The histamine H1 receptor in GT1-7 neuronal cells is regulated by calcium influx and KN-62, a putative inhibitor of calcium/calmodulin protein kinase II

British Journal of Pharmacology

Volumn 118, Issue 5, 1996, Pages 1119-1126

  Reza Zamani, M ^a,b   Bristow, David R ^a  

^a UNIVERSITY OF MANCHESTER   (United Kingdom)

^b UNIVERSITY OF LIVERPOOL   (United Kingdom)

Author keywords

Bradykinin; Calcium oscillation; Calcium calmodulin dependent protein kinase II; GT1 7 neuronal cells; Heterologous desensitization; Histamine H1 receptor; Homologous desensitization; Intracellular calcium

Indexed keywords

1 [N,O BIS(5 ISOQUINOLINESULFONYL) N METHYLTYROSYL] 4 PHENYLPIPERAZINE; BRADYKININ; CALCIUM ION; HISTAMINE; HISTAMINE H1 RECEPTOR; PROTEIN KINASE (CALCIUM,CALMODULIN) II; PROTEIN KINASE INHIBITOR; 1 (5 ISOQUINOLINESULFONYL) 2 METHYLPIPERAZINE; ANTIHISTAMINIC AGENT; CALCIUM; DRUG DERIVATIVE; PROTEIN KINASE (CALCIUM,CALMODULIN);

ARTICLE; CALCIUM CELL LEVEL; CALCIUM TRANSPORT; CONTROLLED STUDY; EXTRACELLULAR CALCIUM; NERVE CELL CULTURE; PRIORITY JOURNAL; RECEPTOR DOWN REGULATION; ANIMAL; CATTLE; CELL CULTURE; DOSE RESPONSE; DRUG ANTAGONISM; DRUG EFFECT; METABOLISM; SIGNAL TRANSDUCTION;

1-(5-ISOQUINOLINESULFONYL)-2-METHYLPIPERAZINE; ANIMALS; BRADYKININ; CA(2+)-CALMODULIN DEPENDENT PROTEIN KINASE; CALCIUM; CATTLE; DOSE-RESPONSE RELATIONSHIP, DRUG; HISTAMINE; HISTAMINE ANTAGONISTS; RECEPTORS, HISTAMINE H1; SIGNAL TRANSDUCTION; TUMOR CELLS, CULTURED;

EID: 0029657867     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1476-5381.1996.tb15514.x     Document Type: Article

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