Molecular design and biological activity of potent and selective protein kinase inhibitors related to balanol

Chemistry and Biology

Volumn 2, Issue 9, 1995, Pages 601-608

  Koide, Kazunori ^a   Bunnage, Mark E ^b   Gomez Paloma, Luigi ^b   Kanter, Joan R ^a   Taylor, Susan S ^a   Brunton, Laurence L ^a   Nicolaou, K C ^a,b  

^a UNIVERSITY OF CALIFORNIA   (United States)

^b SCRIPPS RESEARCH INSTITUTE   (United States)

Author keywords

balanol; balanol analogs; inhibitor; protein kinase A; protein kinase C

Indexed keywords

ADENOSINE TRIPHOSPHATE; AZEPINE DERIVATIVE; BALANOL; CYCLIC AMP DEPENDENT PROTEIN KINASE; ENZYME INHIBITOR; EPIDERMAL GROWTH FACTOR RECEPTOR; HYDROXYBENZOIC ACID DERIVATIVE; PROTEIN KINASE C; PROTEIN TYROSINE KINASE;

ARTICLE; CHEMICAL STRUCTURE; CHEMISTRY; DRUG ANTAGONISM; DRUG DESIGN; KINETICS; METABOLISM; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

ADENOSINE TRIPHOSPHATE; AZEPINES; CYCLIC AMP-DEPENDENT PROTEIN KINASES; DRUG DESIGN; ENZYME INHIBITORS; HYDROXYBENZOIC ACIDS; KINETICS; MODELS, MOLECULAR; PROTEIN KINASE C; RECEPTOR, EPIDERMAL GROWTH FACTOR; SRC-FAMILY KINASES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0029360744     PISSN: 10745521     EISSN: None     Source Type: Journal    
DOI: 10.1016/1074-5521(95)90124-8     Document Type: Article

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