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Volumn 21, Issue 4, 1993, Pages 587-594

Reversible tripeptide thrombin inhibitors as adjunctive agents to coronary thrombolysis: A comparison with heparin in a canine model of coronary artery thrombosis

Author keywords

Adjunct; Heparin; LY294468; Rethrombosis; Thrombin; Thrombolysis

Indexed keywords

ALTEPLASE; EFEGATRAN; HEMOGLOBIN; HEPARIN; LY 178207; TERT BUTOXYCARBONYL DEXTRO PHENYLALANYLPROLYLARGINAL; THROMBIN; THROMBIN INHIBITOR; TISSUE PLASMINOGEN ACTIVATOR; UNCLASSIFIED DRUG;

EID: 0027407160     PISSN: 01602446     EISSN: 15334023     Source Type: Journal    
DOI: 10.1097/00005344-199304000-00012     Document Type: Article
Times cited : (29)

References (34)
  • 1
    • 0022655051 scopus 로고
    • Intravenous recombinant tissue-type plasminogen activator in patients with acute myocardial infarction: A report from the NHLBI thrombolysis in myocardial infarction trial
    • William DO, Borer J, Braunwald E, et al. Intravenous recombinant tissue-type plasminogen activator in patients with acute myocardial infarction: a report from the NHLBI thrombolysis in myocardial infarction trial. Circulation 1986; 73:338-46.
    • (1986) Circulation , vol.73 , pp. 338-346
    • William, D.O.1    Borer, J.2    Braunwald, E.3
  • 2
    • 0025892010 scopus 로고
    • Is thrombolysis alone the best therapy for acute myocardial infarction?
    • Golino P, Willerson JT. Is thrombolysis alone the best therapy for acute myocardial infarction? Tex Heart Institute J 1991;18:50-61.
    • (1991) Tex Heart Institute J , vol.18 , pp. 50-61
    • Golino, P.1    Willerson, J.T.2
  • 3
    • 0023749096 scopus 로고
    • Influence of selective endoperoxide/thromboxane A2 receptor antagonism with sulotroban on lysis time and reocclusion rate after tissue plasminogen activator-induced coronary thrombolysis in the dog
    • Shebuski RJ, Smith JM, Storer BL, Granett JR, Bugelski PJ. Influence of selective endoperoxide/thromboxane A2 receptor antagonism with sulotroban on lysis time and reocclusion rate after tissue plasminogen activator-induced coronary thrombolysis in the dog. J Pharmacol Exp Ther 1988;246: 790-6.
    • (1988) J Pharmacol Exp Ther , vol.246 , pp. 790-796
    • Shebuski, R.J.1    Smith, J.M.2    Storer, B.L.3    Granett, J.R.4    Bugelski, P.J.5
  • 4
    • 0024393955 scopus 로고
    • Role of thrombin and throm-boxane A2 in reocclusion following coronary thrombolysis with tissue-type plasminogen activator
    • Fitzgerald DJ, FitzGerald GA. Role of thrombin and throm-boxane A2 in reocclusion following coronary thrombolysis with tissue-type plasminogen activator. Proc Natl Acad Sci USA 1989;86:7585-9.
    • (1989) Proc Natl Acad Sci USA , vol.86 , pp. 7585-7589
    • Fitzgerald, D.J.1    FitzGerald, G.A.2
  • 5
    • 0024395124 scopus 로고
    • Effect of thromboxane antagonism on recanalization during streptokinase-induced thrombolysis in anesthetized monkeys
    • Schumacher WA, Heran CL. Effect of thromboxane antagonism on recanalization during streptokinase-induced thrombolysis in anesthetized monkeys. J Cardiovasc Pharmacol 1989;13:853-61.
    • (1989) J Cardiovasc Pharmacol , vol.13 , pp. 853-861
    • Schumacher, W.A.1    Heran, C.L.2
  • 6
    • 0025187574 scopus 로고
    • Endogenous prostaglandin endoperoxides and prostacyclin modulate the thrombolytic activity of tissue plasminogen activator
    • Golino P, Rosolowsky M, Yao S-K, et al. Endogenous prostaglandin endoperoxides and prostacyclin modulate the thrombolytic activity of tissue plasminogen activator. J Clin Invest 1990;86:1095-102.
    • (1990) J Clin Invest , vol.86 , pp. 1095-1102
    • Golino, P.1    Rosolowsky, M.2    Yao, S.-K.3
  • 7
    • 0024514676 scopus 로고
    • Simultaneous administration of thromboxane A2- and serotonin S2-receptor antagonists markedly enhances thrombolysis and prevents or delays reocclusion after tissue-type plasminogen activator in a canine model of coronary thrombosis
