Peripheral biological activity of SR 27897: a new potent non-peptide antagonist of CCKA receptors

European Journal of Pharmacology

Volumn 232, Issue 1, 1993, Pages 13-19

  Gully, Danielle ^b   Fréhel, Daniel ^b   Marcy, Claudine ^b   Spinazzé, Arlette ^b   Lespy, Liliane ^b   Neliat, Gervais ^a   Maffrand, Jean Pierre ^b   Le Fur, Gérard ^b  

^a SANOFI   (France)

^b CEREP

Author keywords

Amylase secretion; CCKA receptors; Gall bladder emptying; Gastric emptying; SR 27897

Indexed keywords

[2 [[4 (2 CHLOROPHENYL) 2 THIAZOLYL]AMINOCARBONYL] 1 INDOLYL]ACETIC ACID; CHOLECYSTOKININ; CHOLECYSTOKININ A RECEPTOR; CHOLECYSTOKININ B RECEPTOR; CHOLECYSTOKININ RECEPTOR BLOCKING AGENT; DEVAZEPIDE; GASTRIN; LINTITRIPT; RADIOLIGAND; UNCLASSIFIED DRUG;

ACINAR CELL; AMYLASE RELEASE; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; FEMALE; GALLBLADDER EMPTYING; GUINEA PIG; INTRAVENOUS DRUG ADMINISTRATION; LIGAND BINDING; MALE; MOUSE; NONHUMAN; ORAL DRUG ADMINISTRATION; PANCREAS; PRIORITY JOURNAL; RAT; STOMACH EMPTYING; SUBCUTANEOUS DRUG ADMINISTRATION;

ADMINISTRATION, ORAL; AMYLASES; ANIMAL; BENZODIAZEPINONES; BINDING, COMPETITIVE; CHOLECYSTOKININ; COMPARATIVE STUDY; DEVAZEPIDE; DOSE-RESPONSE RELATIONSHIP, DRUG; FEMALE; GALLBLADDER; GASTRIC EMPTYING; GASTRINS; GUINEA PIGS; IN VITRO; INDOLEACETIC ACIDS; INJECTIONS, INTRAVENOUS; MALE; MICE; PANCREAS; RADIOLIGAND ASSAY; RATS; RATS, WISTAR; RECEPTORS, CHOLECYSTOKININ; STOMACH; THIAZOLES;

EID: 0027393017     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/0014-2999(93)90722-T     Document Type: Article

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