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Bioorganic and Medicinal Chemistry Letters

Volumn 4, Issue 3, 1994, Pages 415-420

1,1-diphenyl-3-dialkylamino-1-silacyclopentane derivatives: A new class of potent and selective 5-HT2A antagonists

(6) Damour, Dominique a Barreau, Michel a Dutruc Rosset, Gilles a Doble, Adam a Piot, Odile a Mignani, Serge a

a SANOFI (France)

Author keywords

[No Author keywords available]

Indexed keywords

1,1 BIS(4 FLUOROPHENYL) 3 (4 PHENYL 1 PIPERAZINYL) 1 SILACYCLOPENTANE; CYCLOPENTANE DERIVATIVE; ORGANOSILICON DERIVATIVE; RITANSERIN; SEROTONIN 2A RECEPTOR; SEROTONIN ANTAGONIST; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BEHAVIOR; BRAIN CORTEX; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; ENANTIOMER; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; MOUSE; NONHUMAN; ORAL DRUG ADMINISTRATION; QUANTITATIVE STRUCTURE ACTIVITY RELATION; RAT; SUBCUTANEOUS DRUG ADMINISTRATION; ULTRAVIOLET SPECTROPHOTOMETRY;

EID: 0028299769 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/0960-894X(94)80007-3 Document Type: Article

Times cited : (17)

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