(−)‐Discretamine, a selective α1D‐adrenoceptor antagonist, isolated from Fissistigma glaucescens

British Journal of Pharmacology

Volumn 112, Issue 4, 1994, Pages 1174-1180

  Ko, Feng‐Nien ^a   Guh, Jih‐Hwa ^a   Yu, Sheu‐Meei ^b   Hou, Yu‐Sheng ^b   Wu, Yang‐Chang ^c   Teng, Che‐Ming ^a  

^a NATIONAL TAIWAN UNIVERSITY   (Taiwan)

^b CHANG GUNG UNIVERSITY   (Taiwan)

^c KAOHSIUNG MEDICAL UNIVERSITY   (Taiwan)

Author keywords

( ) discretamine; Fissistigma glaucescens; rat thoracic aorta; 1D Adrenoceptor antagonist

Indexed keywords

5 METHYLURAPIDIL; ACETYLCHOLINE; ALPHA 1 ADRENERGIC RECEPTOR; ALPHA ADRENERGIC RECEPTOR BLOCKING AGENT; CHLOROETHYLCLONIDINE; DISCRETAMINE; NIFEDIPINE; NORADRENALIN; PHENTOLAMINE; PHENYLEPHRINE; PRAZOSIN;

ANIMAL CELL; ANIMAL TISSUE; AORTA; ARTICLE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; FEMALE; MALE; MUSCLE CONTRACTION; MUSCLE RELAXATION; NONHUMAN; PRIORITY JOURNAL; RAT; SPLEEN; VAS DEFERENS;

ADRENERGIC ALPHA-ANTAGONISTS; ANIMAL; BERBERINE ALKALOIDS; CELLS, CULTURED; FEMALE; INOSITOL PHOSPHATES; MALE; NOREPINEPHRINE; PLANTS; RATS; RATS, WISTAR; RECEPTORS, ADRENERGIC, ALPHA-1; SPLEEN; SUPPORT, NON-U.S. GOV'T; VAS DEFERENS; VASOCONSTRICTION;

EID: 0028169146     PISSN: 00071188     EISSN: 14765381     Source Type: Journal    
DOI: 10.1111/j.1476-5381.1994.tb13207.x     Document Type: Article

References (27)

1. Investigations of contractions mediated by noradrenaline in rat aorta
2. 1‐adrenoceptor mediating contractions of rat aorta, vas deferens and spleen
3. Differences in the adenosine receptors modulating inositol phosphates and cyclic AMP accumulation in mammalian cerebral cortex
4. 1‐adrenergic receptor
5. 2+ in smooth muscle
6. 1MF‐2 and BC3H‐1 clonal cell lines
7. 1‐adrenoceptors in rat blood vessels
8. 1‐adrenoceptor recognition sites by urapidil derivatives and other selective antagonists
9. Classification of phenoxybenzamine/prazosin resistant contractions of rat spleen to norepinephrine by Schild analysis: similarities and differences to postsynaptic alpha‐2 adrenoceptors
10. Pharmacological activity of (−)‐discretamine, a novel vascular α‐adrenoceptor and 5‐hydroxytryptamine receptor antagonist, isolated from
11. 1A‐adrenergic receptor
12. Protein measurement with the Folin phenol reagent
13. Alkaloids of Formosan Fissistigma and Goniothalamus species
14. 2 and affinity constants for pharmacological competitive antagonists be estimated
15. 2+
16. 3H]prazosin binding
17. LIGAND: A versatile computerized approach for characterization of ligand‐binding system
18. 1‐adrenoceptors involved in noradrenaline induced contractions of rat thoracic aorta and dog carotid artery
19. 1‐adrenoceptors in mammalian aortae: subclassification based on chloroethylclonidine, WB4101 and nifedipine
20. 1D‐adrenergic receptor cDNA
21. 1‐adrenoceptor
22. 1‐adrenergic receptor subtype
23. 1C‐adrenoceptor: characterization of signal transduction pathways and mammalian tissue heterogeneity
24. 2+ signalling mechanism and plays a different physiological role
25. 1‐adrenergic receptors
26. 2+ influx
27. 1B‐adrenergic receptor