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Bioorganic and Medicinal Chemistry

Volumn 3, Issue 12, 1995, Pages 1651-1656

Enantioselective inhibition of the epidermal growth factor receptor tyrosine kinase by 4-(α-phenethylamino)quinazolines

(5) Bridges, Alexander J a Cody, Donna R a Zhou, Hairong a McMichael, Amy a Fry, David W a

a PFIZER INC (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 (1 PHENYLETHYLAMINO)QUINAZOLINE; 6,7 DIMETHOXY 4 (1 PHENYLETHYLAMINO)QUINAZOLINE; ADENOSINE TRIPHOSPHATE; EPIDERMAL GROWTH FACTOR RECEPTOR; EPIDERMAL GROWTH FACTOR RECEPTOR KINASE; PROTEIN TYROSINE KINASE; PROTEIN TYROSINE KINASE INHIBITOR; QUINAZOLINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG BINDING; DRUG SYNTHESIS; ENANTIOMER; ENZYME INHIBITION; ENZYME KINETICS; HUMAN; HUMAN CELL; QUANTITATIVE STRUCTURE ACTIVITY RELATION; TUMOR CELL;

ADENOSINE TRIPHOSPHATE; AMINO ACID SEQUENCE; BINDING SITES; ENZYME INHIBITORS; HUMANS; KINETICS; MAGNETIC RESONANCE SPECTROSCOPY; MOLECULAR SEQUENCE DATA; PEPTIDES; PROTEIN CONFORMATION; QUINAZOLINES; RECEPTOR, EPIDERMAL GROWTH FACTOR; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; SUBSTRATE SPECIFICITY;

EID: 0029611204 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/0968-0896(95)00149-2 Document Type: Article

Times cited : (33)

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