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Bioorganic and Medicinal Chemistry Letters

Volumn 5, Issue 12, 1995, Pages 1311-1314

An efficient synthesis of the benzhydrylpiperazine delta opioid agonist (+)-BW373U86

(2) Bishop, Michael J a McNutt, Robert W a

a Burroughs Wellcome Co (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BW 373486; DELTA OPIATE RECEPTOR; DELTA OPIATE RECEPTOR AGONIST; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DRUG SYNTHESIS; STEREOSPECIFICITY; TECHNIQUE;

EID: 0029068024 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/0960-894X(95)00213-D Document Type: Article

Times cited : (67)

References (15)

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4
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- For some examples, see:, B.M. Trost, I. Fleming, Pergamon Press, Oxford
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- Kleinman¹ Volkmann²

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- Yamamoto¹ Kubota² Honda³ Fukui⁴ Asao⁵ Nemoto⁶

8
- 0000716787
- For a review of nucleophilic additions to imines and iminium salts, see:, B.M. Trost, I. Fleming, Pergamon Press, Oxford
- (1991) Comprehensive Organic Synth. , vol.1 , pp. 355-396
- Volkmann¹

9
- 37049081753
- The chemistry of N-substituted benzotriazoles. Part 4. A novel and versatile method for the mono-N-alkylation of aromatic and heteroaromatic amines
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- Katritzky¹ Rachwal² Rachwal³

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- The chemistry of N-substituted benzotriazoles. Part 14. Novel routes to secondary and tertiary amines and to N, N-disubstituted hydroxylamines
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- Katritzky¹ Yannakopoulou² Lue³ Rasala⁴ Urogdi⁵

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- This aldehyde was prepared by heating 4-carboxybenzaldehyde to reflux in neat thionyl chloride until complete dissolution, removing all volatiles, and treating the residue with excess diethylamine in dichloromethane at 0°C. This procedure gives aldehyde 6 in 98% yield without need for further purification.

13
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- Prepared from 3-bromophenol. The silyl protecting group was affixed using t-butyldimethylsilyl chloride with imidazole in DMF. Treatment with n-BuLi in THF at -78°C, followed by addition to a stirring solution of magnesium bromide etherate in THF at 25°C generated the 3-(t-butyldimethyl-silyloxy)phenylmagnesium bromide

14
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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.