    • Golino P, Ashton JH, McNatt J, et al. Simultaneous administration of thromboxane A2- and serotonin S2-receptor antagonists markedly enhances thrombolysis and prevents or delays reocclusion after tissue-type plasminogen activator in a canine model of coronary thrombosis. Circulation 1989;79: 911-9.
    • (1989) Circulation , vol.79 , pp. 911-919
    • Golino, P.1    Ashton, J.H.2    McNatt, J.3
  • 8
    • 0020619733 scopus 로고
    • A murine monoclonal antibody that completely blocks binding of fibrinogen to platelets produces a thrombasthenic-like state in normal platelets and binds to glycoproteins lib and/or Ilia
    • Coller BS, Peershke EI, Scudder LE, Sullivan CA. A murine monoclonal antibody that completely blocks binding of fibrinogen to platelets produces a thrombasthenic-like state in normal platelets and binds to glycoproteins lib and/or Ilia. J Clin Invest 1983;72:325-38.
    • (1983) J Clin Invest , vol.72 , pp. 325-338
    • Coller, B.S.1    Peershke, E.I.2    Scudder, L.E.3    Sullivan, C.A.4
  • 9
    • 0023893546 scopus 로고
    • Monoclonal antibody against the platelet glycoprotein (GP) IIb/IIIa receptor prevents coronary artery reocclusion after reperfusion with re-combinant tissue-type plasminogen activator in dogs
    • Yasuda T, Gold HK, Fallon JT, et al. Monoclonal antibody against the platelet glycoprotein (GP) IIb/IIIa receptor prevents coronary artery reocclusion after reperfusion with re-combinant tissue-type plasminogen activator in dogs. J Clin Invest 1988;81:1284-91.
    • (1988) J Clin Invest , vol.81 , pp. 1284-1291
    • Yasuda, T.1    Gold, H.K.2    Fallon, J.T.3
  • 10
    • 0023637601 scopus 로고
    • New perspectives in cell adhesion: RGD and integrins
    • Ruoslahti E, Perschbacher MD. New perspectives in cell adhesion: RGD and integrins. Science 1987;238:491-7.
    • (1987) Science , vol.238 , pp. 491-497
    • Ruoslahti, E.1    Perschbacher, M.D.2
  • 11
    • 0024829663 scopus 로고
    • Prevention of re-occluding platelet-rich thrombi in canine femoral arteries with a novel peptide antagonist of platelet glycoprotein IIb/IIIa receptors
    • Haskel EJ, Adams SP, Feigen LP, et al. Prevention of re-occluding platelet-rich thrombi in canine femoral arteries with a novel peptide antagonist of platelet glycoprotein IIb/IIIa receptors. Circulation 1989;80:1775-82.
    • (1989) Circulation , vol.80 , pp. 1775-1782
    • Haskel, E.J.1    Adams, S.P.2    Feigen, L.P.3
  • 12
    • 0025350512 scopus 로고
    • Acceleration of recombinant tissue-type plasminogen activator-induced thrombolysis and prevention of reocclusion by the combination of heparin and the Arg-Gly-Asp-containing peptide bitistatin in a canine model of coronary thrombosis
    • Shebuski RJ, Stabilito IJ, Sitko GR, Polokoff MH. Acceleration of recombinant tissue-type plasminogen activator-induced thrombolysis and prevention of reocclusion by the combination of heparin and the Arg-Gly-Asp-containing peptide bitistatin in a canine model of coronary thrombosis. Circulation 1990;82:169-77.
    • (1990) Circulation , vol.82 , pp. 169-177
    • Shebuski, R.J.1    Stabilito, I.J.2    Sitko, G.R.3    Polokoff, M.H.4
  • 13
    • 0026020072 scopus 로고
    • Kistrin, a polypeptide platelet GP IIb/IIIa receptor antagonist, enhances and sustains coronary arterial thrombolysis with recombinant tissue-type plasminogen activator in a canine preparation
    • Yasuda T, Gold HK, Leinbach RC, et al. Kistrin, a polypeptide platelet GP IIb/IIIa receptor antagonist, enhances and sustains coronary arterial thrombolysis with recombinant tissue-type plasminogen activator in a canine preparation. Circulation 1991;83:1038-47.
    • (1991) Circulation , vol.83 , pp. 1038-1047
    • Yasuda, T.1    Gold, H.K.2    Leinbach, R.C.3
  • 16
    • 0025179224 scopus 로고
    • Role of thrombolysis and thrombin in patients with acute coronary occlusion during percutaneous transluminal coronary angioplasty
    • Gulba DC, Daniel WG. Simon R. et al. Role of thrombolysis and thrombin in patients with acute coronary occlusion during percutaneous transluminal coronary angioplasty. J Am Coll Cardiol 1990:16:563-8.
    • (1990) J Am Coll Cardiol , vol.16 , pp. 563-568
