Identification of a hexapeptide inhibitor of the human immunodeficiency virus integrase protein by using a combinatorial chemical library

Proceedings of the National Academy of Sciences of the United States of America

Volumn 92, Issue 25, 1995, Pages 11456-11460

  Puras Lutzke, Ramon A ^a   Eppens, Noor A ^a   Weber, Patricia A ^b   Houghten, Richard A ^c   Plasterk, Ronald H A ^a  

^a NETHERLANDS CANCER INSTITUTE   (Netherlands)

^b Houghten Pharmaceuticals Inc   (United States)

^c TORREY PINES INSTITUTE FOR MOLECULAR STUDIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

OLIGOPEPTIDE; PROTEIN INHIBITOR; VIRUS PROTEIN;

ARTICLE; DNA INTEGRATION; DRUG ACTIVITY; DRUG SCREENING; HUMAN IMMUNODEFICIENCY VIRUS; NONHUMAN; PRIORITY JOURNAL; PROTEIN ANALYSIS; VIRUS INHIBITION;

AMINO ACID SEQUENCE; DNA NUCLEOTIDYLTRANSFERASES; DRUG EVALUATION, PRECLINICAL; ENZYME INHIBITORS; HIV-1; HIV-2; IMMUNODEFICIENCY VIRUS, FELINE; INTEGRASES; MOLECULAR SEQUENCE DATA; MOLONEY MURINE LEUKEMIA VIRUS; OLIGOPEPTIDES; RETROVIRIDAE; STRUCTURE-ACTIVITY RELATIONSHIP; VIRUS INTEGRATION;

FELIDAE; FELINE IMMUNODEFICIENCY VIRUS; HUMAN IMMUNODEFICIENCY VIRUS; HUMAN IMMUNODEFICIENCY VIRUS 2; MOLONEY MURINE LEUKEMIA VIRUS; MURINAE;

EID: 0029557124     PISSN: 00278424     EISSN: None     Source Type: Journal    
DOI: 10.1073/pnas.92.25.11456     Document Type: Article

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