Properties of TAN-67, a nonpeptide δ-opioid receptor agonist, at cloned human δ-and μ-opioid receptors

European Journal of Pharmacology: Molecular Pharmacology

Volumn 291, Issue 2, 1995, Pages 129-134

  Knapp, Richard J ^a   Landsman, Robert ^a   Waite, Sue ^a   Malatynska, Ewa ^a   Varga, Eva ^a   Haq, Wajujahal ^a   Hruby, Victor J ^a   Roeske, William R ^a   Nagase, Hiroshi ^b   Yamamura, Henry I ^a  

^a UNIVERSITY OF ARIZONA   (United States)

^b TORAY INDUSTRIES INC   (Japan)

Author keywords

Adenylyl cylase; cAMP; Endorphin receptor; Radioligand binding; Recombinant cell

Indexed keywords

1,2,3,4,4A,5,12,12AALPHA OCTAHYDRO 4AALPHA (3 HYDROXYPHENYL) 2 METHYLQUINOLINO[2,3 G]ISOQUINOLINE; 4 CHLORO DPDPE; ADENYLATE CYCLASE; CYCLIC AMP; DELTA OPIATE RECEPTOR; DELTA OPIATE RECEPTOR AGONIST; DEXTRO PHENYLALANYLCYSTEINYLTYROSYL DEXTRO TRYPTOPHYLORNITHYLTHREONYLPENICILLAMINYLTHREONINAMIDE 2,7 DISULFIDE; ENKEPHALIN DERIVATIVE; ENKEPHALIN[2 DEXTRO ALANINE 4 METHYLPHENYLALANINE 5 GLYCINE]; FORSKOLIN; MU OPIATE RECEPTOR; NALTRINDOLE; RADIOLIGAND; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CHO CELL; CONTROLLED STUDY; DRUG POTENCY; DRUG SELECTIVITY; ENZYME ACTIVATION; FIBROBLAST; HUMAN; MOLECULAR CLONING; MOUSE; NONHUMAN; PRIORITY JOURNAL; RECEPTOR BINDING;

ANALGESICS; ANIMAL; BINDING, COMPETITIVE; CHO CELLS; CLONING, MOLECULAR; CYCLIC AMP; FORSKOLIN; HAMSTERS; HUMAN; QUINOLINES; RADIOLIGAND ASSAY; RECEPTORS, OPIOID, DELTA; RECEPTORS, OPIOID, MU; SUPPORT, U.S. GOV'T, P.H.S.;

EID: 0028972805     PISSN: 09224106     EISSN: None     Source Type: Journal    
DOI: 10.1016/0922-4106(95)90134-5     Document Type: Article

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