Comparison of [3H]YM060 binding to native and cloned rat 5-HT3 receptors

European Journal of Pharmacology

Volumn 296, Issue 2, 1996, Pages 227-230

  Akuzawa, Shinobu ^a,b   Miyake, Akira ^b   Miyata, Keiji ^b   Fukutomi, Hisayuki ^a  

^a UNIVERSITY OF TSUKUBA   (Japan)

^b ASTELLAS PHARMA INC   (Japan)

Author keywords

5 HT3 receptor; 5 HT3 receptor, cloned, rat; Cerebral cortex; Colon; Ileum; 3H YM060 ( methyl 3H ( ) (R) 5 (1 methyl 1H indol 3 yl)carbonyl 4,5,6,7 tetrahydro 1H benzimidazole monohydrochloride)

Indexed keywords

1 (3 CHLOROPHENYL)BIGUANIDE; 2 METHYLSEROTONIN; 4,5,6,7 TETRAHYDRO 5 (1 INDOLYLCARBONYL)BENZIMIDAZOLE; COMPLEMENTARY DNA; GRANISETRON; ONDANSETRON; RADIOLIGAND; RAMOSETRON; SEROTONIN; SEROTONIN 3 RECEPTOR; SEROTONIN AGONIST; SEROTONIN ANTAGONIST; TROPISETRON; BENZIMIDAZOLE DERIVATIVE; SEROTONIN RECEPTOR;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; BINDING COMPETITION; BRAIN CORTEX; COLON; CONTROLLED STUDY; DISSOCIATION CONSTANT; ILEUM; MALE; MOLECULAR CLONING; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR BINDING; ANIMAL; COMPARATIVE STUDY; GENETICS; IN VITRO STUDY; METABOLISM; PROTEIN BINDING; RADIOASSAY; WISTAR RAT;

ANIMALS; BENZIMIDAZOLES; CLONING, MOLECULAR; MALE; PROTEIN BINDING; RADIOLIGAND ASSAY; RATS; RATS, WISTAR; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT3; SEROTONIN ANTAGONISTS;

EID: 0029670664     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/0014-2999(95)00798-9     Document Type: Article

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