    • Gulba, D.C.1    Daniel, W.G.2    Simon, R.3
  • 17
    • 0025563384 scopus 로고
    • Hirudin, heparin, and placebo during deep arterial injury in the pig
    • Heras M, Chesebro JH, Webster MWI, et al. Hirudin, heparin, and placebo during deep arterial injury in the pig. Circulation 1990;82:1476-84.
    • (1990) Circulation , vol.82 , pp. 1476-1484
    • Heras, M.1    Chesebro, J.H.2    Webster, M.W.I.3
  • 18
    • 0024411829 scopus 로고
    • Thrombin is an important mediator of platelet aggregation in stenosed canine coronary arteries with endothelial injury
    • Eidt JF, Allison P, Noble S, et al. Thrombin is an important mediator of platelet aggregation in stenosed canine coronary arteries with endothelial injury. J Clin Invest 1989;84:18-27.
    • (1989) J Clin Invest , vol.84 , pp. 18-27
    • Eidt, J.F.1    Allison, P.2    Noble, S.3
  • 20
    • 0025100680 scopus 로고
    • Heparin-resistant thrombus formation by endovascular stents in baboons. Interruption by a synthetic antithrombin
    • Krupski WC, Bass A, Kelly AB, Marzec UM, Hanson SR, Harker LA. Heparin-resistant thrombus formation by endovascular stents in baboons. Interruption by a synthetic antithrombin. Circulation 1990;81:570-7.
    • (1990) Circulation , vol.81 , pp. 570-577
    • Krupski, W.C.1    Bass, A.2    Kelly, A.B.3    Marzec, U.M.4    Hanson, S.R.5    Harker, L.A.6
  • 21
    • 0025676311 scopus 로고
    • Prevention of reocclusion by MCI-9038, a thrombin inhibitor, following t-PA-induced thrombolysis in a canine model of femoral arterial thrombosis
    • Mellot MJ, Connolly TM, York SJ, Bush LR. Prevention of reocclusion by MCI-9038, a thrombin inhibitor, following t-PA-induced thrombolysis in a canine model of femoral arterial thrombosis. Thromb Haemost 1990;64:526-34.
    • (1990) Thromb Haemost , vol.64 , pp. 526-534
    • Mellot, M.J.1    Connolly, T.M.2    York, S.J.3    Bush, L.R.4
  • 22
    • 0025143892 scopus 로고
    • Comparative effects of aspirin, a synthetic thrombin inhibitor and a monoclonal antiplatelet glycoprotein Hb/IIIa antibody on coronary artery reperfusion, reocclusion and bleeding with recombinant tissue-type plasminogen activator in a canine preparation
    • Yasuda T, Gold HK, Yaoita H, et al. Comparative effects of aspirin, a synthetic thrombin inhibitor and a monoclonal antiplatelet glycoprotein Hb/IIIa antibody on coronary artery reperfusion, reocclusion and bleeding with recombinant tissue-type plasminogen activator in a canine preparation. J Am Coll Cardiol 1990;16:714-22.
    • (1990) J Am Coll Cardiol , vol.16 , pp. 714-722
    • Yasuda, T.1    Gold, H.K.2    Yaoita, H.3
  • 23
    • 0026099431 scopus 로고
    • Relative efficacy of antithrombin compared with antiplatelet agents in accelerating coronary thrombolysis and preventing early reocclusion
    • Haskel EJ, Prager NA, Sobel BE, Abendschein DR. Relative efficacy of antithrombin compared with antiplatelet agents in accelerating coronary thrombolysis and preventing early reocclusion. Circulation 1991;83:1048-56.
    • (1991) Circulation , vol.83 , pp. 1048-1056
    • Haskel, E.J.1    Prager, N.A.2    Sobel, B.E.3    Abendschein, D.R.4
  • 24
    • 0026558347 scopus 로고
    • Conjunctive enhancement of enzymatic thrombolysis and prevention of thrombotic reocclusion with selective factor Xa inhibitor, tick anticoagulant peptide: Comparison to hirudin and heparin in a canine model of acute coronary artery thrombosis
    • Sitko GR, Ramjit DR, Stabilito II, Lehman D, Lynch JJ, Vlasuk GP. Conjunctive enhancement of enzymatic thrombolysis and prevention of thrombotic reocclusion with selective factor Xa inhibitor, tick anticoagulant peptide: comparison to hirudin and heparin in a canine model of acute coronary artery thrombosis. Circulation 1992;85:805-15.
    • (1992) Circulation , vol.85 , pp. 805-815
    • Sitko, G.R.1    Ramjit, D.R.2    Stabilito, I.I.3    Lehman, D.4    Lynch, J.J.5    Vlasuk, G.P.6
  • 25
    • 0026651846 scopus 로고
    • Pharmacological assessment of the antithrombotic activity of the peptide thrombin inhibitor, D-methyl-phenylalanyl-prolyl-arginal (GYKI-14766), in a canine model of coronary artery thrombosis
