Substrates of human hepatic cytochrome P450 3A4

Toxicology

Volumn 104, Issue 1-3, 1995, Pages 1-8

  Li, Albert P ^a   Kaminski, Donald L ^a   Rasmussen, Asenath ^a  

^a SAINT LOUIS UNIVERSITY   (United States)

Author keywords

Biotransformation; Cytochrome P450; Cytochrome P450 3A4; Human drug metabolism; Xenobiotics

Indexed keywords

AMIODARONE; ANALGESIC AGENT; ANTIANDROGEN; ANTIARRHYTHMIC AGENT; ANTIBIOTIC AGENT; ANTICONVULSIVE AGENT; ANTIDEPRESSANT AGENT; ANTIESTROGEN; ANTIHISTAMINIC AGENT; ANTILIPEMIC AGENT; ANTINEOPLASTIC AGENT; ANTITUSSIVE AGENT; CAFFEINE; CHEMICAL AGENT; CLONAZEPAM; COCAINE; CONTRACEPTIVE AGENT; CYTOCHROME; CYTOCHROME P450 ISOENZYME; DEXTROMETHORPHAN; DILTIAZEM; DRUG; ESTRADIOL; HORMONE; IFOSFAMIDE; IMMUNOSUPPRESSIVE AGENT; OPIATE; PSYCHOTROPIC AGENT; STEROID; UNINDEXED DRUG;

DRUG METABOLISM; ENZYME SUBSTRATE; HUMAN; HUMAN CELL; LIVER CELL; NONHUMAN; PRIORITY JOURNAL; REVIEW; XENOBIOTIC METABOLISM; YEAST;

BIOTRANSFORMATION; CELLS, CULTURED; CYTOCHROME P-450 ENZYME SYSTEM; ENZYME INDUCTION; ENZYME INHIBITORS; HUMANS; HYDROXYLATION; LIVER; MICROSOMES, LIVER; MIXED FUNCTION OXYGENASES; OXIDATION-REDUCTION; STRUCTURE-ACTIVITY RELATIONSHIP; SUBSTRATE SPECIFICITY; XENOBIOTICS;

EID: 0029584276     PISSN: 0300483X     EISSN: None     Source Type: Journal    
DOI: 10.1016/0300-483X(95)03155-9     Document Type: Review

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