Studies on pyrrolidinones. an improved synthesis of pyroglutamoyl chloride

Synthetic Communications

Volumn 24, Issue 18, 1994, Pages 2597-2607

  Rigo, BenoîT ^a   Ghammarti, Samira El ^a   Gautret, Philippe ^a   Couturier, Daniel ^b  

^a Ecole des Hautes Etudes d'Ingenieur   (France)

^b UNIV LILLE   (France)

Author keywords

[No Author keywords available]

Indexed keywords

AMINO ACID DERIVATIVE; PYROGLUTAMIC ACID DERIVATIVE; PYROGLUTAMOYL CHLORIDE; PYRROLIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG SYNTHESIS; INFRARED SPECTROPHOTOMETRY; NUCLEAR MAGNETIC RESONANCE; REACTION ANALYSIS;

EID: 0028050128     PISSN: 00397911     EISSN: 15322432     Source Type: Journal    
DOI: 10.1080/00397919408010572     Document Type: Article

References (36)

1. Rigo, B.; Cauliez, P.; Fasseur, D.; Sauvage, F.X.; Trends Heterocycl. Chem. 1991, 2, 155 and references cited therein.
2. Breda, A.; thesis, Lille, France, N° 77, 1967.
3. Effenberger, F.; Mü ller, W.; Isak, H.; Chem. Ber. 1987, 120, 45.
4. Mü ller, W.; Dorsch, W.; Effenberger, F.; Chem. Ber. 1987, 120, 55.
5. Abderhalden, E.; Suwa, A.; Ber. 1910, 43, 2.
6. Abderhalden, E.; Wurm, E.; Z. Physiol. Chem. 1912, 82, 160.
7. Thomas, Dr. Karl, G.m.b.H.; German Patent 2102 172, 1972;s
8. Chem. Abstr. 1972, 77, 151900j.
9. Pharmindustrie; Japan patent 80 45688, 1980;
10. Chem. Abstr. 1980, 93, 150112x.
11. Gibian, H.; Klieger, E.; Ann. Chem. 1961, 640, 145.
12. Lee, M.; Coulter, D.M.; Lowm, J.W.; J. Org. Chem. 1988, 53, 1855.
13. Flouret, G.; J. Med. Chem. 1970, 13, 843.
14. Poli Industria Chimica S.p.A.; European Patent 2767 52, 1988;
15. Chem. Abstr. 1988, 109, 190876e.
16. Capecchi, J.T.; Loudon, G.M.; J. Med. Chem. 1985, 8, 140.
17. IRE-Celltarg S.A.; European Patent 362031, 1990;
18. Chem. Abstr. 1990, 113, 132026z.
19. Angler, R.B.; Waller, C.W.; Hutchings, B.L.; Boothe, J.H.; Mowat, J.H.; Semb, J.; Subbarow, Y.; J. Am. Chem. Soc. 1950, 72, 74.
20. Colgate-Pallmolive Co.; U.S. Patent 3308157, 1967;
21. Chem. Abstr. 1967, 67, 43590t.
22. Sagami Chemical Research Center; Japan Patent 79119454, 1979;
23. Chem. Abstr. 1980, 92, 111291q.
24. Rigo, B., Lespagnol, C.; Pauly, M.J.; J. Heterocyclic Chem. 1988, 25, 59.
25. Haü s ler, J., Schmidt, U.; Chem. Ber. 1974, 107, 145.
26. Kricheldorf, H.R.; Liebigs Ann. Chem. 1971, 748, 101.
27. Domagala, J.H.; J. Org. Chem. 1984, 49, 126.
28. Raha, G.; Org. Synth., coll. Vol. 4, 263 (1963).
29. King, J.A.; Mc Millan, F.H.; J. Am. Chem. Soc. 1952, 74, 2859.
30. Beecham, A.F.; J. Am. Chem. Soc. 1954, 76, 4613.
31. Kolocouris, N.; Bull. Soc. Chim. France, 1973, 1053.
32. Rigo, B.; Kolocouris N.; J. Heterocyclic Chem., 1983, 20, 893.
33. Fritz, H.; Sutter, P.; Weis, C. D.; J. Org. Chem. 1986, 51, 558.
34. Pigache, P.; French Patent 1517 697, 1968;
35. Chem. Abstr., 1969, 71, 3267u.
36. Rigo, B.; Lespagnol, C.; Pauly, M.; J. Heterocyclic Chem., 1988, 25, 49.