New electrophilic reactions of 2,2′-bisindolyls with acid chlorides and carbodienophiles

Journal of Heterocyclic Chemistry

Volumn 33, Issue 3, 1996, Pages 623-631

  Pindur, U ^a   Kim, Y S ^a  

^a JOHANNES GUTENBERG UNIVERSITY   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

CARBAZOLE DERIVATIVE; INDOLE DERIVATIVE;

ARTICLE; DRUG STRUCTURE; DRUG SYNTHESIS; NUCLEAR MAGNETIC RESONANCE; REACTION ANALYSIS;

EID: 0029740185     PISSN: 0022152X     EISSN: None     Source Type: Journal    
DOI: 10.1002/jhet.5570330317     Document Type: Article

References (13)

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3. J. H. Hartenstein and C. Schächtele, The Design of Protein Kinase C Inhibitors in Perspectives in Medicinal Chemistry, B. Testa, ed, Helvetica Chimica Acta, Basel and VCH Weinheim, 1992, pp 99-119.
4. U. Pindur, Y.-S. Kim and D. Schollmeyer, J. Heterocyclic Chem., 31, 377 (1994).
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6. U. Pindur, Y.-S. Kim and D. Schollmeyer, J. Heterocyclic Chem., 32, 1335 (1995).
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11. For structural aspects of atropisomers see: M. Oki, Top. Stereochem., 14, 1 (1983).
12. The protein kinase C α inhibition assay was performed by P. M. Blumberg, in the National Cancer Institute, Molecular Mechanisms of Tumor Promotion Section, Bethesda, MD; USA; A. P. Kozikowski, P. M. Blumberg J. Am. Chem. Soc., 117, 6666 (1995).
13. D. Schollmeyer, Y.-S. Kim and U. Pindur, structural results in preparation for Acta Crystallogr. Sect C.