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Bioorganic and Medicinal Chemistry Letters

Volumn 4, Issue 15, 1994, Pages 1795-1800

Dual metalloprotease inhibitors. II. Effect of substitution and stereochemistry on benzazepinone based mercaptoacetyls

(13) Robl, Jeffrey A a Simpkins, Ligaya M a Sulsky, Richard a Sieber McMaster, Ellen a Stevenson, Jay a Kelly, Yolanda F a Sun, Chong Qing a Misra, Raj N a Ryono, Denis E a Asaad, Magdi M a Bird, J Eileen a Trippodo, Nick C a Karanewsky, Donald S a

a BRISTOL MYERS SQUIBB (United States)

Author keywords

[No Author keywords available]

Indexed keywords

1,3,4,5 TETRAHYDRO 3 MERCAPTOACETAMIDO 2 OXO 1 BENZAZEPINEACETIC ACID; BENZAZEPINE DERIVATIVE; DIPEPTIDYL CARBOXYPEPTIDASE; DIPEPTIDYL CARBOXYPEPTIDASE INHIBITOR; ENZYME INHIBITOR; MEMBRANE METALLOENDOPEPTIDASE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; ENZYME INHIBITION; INTRAVENOUS DRUG ADMINISTRATION; NONHUMAN; PRESSOR RESPONSE; RAT; STEREOCHEMISTRY; STRUCTURE ACTIVITY RELATION;

EID: 0027966939 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(01)80373-5 Document Type: Article

Times cited : (32)

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