inhibitor prodrugs in rats: Enalapril and fosinopril
    • D. I. Friedman and G. L. Amidon. Passive and carrier-mediated intestinal absorption components of two angiotensin converting enzyme (ACE) inhibitor prodrugs in rats: enalapril and fosinopril. Pharm. Res. 6:1043-1047 (1989).
    • (1989) Pharm. Res. , vol.6 , pp. 1043-1047
    • Friedman, D.I.1    Amidon, G.L.2
  • 2
    • 9344266236 scopus 로고
    • Noncompetitive inhibition of intestinal cephradine uptake by enalapril: An enalapril specific inhibitory binding site on the peptide carrier
    • H. Yuasa, G. L. Amidon, and D. Fleisher. Noncompetitive inhibition of intestinal cephradine uptake by enalapril: An enalapril specific inhibitory binding site on the peptide carrier, Pharm. Res. 8:(10), S-221 (1991).
    • (1991) Pharm. Res. , vol.8 , Issue.10
    • Yuasa, H.1    Amidon, G.L.2    Fleisher, D.3
  • 3
    • 9344224448 scopus 로고
    • Transport characterization of the ACE inhibitor enalapril in rabbit intestinal brush border membrane vesicles
    • S. Yee, and G. L. Amidon. Transport characterization of the ACE inhibitor enalapril in rabbit intestinal brush border membrane vesicles, Pharm. Res. 8:(10), S-198 (1991).
    • (1991) Pharm. Res. , vol.8 , Issue.10
    • Yee, S.1    Amidon, G.L.2
  • 4
    • 0028905095 scopus 로고
    • Angiotensin-converting enzyme (ACE) inhibitor transport in human intestinal epithelial (Caco-2) cells
    • D. T. Thwaites, M. Cavet, B. H. Hirst, and N. Simmons. Angiotensin-converting enzyme (ACE) inhibitor transport in human intestinal epithelial (Caco-2) cells, Brit. J. Pharmacol. 114:981-986 (1995).
    • (1995) Brit. J. Pharmacol. , vol.114 , pp. 981-986
    • Thwaites, D.T.1    Cavet, M.2    Hirst, B.H.3    Simmons, N.4
  • 5
    • 0029991885 scopus 로고    scopus 로고
    • Distribution of the dipeptide transporter system along the gastrointestinal tract of rats based on absorption of a stable and specific probe, SQ-29852
    • A. M. Marino, S. Chong, S. A. Dando, K. J. Kripalani, M. S. Bathala, and R. A. Morrison. Distribution of the dipeptide transporter system along the gastrointestinal tract of rats based on absorption of a stable and specific probe, SQ-29852, J. Pharm. Sci. 85:282-286 (1996).
    • (1996) J. Pharm. Sci. , vol.85 , pp. 282-286
    • Marino, A.M.1    Chong, S.2    Dando, S.A.3    Kripalani, K.J.4    Bathala, M.S.5    Morrison, R.A.6
  • 6
    • 0000566243 scopus 로고
    • Systematic evaluation of the structural requirements for the intestinal dipeptide transporter system
    • V. A. Moore, S. Chong, S. A. Dando, W. Lau, W. J. Irwin, P. Timmins, and R. A. Morrison. Systematic evaluation of the structural requirements for the intestinal dipeptide transporter system, Pharm. Res. 12:(9) (suppl), S-301 (1995).
    • (1995) Pharm. Res. , vol.12 , Issue.9 SUPPL.
    • Moore, V.A.1    Chong, S.2    Dando, S.A.3    Lau, W.4    Irwin, W.J.5    Timmins, P.6    Morrison, R.A.7
  • 7
    • 0025046860 scopus 로고
    • Uptake of the cephalosporin, cephalexin, by a dipeptide transport carrier in the human intestinal cell line, Caco2
    • A. H. Dantzig and L. Bergin. Uptake of the cephalosporin, cephalexin, by a dipeptide transport carrier in the human intestinal cell line, Caco2, Biochemica et Biophysica Acta 1027:211-217 (1990).
    • (1990) Biochemica et Biophysica Acta , vol.1027 , pp. 211-217
    • Dantzig, A.H.1    Bergin, L.2
  • 8
    • 0028345208 scopus 로고
    • Transport mechanism responsible for the absorption of loracarbef, cefixime, and cefuroxime axetil into human intestinal Caco-2 cells
    • A. H. Dantzig, D. C. Duckworth, and L. B. Tabas. Transport mechanism responsible for the absorption of loracarbef, cefixime, and cefuroxime axetil into human intestinal Caco-2 cells, Biochim. Biophys. Acta. 1191:7-13 (1994).
