Modulation of skin drug penetration;Modulation der Wirkstoffpenetration in die Haut

Pharmazie

Volumn 51, Issue 9, 1996, Pages 619-637

  Kalbitz, J ^a   Neubert, R ^a,b   Wohlrab, W ^a  

^a MARTIN LUTHER UNIVERSITY HALLE WITTENBERG   (Germany)

^b Inst F Pharmazeut Technol B   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

ERYTHROMYCIN; GRISEOFULVIN; HYDROCORTISONE; PENETRATION ENHANCING AGENT;

DRUG ABSORPTION; DRUG DIFFUSION; DRUG PENETRATION; DRUG UPTAKE; HUMAN; HUMAN TISSUE; REVIEW; SKIN PENETRATION; SKIN PERMEABILITY; STRATUM CORNEUM; TOPICAL DRUG ADMINISTRATION;

ADMINISTRATION, CUTANEOUS; ADMINISTRATION, TOPICAL; ANIMALS; HUMANS; SKIN ABSORPTION;

EID: 0029744785     PISSN: 00317144     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Review

References (124)

1. Lambert, W. J.; Kudlar, R. J.; Hollard, J. M.; Curry, J. T.: Int. J. Pharm. 45, 181 (1993).
2. Pfister, W. R.; Dean, S.; Hsieh, S. T.: Pharm. Tech. 8, 132 (1990)
3. Nightingale, J.; Kurihara-Bergstrom, T.; Mirley, C.; Signor, C.; DeNoble, L.: Hcl. Proc. Int. Symp. Control. Rel. Bioact. Mater. 19, 246 (1992)
4. Chien, Y. W.; Xu, H.; Chiang, C. C.; Hung, Y. C.: Pharm. Res. 5, 103 (1988)
5. Devaux, P. F.; Seigneuret, M.: Biochim. Biophys. Acta 822, 463 (1985)
6. Stoughton, R. B.: Arch. Dermatol. 91, 657 (1965)
7. Kligman, A. M.: J. Am. Med. Assoc. 193, 796 (1965)
8. Mallory, S. B.; Lehman, P. A.; Vanderpool, D. R.; Franz, T. J.: Pediatr. Dermatol. 10, 370 (1993)
9. Barry, B. W.: J. Control. Rel. 6, 85 (1987)
10. Sekura, D. L.; Scala, J.: Adv. Biol. Skin 12, 257 (1972)
11. McCullough, J. L.; Snyder, D. S.; Weinstein, G. D.; Friedland, A.; Stein, B.: J. Invest. Dermatol. 66, 103 (1976)
12. Chowhan, Z. T.; Pritchard, R.: J. Pharm. Sci. 67, 1272 (1978)
13. Touitou, E.: Int. J. Pharm. 43, 1 (1988)
14. Goodman, M.; Barry, B. W.: J. Invest. Dermatol. 91, 323 (1988)
15. Touitou, E.; Abed, L.: Int. J. Pharm. 27, 89 (1985)
16. Wiechers, J. W.; De Zeeuw, R. A.; in: Honan, M. (ed.): Drug Design and Delivery, Vol. 6, Harwood Academic Publishers, London, 1990
17. Hadcraft, J.; Williams, D. G.; Allah, G. in: Walters, K. A.; Hadcraft, J. (eds.): Pharmaceutical Skin Penetration Enhancement, Marcel Dekker, New York, Basel 1993
18. Barry, B. W.; Bennett, S. L.: J. Pharm. Pharmacol. 39, 535 (1987)
19. Okamoto, H.; Hashida, M.; Sezaki, H.: J. Pharm. Sci. 77, 418 (1988)
20. Allan, G. in: Smith, E. W.; Maibach, H. I. (eds.): Percutaneous Penetration Enhancers, p. 129 CRC-Press, Boca Raton, New York, London, Tokyo 1995
21. Wester, R. C.; Maibach, H. I. in: Smith, E. W.; Maibach, H. I. (eds.): Percutaneous Penetration Enhancers, p. 159 CRC-Press, Boca Raton, New York, London, Tokyo 1995
22. Wiechers, J. W. in: Smith, E. W.; Maibach, H. I. (ed.): Percutaneous Penetration Enhancers, p. 165 CRC-Press, Boca Raton, New York, London, Tokyo 1995
23. Mirejovsky, D.; Takruri, H.: J. Pharm. Sci. 75, 1089 (1986)
24. Okamoto, H.; Hashida, M.; Sezaki, H.: J. Pharm. Sci. 77, 418 (1988)
