Dopamine D2 receptor model explains binding affinity of neuroleptics: Piquindone and its structure activity relationships

Drug Design and Discovery

Volumn 13, Issue 3-4, 1996, Pages 49-62

  Teeter, Martha M ^a   Durand, Curtiss J ^b  

^a BOSTON COLLEGE   (United States)

^b BOSTON UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

D2 receptor model; Modeling; Piquindone

Indexed keywords

DOPAMINE 2 RECEPTOR; GUANINE NUCLEOTIDE BINDING PROTEIN; NEUROLEPTIC AGENT; PIQUINDONE; BACTERIORHODOPSIN; ISOQUINOLINE DERIVATIVE; RHODOPSIN; RO 22-1319;

BINDING AFFINITY; CONFERENCE PAPER; DRUG BINDING SITE; DRUG RECEPTOR BINDING; STRUCTURE ACTIVITY RELATION; ARTICLE; BINDING SITE; CHEMICAL STRUCTURE; CHEMISTRY; CONFORMATION; METABOLISM; PROTEIN BINDING; PROTEIN TERTIARY STRUCTURE;

ANTIPSYCHOTIC AGENTS; BACTERIORHODOPSINS; BINDING SITES; GTP-BINDING PROTEINS; ISOQUINOLINES; MODELS, MOLECULAR; MOLECULAR CONFORMATION; PROTEIN BINDING; PROTEIN STRUCTURE, TERTIARY; RECEPTORS, DOPAMINE D2; RHODOPSIN; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0029658596     PISSN: 10559612     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Conference Paper

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