Effects of permeation enhancers on the transport of a peptidomimetic thrombin inhibitor (CRC 220) in a human intestinal cell line (Caco-2)

Pharmaceutical Research

Volumn 13, Issue 8, 1996, Pages 1219-1227

  Werner, Ute ^a   Kissel, Thomas ^a   Reers, Martin ^b  

^a PHILIPPS UNIVERSITY MARBURG   (Germany)

^b Behringwerke AG   (Germany)

Author keywords

Cell monolayers; Cytotoxicity; Micellar systems; Peptide transport; Permeation enhancers

Indexed keywords

CHOLESTEROL; CRC 220; LACTATE DEHYDROGENASE; OLEIC ACID; PHOSPHATIDYLCHOLINE; POLYOXYETHYLENE DERIVATIVE; TAUROCHOLIC ACID; THROMBIN INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; CELL MEMBRANE PERMEABILITY; CELL VIABILITY; CONTROLLED STUDY; CYTOCHEMISTRY; DRUG TRANSPORT; ELECTRIC RESISTANCE; HUMAN; HUMAN CELL; INTESTINE CELL; MICELLE; PRIORITY JOURNAL;

ANTITHROMBINS; BIOLOGICAL TRANSPORT; CACO-2 CELLS; DIPEPTIDES; EPITHELIUM; HUMANS; MEMBRANE POTENTIALS; MICELLES; PERMEABILITY; PHOSPHOLIPIDS; PIPERIDINES;

EID: 0029775162     PISSN: 07248741     EISSN: None     Source Type: Journal    
DOI: 10.1023/A:1016020505313     Document Type: Article

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