25. Bouwstra, J. A.; Gooris, G. S.; Brussee, J.; Salomons de-Vries, M. A.; Bras, W.: Int. J. Pharm. 79, 141 (1992)
26. Bouwstra, J. A.; DeVries, M. A.; Bras, W.; Brussee, J.; Gooris, G. S.: Proc. Int. Sym. Control. Rel. Bioact. Mater. 17, 33 (1990)
27. Akitoshi, Y.; Takayama, K.; Machida, Y.; Nagai, T.: Drug Des. Deliv. 2, 239 (1988)
28. Michniak, B. B.; Player, M. R.; Chapman Jr.; J. M.; Sowell, J. W.: Int. J. Pharm. 91, 85 (1993)
29. Michniak, B. B.; Player, M. R.; Fuhrman, L. C.; Christensen, C. A.; Chapman Jr., J. M.; Sowell Sr., J. W.: Int. J. Pharm. 94, 203 (1993)
30. Minaskanian, G.; Peck, J. V. U. S. Patent 5, 142044, 1992
31. Bonina, F. P.; Montenegro, L.; De Capraris, P.; Bousquet, E.; Tirendi, S.; Int. J. Pharm. 77, 21 (1991)
32. Sasaki, H.; Kojima, M.; Mori, Y.; Nakamura, J.; Shibasaki, J.: Int. J. Pharm. 44, 15 (1988)
33. Resh, W.; Stoughton, R. B.: Arch. Dermatol. 112, 182 (1976)
34. Bonina, F. P.; Montenegro, L.: Int. J. Pharm. 82, 171 (1992)
35. Santus, G. C.; Baker, R. W.: J. Control. Rel. 25, 1 (1993)
36. Yano, T.; Higo, N.; Fukuda, K.; Tsuji, M.; Noda, K.; Otagiri, M.: J. Pharm. Pharmacol. 45, 775 (1993)
37. Lambert, W. J.; Kudla, R. J.; Holland, J. M.; Curry, J. T.: Int. J. Pharm. 95, 181 (1991)
38. Hoelgaard, A.; Mollgaard, B.; Baker, E.: Int. J. Pharm. 43, 233 (1988)
39. Sasaki, H.; Kojima, M.; Nakamura, J.; Shibasaki, J.: J. Pharm. Pharmacol. 42, 196 (1990)
40. Barry, B. W.: J Control. Rel. 6, 85 (1987)
41. Ponec, M.; Haverkort, M.; Soei, Y. L.; Kempenaar, J.; Brussee, J.; Bodde, H.: J. Pharm. Sci. 78, 738 (1989)
42. Feldman, R.; Maibach, H. I.: Arch. Dermatol. 109, 58 (1974)
43. Kim, C. K.; Kim, J. J.; Chi, S. C.; Shim, C. K.: Int. J. Pharm. 99, 109 (1993)
44. Wong, O.; Huntington, J.; Konishi, R.; Rytting, J. H.; Higuchi, T.: J. Pharm. Sci. 77, 967 (1988)
45. Wong, O.; Rytting, J. H. in: Smith, E. W.; Maibach, H. I. (eds.): Percutaneous Penetration Enhancers, p. 297, CRC Press, Boca Raton, New York, London, Tokyo 1995
46. Wongpayapkul, L.; Chow, D.: Paper PDD7053, APPS 6th Annu. Meet. Washington, D. C., 1991
47. Wong, O.; Huntington, J.; Nishihata, T.; Rytting, J. H.: Pharm. Res. 6, 286 (1989)
48. Büyüktimkin, S.; Büyüktimkin, N.; Rytting, J. H.: Pharm. Res. 10, 1632 (1993)
49. Büyüktimkin, N.; Büyüktimkin, S.; Rytting, J. H.: Paper PDD 7050, AAPS 6th Annu. Meet. Washington, D.C., 1991
50. Hirvonen, J., Rajala, R.; Vihervaara, P.; Laine, E.; Paronen, P.; Urtti, A.: Eur. J. Pharm. Biopharm., in press
51. Büyüktimkin, S.; Büyüktimkin, N.; Rytting, R. H.: Paper PDD 7266, AAPS 8th Annu. Meet. Orlando, FL, 1993
52. Ritschel, W. A.; Sprockel, O. L.: Drugs Today 24, 613 (1988)
53. Barry, B. W. in: Barry, B. W. (ed.): Dermatological Formulations Marcel Dekker Inc., New York, Basel 1983
54. Bendas, B.; Neubert, R.; Wohlrab, W. in: Smith, E. W.; Maibach, H. I. (ed.): Percutaneous Penetration Enhancers, p. 61, CRC-Press, Boca Raton, New York, London, Tokyo 1995
