A chemoselective approach to functionalize the C-10 position of 10-deacetylbaccatin III. Synthesis and biological properties of novel C-10 Taxol® analogues

Tetrahedron Letters

Volumn 35, Issue 31, 1994, Pages 5543-5546

  Kant, Joydeep ^a   O'Keeffe, Wendy S ^a   Chen, Shu Hui ^a   Farina, Vittorio ^a   Fairchild, Craig ^a,b   Johnston, Kathy ^a,b   Kadow, John F ^a   Long, Byron H ^a,b   Vyas, Dolatrai ^a  

^a BRISTOL MYERS SQUIBB   (United States)

^b BRISTOL MYERS SQUIBB PHARMACEUTICAL RESEARCH INSTITUTE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BACCATIN III; CARBAMIC ACID DERIVATIVE; CARBONIC ACID DERIVATIVE; DIMETHYL ETHER; DOCETAXEL; DRUG ANALOG; ESTER DERIVATIVE; ETHER DERIVATIVE; FUNCTIONAL GROUP; HYDROXYL GROUP; ISOSERINE; PACLITAXEL; SULFONIC ACID DERIVATIVE; TUBULIN;

ACETYLATION; ANTINEOPLASTIC ACTIVITY; ARTICLE; CELL DIVISION; CYTOTOXICITY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; HYDROGEN BOND; MICROTUBULE ASSEMBLY; OVARY CARCINOMA;

EID: 0027981391     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(00)77242-X     Document Type: Article

References (19)

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