Correlation between guanine nucleotide effect and reversible binding property of endothelin analogs

Neuropeptides

Volumn 30, Issue 1, 1996, Pages 109-114

  Nambi, P ^a   Pullen, M ^a   Aiyar, N ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

DIAGNOSTIC AGENT; ENDOTHELIN; ENDOTHELIN RECEPTOR; GUANINE NUCLEOTIDE; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); PEPTIDE FRAGMENT; RADIOACTIVE IODINE; SUCCINYLENDOTHELIN 1 [8-21][9 GLUTAMIC ACID 11,15 ALANINE]; ENDOTHELIN RECEPTOR AGONIST; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE TRIPHOSPHATE DERIVATIVE;

ANIMAL; ARTICLE; CELL MEMBRANE; CHO CELL; DOG; DRUG ANTAGONISM; DRUG EFFECT; GENETIC TRANSFECTION; GUINEA PIG; HAMSTER; HUMAN; IN VITRO STUDY; KINETICS; LUNG; METABOLISM; RADIOASSAY; RAT; SWINE; ANIMAL CELL; CELL CULTURE; CHINESE HAMSTER; CONTROLLED STUDY; FEMALE; HUMAN TISSUE; NONHUMAN; OVARY CELL; PRIORITY JOURNAL; RECEPTOR BINDING;

ANIMALS; CELL MEMBRANE; CHO CELLS; CRICETINAE; DOGS; ENDOTHELINS; GUANINE NUCLEOTIDES; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); GUINEA PIGS; HUMANS; IODINE RADIOISOTOPES; KINETICS; LUNG; PEPTIDE FRAGMENTS; RADIOLIGAND ASSAY; RATS; RECEPTORS, ENDOTHELIN; SWINE; TRANSFECTION;

ANIMALIA; CANIS FAMILIARIS; CAVIA PORCELLUS; CRICETINAE; SUS SCROFA;

EID: 0029670307     PISSN: 01434179     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0143-4179(96)90063-3     Document Type: Article

References (22)

1. Yanagisawa M, Kurihara M, Kimura S, et al. Endothelin: a novel potent vasoconstrictor peptide produced by vascular endothelial cells. Nature 1988; 332: 411-415.
2. Inoue A, Yanagisawa M, Kimura S, et al. The human endothelial family: three structurally and pharmacologically distinct isopeptides predicted by three separate genes. Proc Natl Acad Sci USA 1989; 86: 2863-2867.
3. Kloog Y, Ambar I, Sokolovsky M, Wollberg Z. Sarafotoxin, a novel vasoconstrictor peptide: phosphoinositide hydrolysis in rat heart and brain. Science 1988; 242: 268-270.
4. Kloog Y, Sokolovsky M. Similarities in mode and sites of action of sarafotoxins and endothelins. Trends Pharmacol Sci 1989; 10: 212-214.
5. Nambi P, Pullen M, Feuerstein G. Identification of endothelin receptors in various regions of rat brain. Neuropeptides 1990; 16: 195-199.
6. Nambi P, Pullen M, Wu H-L, Aiyar N, Ohlstein E H, Edwards R M. Identification of endothelin receptor subtypes in human renal cortex and medulla using subtype-selective ligands. Endocrinology .1992; 131: 1081-1086.
7. Nambi P, Wu H-L, Pullen M, Aiyar N, Bryan H, Elliott J D. Identification of endothelin receptor subtypes in rat kidney cortex using subtype-selective ligands. Mol Pharmacol 1992; 42: 336-339.
8. Martins E R, Brenner B M, Ballerman B J. Heterogeneity of cell surface endothelin receptors. J Biol Chem 1990; 265: 14044-14049.
9. Brooks D P, DePalma P D, Pullen M, Nambi P. Characterization of canine renal endothelin receptor subtypes and their function. J Pharmacol Exp Ther 1994; 268: 1091-1097
10. Simonson M S, Dunn M J. Cellular signalling by peptides of the endothelin gene family. FASEB J 1990; 4: 2989-3000.
11. Arai H, Hori S, Aramori H, Ohkubo H, Nakanishi S. Cloning and expression of a cDNA encoding an endothelin receptor. Nature 1990; 348: 730-732.
12. Elshourbagy N, Korman D, Nuthulaganti P et al. Molecular characterization and regulation of the human endothelin receptors. J Biol Chem 1993; 268: 3873-3879.
13. Sakurai T, Yanagisawa M, Takuwa Y et al. Cloning of a cDNA encoding a non-isopeptide-selective subtype of the endothelin receptor. Nature 1990; 348: 732-735.
14. Karne S, Jayawickreme C K Lerner M R. Cloning and characterization of an endothelin-3 specific receptor (ETC receptor) from Xenopus laevis dermal melanophores. J Biol Chem 1993; 268: 19126-19133.
15. Kumar C, Mwangi V, Nuthulaganti P, et al. Cloning and characterization of a novel endothelin receptor from Xenopus heart. J Biol Chem 1994; 269: 13414-13420.
16. Gilman A G. G proteins: transducers of receptor-generated signals. Ann Rev Biochem 1987; 56: 615-649.
17. Dohlman H G, Thorner J, Caron M G, Lefkowitz R J. Model systems for the study of seven transmembrane-segment receptors. Ann Rev Biochem 1991; 60: 653-688.
18. 125I]-IRL-1620, a potent agonist specific for endothelin-B receptors. J Pharmacol Exp Ther 1994; 268: 202-207.
19. 125I]-IRL-1620. Biochem Biophys Res Commun 1992; 185: 867-873.
20. B receptor. Biochem Biophys Res Commun 1992; 184: 953-959.
21. B receptor. Cardiovasc Drug Rev 1993; 11: 253-270.
22. B-selective agonist displays species differences in its binding characteristics. Neuropeptides 1995; 28: 191-196.