Effects of fluoxetine given chronically on the responsiveness of 5-HT receptor subpopulations to their agonists

European Neuropsychopharmacology

Volumn 3, Issue 2, 1993, Pages 85-94

  Maj, J ^a   Moryl, E ^a  

^a INSTITUTE OF PHARMACOLOGY   (Poland)

Author keywords

5 Hydroxytryptamine receptor subpopulations; Fluoxetine; Mice; Rats

Indexed keywords

2 DIPROPYLAMINO 8 HYDROXYTETRALIN; CPP; FENFLURAMINE; FLUOXETINE; SEROTONIN RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; BEHAVIOR; HYPERTHERMIA; INTRAPERITONEAL DRUG ADMINISTRATION; MALE; MOUSE; NONHUMAN; PRIORITY JOURNAL; RAT;

5-HYDROXYTRYPTOPHAN; 8-HYDROXY-2-(DI-N-PROPYLAMINO)TETRALIN; ANIMAL; BEHAVIOR, ANIMAL; BODY TEMPERATURE; EXPLORATORY BEHAVIOR; FENFLURAMINE; FLUOXETINE; MALE; MICE; MOTOR ACTIVITY; PIPERAZINES; RATS; RATS, WISTAR; RECEPTORS, SEROTONIN; SEROTONIN AGONISTS;

EID: 0027849695     PISSN: 0924977X     EISSN: None     Source Type: Journal    
DOI: 10.1016/0924-977X(93)90259-O     Document Type: Article

References (44)

1. 2 receptor affinity is also influenced by other transmitters
2. Fluoxetine. A review of its pharmacodynamic and pharmacokinetic properties and therapeutic efficacy in depressive illness
3. Long-term 5-HT reuptake blockade, but not monoamine oxidase inhibition, decreases the function of terminal 5-HT autoreceptors: an electrophysiological study in rat brain
4. A method for assessing the effects of drugs on the central actions of 5-hydroxytryptamine
5. Tricyclic antidepressants: long-term treatment increases responsivity of rat forebrain neurons to serotonin
6. 2-mediated behavior in the rat following noradrenergic or serotonergic denervation
7. 1B binding sites
8. 1B) receptors
9. Chronic antidepressant treatment and central 5-HT synapses
10. 2 receptors
11. Presynaptic serotonin receptor-mediated response in mice attenuated by antidepressant drugs and electroconvulsive shock
12. Acute effects of atypical antidepressants on various receptors in the brain
13. 8-Hydroxy-2-(di-n-propylamino)-tetralin, 8-OH-DPAT, a potent and selective simplified ergot congener with central 5-HT-receptor stimulating activity
14. 5-Hydroxytryptamine receptors and effector coupling mechanisms in peripheral tissues
15. 1B recognition sites
16. Effects of chronic fluoxetine administration on serotonin metabolism
17. Chemistry and pharmacology of compounds related to 4-(4-hydroxy-4-phenyl-piperidino)-butyrophenone. Part IV. Influence of haloperidol (R-1625) and of chlorpromazine on the behaviour of rats in an unfamiliar ‘open field’ situation
18. 1C receptors
19. Hyperthermia induced by m-trifluoromethylphenylpiperazine (TFMPP) or m-chlorophenylpiperazine (m-CPP) in head adapted rats
20. Exploratory hypoactivity induced by m-trifluoromethylphenylpiperazine (TFMPP) and m-chlorophenylpiperazine (m-CPP)
21. The use of specific serotonin uptake inhibitors as antidepressants
22. Central serotoninmimetic action of phenylpiperazines
23. Effects of sertraline and citalopram given repeatedly on the responsiveness of 5-HT receptor subpopulations
24. 1B receptors?
25. 1 recognition site
26. Molecular pharmacology of 5-HT-uptake inhibitors
27. 1A receptor antagonists on 8-OH-DPAT-induced hypothermia in rats and mice
28. Different action of 5-hydroxytryptamine (5-HT) uptake inhibitors on fenfluramine- but not p-chloroamphetamine-induced hyperthermia in rats
29. Zimelidine and clomipramine: different influence on fenfluramine but not p-chloroamphetamine-induced pharmacological effects
30. 2 receptor antagonist
31. Long-term antidepressant treatment decreases spiroperidol-labeled serotonin receptor binding
32. 3H]-spiperone binding in rat frontal cortex and serotonin receptor mediated behaviour
33. Antagonism of fenfluramine-induced hyperthermia in rats by some, but not all, selective inhibitors of 5-hydroxytryptamine uptake
34. Antagonism of fenfluramine-induced hypothermia: a measure of central serotonin inhibition
35. Biochemical effects of the antidepressant paroxetine, a specific 5-hydroxytryptamine uptake inhibitor
36. 1 receptor and of the catecholaminergic system in the behavioral response to 8-hydroxy-2(di-n-propylamino)tetralin in the rat
37. The relationship between response to fluoxetine plasma levels, imipramine binding to platelet membranes and whole-blood 5-HT
38. 1 receptors in the vertebrate brain. Regional distribution examined by autoradiography
39. Fluoxetine: a specific serotonin uptake inhibitor being studied in depression
40. 1A receptors in rat brain following antidepressant drug treatment
41. A selective inhibitor of serotonin uptake: Lilly 110140 3-(p-trifluoromethylphenoxy)-N-methyl-3-phenylpropylamine
42. Chronic effects of fluoxetine a selective inhibitor of serotonin uptake on neurotransmitter receptors
43. Affinities of fluoxetine, its enantiomers, and other inhibitors of serotonin uptake for subtypes of serotonin receptors
44. The behavioural effects of 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH-DPAT) in mice