    • (1994) Biochim. Biophys. Acta. , vol.1191 , pp. 7-13
    • Dantzig, A.H.1    Duckworth, D.C.2    Tabas, L.B.3
  • 9
    • 0024909165 scopus 로고
    • Intestinal absorption mechanism of dipeptide angiotensin converting enzyme inhibitors of the lysyl-proline type: Lisinopril and SQ 29,852
    • D. I. Friedman and G. L. Amidon, Intestinal absorption mechanism of dipeptide angiotensin converting enzyme inhibitors of the lysyl-proline type: lisinopril and SQ 29,852, J. Pharm. Sci. 78:995-998 (1989).
    • (1989) J. Pharm. Sci. , vol.78 , pp. 995-998
    • Friedman, D.I.1    Amidon, G.L.2
  • 10
    • 0027987417 scopus 로고
    • Mechanism and kinetics of transcellular transport of a new beta-lactam antibiotic across an intestinal epithelial membrane model system (Caco-2)
    • M. Hu, J. Chen, Y. Zhu, A. H. Dantzig, R. E. Stratford, and M. T. Kuhfeld. Mechanism and kinetics of transcellular transport of a new beta-lactam antibiotic across an intestinal epithelial membrane model system (Caco-2), Pharm. Res. 11:(10), 1405-13 (1994).
    • (1994) Pharm. Res. , vol.11 , Issue.10 , pp. 1405-1413
    • Hu, M.1    Chen, J.2    Zhu, Y.3    Dantzig, A.H.4    Stratford, R.E.5    Kuhfeld, M.T.6
  • 11
    • 0000710670 scopus 로고
    • Uptake and transport of an ACE-inhibitor (SQ-29852) by Caco-2 cells
    • P. L. Nicklin, W. J. Irwin, and P. Timmins. Uptake and transport of an ACE-inhibitor (SQ-29852) by Caco-2 cells, J. Pharm. Pharmacol. 44:1091 (1992).
    • (1992) J. Pharm. Pharmacol. , vol.44 , pp. 1091
    • Nicklin, P.L.1    Irwin, W.J.2    Timmins, P.3
  • 14
    • 0025143832 scopus 로고
    • Contribution of passive and transport mechanisms to the intestinal absorption of β-lactam antibiotics
    • M. Sugawara, H. Saitoh, K. Iseki, K. Miyazaki, and T. Arita. Contribution of passive and transport mechanisms to the intestinal absorption of β-lactam antibiotics, J. Pharm. Pharmacol. 42:314-318 (1989).
    • (1989) J. Pharm. Pharmacol. , vol.42 , pp. 314-318
    • Sugawara, M.1    Saitoh, H.2    Iseki, K.3    Miyazaki, K.4    Arita, T.5
  • 15
    • 0011880372 scopus 로고
    • In vitro uptake of SQ-29852 by everted rat intestinal rings
    • B. H. Stewart, S. A. Dando, and R. A. Morrison. In vitro uptake of SQ-29852 by everted rat intestinal rings, Pharm. Res. 7:(9) (suppl), S-156 (1990).
    • (1990) Pharm. Res. , vol.7 , Issue.9 SUPPL.
    • Stewart, B.H.1    Dando, S.A.2    Morrison, R.A.3
  • 16
    • 0029939330 scopus 로고    scopus 로고
    • In vitro permeability through Caco-2 cells is not quantitatively predictive of in vivo absorption for drugs absorbed via the dipeptide transporter system
    • S. Chong, S. A. Dando, and R. A. Morrison. In vitro permeability through Caco-2 cells is not quantitatively predictive of in vivo absorption for drugs absorbed via the dipeptide transporter system, Pharm. Res. 13:(1), (1996).
    • (1996) Pharm. Res. , vol.13 , Issue.1
    • Chong, S.1    Dando, S.A.2    Morrison, R.A.3
  • 17
    • 4244052183 scopus 로고
    • Inhibition of uptake by the oligopeptide transporter does not correlate with transepithelial transport
    • K. Tamura, P. K. Bhatnagar, J. S. Takata, C.-P. Lee, P. L. Smith, and R. T. Borchardt. Inhibition of uptake by the oligopeptide transporter does not correlate with transepithelial transport, Pharm. Res. 12:(9) (suppl), S-302 (1995).
    • (1995) Pharm. Res. , vol.12 , Issue.9 SUPPL.
    • Tamura, K.1    Bhatnagar, P.K.2    Takata, J.S.3    Lee, C.-P.4    Smith, P.L.5    Borchardt, R.T.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.