55. Bouwstra, J. A.; de Vries, T. A.; Goovis, G. S.; Bras, W.; Brussel, J.; Ponec, T.: J. Control. Rel. 15, 209 (1991)
56. Takeuchi, Y.; Yasukawa, H.; Yamaoka, Y.; Kato, Y.; Morimoto, Y.; Fukumori, Y.; Fukuda, T.: Chem. Pharm. Bull. 40, 1887 (1992)
57. Hoogsraate, A. J.; Verhoef, J.; Brussel, J.; Ijzerman, A. P.; Spies, F.; Boddé, H. E.: Int. J. Pharm. 76, 37 (1991)
58. Bettley, F. R.; Donoghue, E.: Nature 17, 185 (1960)
59. Bettley, F. R.; Br. J. Dermatol. 75, 113 (1963)
60. Kushla, G. P.; Zatz, J. L.; Mills Jr., O. H.; Berger, R. S.: J. Pharm. Sci. 82, 118 (1993)
61. Scheuplein, R.; Ross, L.: J. Soc. Cosmet. Chem. 21, 853 (1970)
62. Takahashi, M.; Aizawa, M.; Miyazawa, K.; Machida, Y.: J. Soc. Cosmet. Chem. 38, 21 (1987)
63. Ridout, G.; Hinz, R. S.; Hostynek, J. J.; Reddy, A. K.; Wiersema, R. J.; Hodson, C. D.; Lorence, C. R.; Guy, R. H.: Fund. Appl. Toxicol. 16, 41 (1991)
64. Prottey, C.; Ferguson, T.: J. Soc. Cosmet. Chem. 26, 29 (1975)
65. Cappel, M. J.; Kreuter, J.: Int. J. Pharm. 69, 143 (1991)
66. Shen, W. W.; Danti, A. G.; Bruscato, F. N.: J. Pharm. Sci. 65, 1780 (1976)
67. Nishiyama, T.; Iwata, Y.; Nakajima, K.; Mitsui, T.: J. Soc. Cosmet. Chem. 34, 263 (1983)
68. Chiang, C. H.; Lai, J. S.; Yang, K. H.: Drug Dev. Ind. Pharm. 17, 91 (1991)
69. Ogiso, T.; Iwaki, M.; Yoneda, I.; Horinouchi, M.; Yamashita, K.: Chem. Pharm. Bull. 39, 449 (1991)
70. Yamahara, J.; Kashiwa, H.; Kishi, K.; Fujimura, H.: Chem. Pharm. Bull. 37, 855 (1989)
71. Williams, A. C.; Barry, B. W.: Int. J. Pharm. 57, R7 (1989)
72. Williams, A. C.; Barry, B. W.: Pharm. Res. 8, 17 (1991)
73. Okabe, H.; Takayama, K.; Ogura, A.; Nagai, T.: Drugs Des. Deliv. 4, 313 (1989)
74. Williams, A. C.; Barry, B. W.: Int. J. Pharm. 74, 157 (1991)
75. Cornwell, P. A.; Barry, B. W.: Int. J. Pharm. 94, 189 (1993)
76. Bettley, F. R.: Br. J. Dermatol. 73, 448 (1961)
77. Bond, J. R.; Barry, B. W.; J. Invest. Dermatol. 90, 810 (1988)
78. Aungst, B. J.; Blake, J. A.; Hussein, M. A.: Pharm. Res. 7, 712 (1990)
79. Aungst, B. J.; Rogers, N. J.; Shefter, E.: Int. J. Pharm. 33, 225 (1986)
80. Ogsio, T.; Shintani, M.: J. Pharm. Sci. 79, 1065 (1990)
81. Komata, Y.; Inaoka, M.; Kaneko, A.; Fujie, T.: J. Pharm. Sci. 81, 744 (1992)
82. Aungst, B. J.: Pharm. Res. 6, 244 (1989)
83. Ongpipattanakul, B.; Burnette, R. R.; Potts, R. O.; Francoeur, M. L.: Pharm. Res. 8, 350 (1991)
84. Arima, H.; Adachi, H.; Irie, T.; Uekama, K,; Pitha, J.: Pharm. Res., 7, 1152 (1990)
85. Okamoto, H.; Komatsu, H.; Hashida, M.; Sezaki, H.: Int. J. Pharm. 30, 35 (1986)
86. Uekama, K.; Adachi, H.; Irie, T.; Yano, T.; Saita, M.; Noda, K.: J. Pharm. Pharmacol. 44, 119 (1992)
87. Adachi, H.; Irie, T.; Uekama, K.; Manako, T.; Yano, T.; Saita, M.: Eur. J. Pharm. Sci. 1, 117 (1993)
88. Vassoille, C., Falson-Rieg, F.: Prediction of Percutaneous Penetration 4a, C39 (1995)
89. Falson-Rieg, F.; Lafforgue, C.: Prediction of Percutaneous Penetration 4a, C40 (1995)
