Design of Potent Non-Peptide Competitive Antagonists of the Human Bradykinin B2 Receptor

Journal of Medicinal Chemistry

Volumn 36, Issue 17, 1993, Pages 2583-2584

  Salvino, Joseph M ^a   Seoane, Peter R ^a   Douty, Brent D ^a   Awad, Mohamad M A ^a   Dolle, Roland E ^a   Houck, Wayne T ^a   Faunce, David M ^a   Sawutz, David G ^a  

^a EASTMAN KODAK COMPANY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMINO ACID; BRADYKININ; BRADYKININ B2 RECEPTOR; RECEPTOR BLOCKING AGENT;

ANIMAL TISSUE; ARTICLE; BINDING SITE; DRUG DESIGN; DRUG POTENCY; DRUG STRUCTURE; GUINEA PIG; HYDROPHOBICITY; INFLAMMATION; NONHUMAN; PAIN; PRIORITY JOURNAL; RECEPTOR AFFINITY; RECEPTOR BLOCKING; STRUCTURE ACTIVITY RELATION;

AMINO ACID SEQUENCE; ANIMAL; BINDING, COMPETITIVE; GUINEA PIGS; HUMAN; MOLECULAR SEQUENCE DATA; MUSCLE CONTRACTION; MUSCLE, SMOOTH; NAPHTHALENES; ORGANOPHOSPHORUS COMPOUNDS; RATS; RECEPTORS, BRADYKININ; RECEPTORS, NEUROTRANSMITTER; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0027220896     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm00069a021     Document Type: Editorial

References (16)

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