    • Jackson CV, Crowe VG, Frank JD, et al. Pharmacological assessment of the antithrombotic activity of the peptide thrombin inhibitor, D-methyl-phenylalanyl-prolyl-arginal (GYKI-14766), in a canine model of coronary artery thrombosis. J Pharmacol Exp Ther 1992;261:546-52.
    • (1992) J Pharmacol Exp Ther , vol.261 , pp. 546-552
    • Jackson, C.V.1    Crowe, V.G.2    Frank, J.D.3
  • 26
    • 0025111362 scopus 로고
    • Thrombolytic activity of a novel plasminogen activator, LY210825, compared with recombinant tissue-type plasminogen activator in a canine model of coronary artery thrombosis
    • Jackson CV, Crowe VG, Craft TJ, et al. Thrombolytic activity of a novel plasminogen activator, LY210825, compared with recombinant tissue-type plasminogen activator in a canine model of coronary artery thrombosis. Circulation 1990;82:930-40.
    • (1990) Circulation , vol.82 , pp. 930-940
    • Jackson, C.V.1    Crowe, V.G.2    Craft, T.J.3
  • 27
    • 0025146426 scopus 로고
    • Clot-bound thrombin is protected from inhibition by heparin-antithrombin III but is susceptible to inactivation by antithrombin Ill-independent inhibitors
    • Weitz JI, Hudoba M, Massel D, Maraganore J, Hirsh J. Clot-bound thrombin is protected from inhibition by heparin-antithrombin III but is susceptible to inactivation by antithrombin Ill-independent inhibitors. J Clin Invest 1990;86: 385-91.
    • (1990) J Clin Invest , vol.86 , pp. 385-391
    • Weitz, J.I.1    Hudoba, M.2    Massel, D.3    Maraganore, J.4    Hirsh, J.5
  • 28
    • 0025328906 scopus 로고
    • Highly active and selective anticoagulants: D-Phe-Pro-Arg-H, a free tripeptide aldehyde prone to spontaneous inactivation, and its stable N-methyl derivative, D-MePhe-Pro-Arg-H
    • Bajusz S, Szell E, Badgy D, et al. Highly active and selective anticoagulants: D-Phe-Pro-Arg-H, a free tripeptide aldehyde prone to spontaneous inactivation, and its stable N-methyl derivative, D-MePhe-Pro-Arg-H. J Med Chem 1990;33: 1729-35.
    • (1990) J Med Chem , vol.33 , pp. 1729-1735
    • Bajusz, S.1    Szell, E.2    Badgy, D.3
  • 30
    • 0017252128 scopus 로고
    • Human platelet factor 4; purification and characterization by affinity chromatography
    • Levine SP, Wohl H. Human platelet factor 4; purification and characterization by affinity chromatography. J Biol Chem 1976;251:324-8.
    • (1976) J Biol Chem , vol.251 , pp. 324-328
    • Levine, S.P.1    Wohl, H.2
  • 31
    • 0017154001 scopus 로고
    • Purification and binding properties of human platelet factor four
    • Handin RI, Cohen HJ. Purification and binding properties of human platelet factor four. J Biol Chem 1976;251:4273-82.
    • (1976) J Biol Chem , vol.251 , pp. 4273-4282
    • Handin, R.I.1    Cohen, H.J.2
  • 32
    • 0025174706 scopus 로고
    • Inhibition of coagulation and thrombin-induced platelet activities by a synthetic dodecapeptide modeled on the carboxyterminus of hirudin
    • Jakubowski JA, Maraganore JM. Inhibition of coagulation and thrombin-induced platelet activities by a synthetic dodecapeptide modeled on the carboxyterminus of hirudin. Blood 1990;75:399-406.
    • (1990) Blood , vol.75 , pp. 399-406
    • Jakubowski, J.A.1    Maraganore, J.M.2
  • 33
    • 0024670167 scopus 로고
    • Fibrin monomer protects thrombin from inactivation by heparin-antithrombin III: Implications for heparin efficacy
    • Hoog PJ, Jackson CM. Fibrin monomer protects thrombin from inactivation by heparin-antithrombin III: implications for heparin efficacy. Proc Natl Acad Sci USA 1989;86:3619-23.
    • (1989) Proc Natl Acad Sci USA , vol.86 , pp. 3619-3623
    • Hoog, P.J.1    Jackson, C.M.2
  • 34
    • 0025242653 scopus 로고
    • Enhancing effect by heparin on shear-induced platelet aggregation
    • Kawano K, Ikeda Y, Handa M, et al. Enhancing effect by heparin on shear-induced platelet aggregation. Sem Thromb Haemost 1990;16:60-5.
    • (1990) Sem Thromb Haemost , vol.16 , pp. 60-65
    • Kawano, K.1    Ikeda, Y.2    Handa, M.3


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