90. Toulon, A.; Besnard, M.; Leclerc, B.; Weingarten, C.; Salin-Drouin, D.; Courraze, G.: S.T.P. Pharma Sci. 1, 76 (1991)
91. Freeman, D. J.; Sheth, N. V.; Spruance, S. P.: Antimicrob. Agents Chemother. 29, 730 (1986)
92. Creasey, N. H.; Battensby, J.; Fletcher, J. A.: Curr. Probl. Dermatol. 7, 95 (1978)
93. Schneider, I.-M.; Dobner, B.; Neubert, R.; Wohlrab, W.: J. Pharm. Pharmacol., in press
94. Matschiner, S.; Neubert, R.; Wohlrab, W. in: Smith. E. W.; Maibach, H. I. (eds.): Percutaneous penetration enhancers, p. 407, CRC Press, Boca Raton, New York, London, Tokyo 1995
95. Davies, S. S.; Kinkel, K. F. M.; Olejnik, O.; Tomlinson, E.: J. Pharm. Pharmacol. 3, 104 (1981)
96. Chen, C. R.; Zatz, J. L.; Reilly, E.: Drug Dev. Ind. Pharm. 19, 1265 (1993)
97. Tan, E. L.; Liu, J. C.; Chien, W.: Pharm. Res. 6, S-171 (1989)
98. Young, C. S.; Shim, C. K.; Lee, M. H.; Kim, S. K.: Int. J. Pharm. 45, 59 (1988)
99. Green, P. G.; Guy, R. H.; Hadgraft, J.: Int. J. Pharm. 48, 103 (1988)
100. Röding, J.; Ghyczy, M.: Seifen, Oele, Fette, Wachse 10, 372 (1991)
101. Juninger, H. E.; Hofland, H. E.; Bouwstra, J. A.: Cosmet. Toilet. 106, 45 (1991)
102. Egbaria, K.; Weiner, N. in: Braun-Falco, O.; Korting, H. C.; Maibach, H. I. (eds.): Liposome Dermatics, p. 172, Springer-Verlag, Heidelberg 1992
103. Mezei, M.; Gulasekharam, V.: Life Sci. 26, 1473 (1980)
104. Lieb, L. M.; Ramachandran, C.; Weiner, N.; in: Braun-Falco, O.; Korting, H. C.; Maibach, H. I. (eds.): Liposome Dermatics, Springer-Verlag, Heidelberg 1992
105. Meybeck, A.; Bonte, F.; Redzinak, G.: presented at 5th Int. Conf. Pharmaceutical Technology, Paris, May 30 to June 1, 1989, 399
106. Korting, H. C.; Schäfer-Korting, M.; Hart, A.; Laux, P.; Schmid, M.: Eur. J. Clin. Pharmacol. 44, 315 (1993)
107. Schäfer-Korting, M.; Korting, H. C.; Ponce-Pälschl, E.: Ccinvestig., 72, 1086, 1994
108. Gesztes, A.; Mezei, M.: Anesth. Analg. 67, 1079 (1988)
109. Molitor, H.; Fernandez, L.: Am. J. Med. Sci. 198, 778 (1993)
110. Novak, E. J.: Arch. Phys. Med. Rehab. 45, 1231 (1964)
111. Dynnik, T. K.: Vrach. Del. 115 (1977)
112. Fahim, M.: J. Med. 9, 245 (1978)
113. Fahim, M.: J. Med. 11, 143 (1980)
114. Barry, B. W.; Woodford, R. K.: Br. J. Dermatol. 91, 323 (1974)
115. Brucks, R.; Nanavaty, M.; Jung, D.; Siegel, F.: Pharm. Res. 6, 697 (1982)
116. Levy, D.; Kost, J.; Meshulam, Y.; Langer, R.: J. Clin. Invest. 83, 2074 (1989)
117. Bommannan, D.; Okuyama, H.; Stauffer, P.; Guy, R. H.: Pharm. Res. 9, 559 (1989)
118. Miyazaki, S.; Mizuoka, H.; Oda, M.; Takada, M.: J. Pharm. Pharmacol. 43, 115 (1991)
119. Tachibana, K.: Pharm. Res. 9, 952 (1992)
120. McElnay, J. C.; Kennedy, T. A.; Harland, R.: Int. J. Pharm. 40, 105 (1987)
121. Paaske, W. P.; Hovind, H.; Sejrsen, P.: Scand. J. Clin. Lab. Invest. 31, 389 (1973)
122. Bommannan, D.; Menon, G. K.; Okuyama, H.; Elias, P. M.; Guy, R. H.: Pharm. Res. 9, 1043 (1992)
123. Elias, P. M.: Int. J. Derm. 20, 1 (1981)
124. Barry, B. W.: Skin Pharmakol. 1, 121 (1987)