Fluorinated benzamide neuroleptics-III. Development of (S)-N-[(1-allyl-2-pyrrolidinyl)methyl]-5-(3-[18F]fluoropropyl)-2,3-dimethoxybenzamide as an improved dopamine D-2 receptor tracer

Nuclear Medicine and Biology

Volumn 22, Issue 3, 1995, Pages 283-296

  Mukherjee, Jogeshwar ^a   Yang, Zhi Ying ^a   Das, Malay K ^a   Brown, Terry ^a  

^a Franklin McLean Memorial Research Institute   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

8 CHLORO 2,3,4,5 TETRAHYDRO 3 METHYL 5 PHENYL 1H 3 BENZAZEPIN 7 OL HYDROGEN MALEATE; BENZAMIDE DERIVATIVE; DOPAMINE RECEPTOR; DOPAMINE RECEPTOR BLOCKING AGENT; EPIDEPRIDE; FALLYPRIDE; FLUORINE 18; HALOPERIDOL; NEUROLEPTIC AGENT; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; BRAIN; CONTROLLED STUDY; DRUG SYNTHESIS; INTRAVENOUS DRUG ADMINISTRATION; ISOTOPE LABELING; MONKEY; POSITRON EMISSION TOMOGRAPHY;

ANIMAL; ANTIPSYCHOTIC AGENTS; BENZAMIDES; BINDING, COMPETITIVE; BRAIN; CEBUS; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; FLUORINE RADIOISOTOPES; MACACA MULATTA; MALE; MOLECULAR STRUCTURE; PYRROLIDINES; RADIOACTIVE TRACERS; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, DOPAMINE D2; STRUCTURE-ACTIVITY RELATIONSHIP; SUPPORT, NON-U.S. GOV'T; SUPPORT, U.S. GOV'T, NON-P.H.S.; TISSUE DISTRIBUTION; TOMOGRAPHY, EMISSION-COMPUTED;

EID: 0028964653     PISSN: 09698051     EISSN: None     Source Type: Journal    
DOI: 10.1016/0969-8051(94)00117-3     Document Type: Article

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