Endothelin ETA and ETB receptors mediate endothelin-1-induced apamin-sensitive relaxation in the guinea pig ileum

Japanese Journal of Pharmacology

Volumn 70, Issue 3, 1996, Pages 259-267

  Shan, Li Hua ^a   Nishiyama, Mariko ^a   Shibasaki, Tadao ^b   Moroi, Kayoko ^a   Goto, Katsutoshi ^b   Masaki, Tomoh ^c   Kimura, Sadao ^a  

^a CHIBA UNIVERSITY SCHOOL OF MEDICINE   (Japan)

^b UNIVERSITY OF TSUKUBA   (Japan)

^c KYOTO UNIVERSITY   (Japan)

Author keywords

Apamin; Endothelin; Endothelin receptor; Ileal smooth muscle (guinea pig); Relaxation

Indexed keywords

APAMIN; CARBACHOL; CYCLO(DEXTRO TRYPTOPHYL DEXTRO ASPARTYLPROLYL DEXTRO VALYLLEUCYL); ENDOTHELIN 1; ENDOTHELIN 3; ENDOTHELIN A RECEPTOR; ENDOTHELIN B RECEPTOR; N (2,6 DIMETHYLPIPERIDINOCARBONYL) 4 METHYLLEUCYL DEXTRO (1 METHOXYCARBONYLTRYPTOPHANYL) DEXTRO NORLEUCINE; N ACETYL 3,3 DIPHENYL DEXTRO ALANYLLEUCYLASPARTYLISOLEUCYLISOLEUCYLTRYPTOPHAN; POTASSIUM CHANNEL; SARAFOTOXIN S6C; SUCCINYLENDOTHELIN 1 [8-21][9 GLUTAMIC ACID 11,15 ALANINE]; CYCLO(TRP ASP PRO VAL LEU); CYCLO(TRP-ASP-PRO-VAL-LEU); CYCLOPEPTIDE; ENDOTHELIN; ENDOTHELIN RECEPTOR; PEPTIDE FRAGMENT; SARAFOTOXINS S6; VIPER VENOM;

ANIMAL TISSUE; ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; GUINEA PIG; ILEUM; ILEUM CONTRACTION; MALE; NONHUMAN; SMOOTH MUSCLE RELAXATION; ANIMAL; COMPARATIVE STUDY; DOSE RESPONSE; DRUG EFFECT; IN VITRO STUDY; MUSCLE RELAXATION; PHYSIOLOGY; SMOOTH MUSCLE;

ANIMALS; APAMIN; DOSE-RESPONSE RELATIONSHIP, DRUG; ENDOTHELINS; GUINEA PIGS; ILEUM; MALE; MUSCLE RELAXATION; MUSCLE, SMOOTH; PEPTIDE FRAGMENTS; PEPTIDES, CYCLIC; RECEPTORS, ENDOTHELIN; VIPER VENOMS;

EID: 0029658330     PISSN: 00215198     EISSN: None     Source Type: Journal    
DOI: 10.1254/jjp.70.259     Document Type: Article

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