Metalation of diazines. XI. Directed ortho‐lithiation of fluoropyrimidines and application to synthesis of an azacarboline

Journal of Heterocyclic Chemistry

Volumn 31, Issue 6, 1994, Pages 1311-1315

  Ple N ^a   Turck, A ^a   Heynderickx, A ^a   Queguiner G ^a  

^a IRCOF   (France)

Author keywords

[No Author keywords available]

Indexed keywords

3 THIOMETHYL 9H PYRIMIDO[4,5 B]INDOLE; INDOLE DERIVATIVE; PYRIMIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG SYNTHESIS; REACTION ANALYSIS; STEREOCHEMISTRY;

EID: 0028569598     PISSN: 0022152X     EISSN: 19435193     Source Type: Journal    
DOI: 10.1002/jhet.5570310602     Document Type: Article

References (29)

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2. Metallation of diazinesII. First metallation of pyridazine, metallation of 2,4-dichloropyrimidine
3. Metallation of diazines.III. New synthesis of analogues of trimethoprim and of bacimethrin
4. Metallation of diazines.V. Synthesis of analogues of biologically active molecules
5. Metalation of diazines.VI. Metalation of pivaloylaminopyrazine andN-t-butylpyrazinamide. Unusual regioselectivity in the metalation reaction
6. A facile synthesis of 9H-pyrimido [4,5-b]indoleviaphotolysis of 4-azido-5-phenylpyrimidine
7. Triazolo[4,5-d]pyrimidines. VII. The Photo-chemical Transformation of 3-phenyl-3H -1,2,3-triazolo[4,5-d]pyrimidines into 9H -Pyrimido[4,5-b]indoles