CGP 52432: a novel potent and selective GABAB autoreceptor antagonist in rat cerebral cortex

European Journal of Pharmacology

Volumn 237, Issue 2-3, 1993, Pages 191-195

  Lanza, Marco ^a   Fassio, Anna ^a   Gemignani, Anita ^a   Bonanno, Giambattista ^a   Raiteri, Maurizio ^a  

^a UNIVERSITY OF GENOA   (Italy)

Author keywords

CGP 52432; GABA autoreceptors; GABA release; GABAB receptor subtypes; Glutamate release; Somatostatin release

Indexed keywords

4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID B RECEPTOR; 4 AMINOBUTYRIC ACID RECEPTOR BLOCKING AGENT; [3 (3,4 DICHLOROBENZYLAMINO)PROPYL](DIETHOXYMETHYL)PHOSPHINIC ACID; AUTORECEPTOR; BACLOFEN; GLUTAMIC ACID; POTASSIUM ION; RECEPTOR SUBTYPE; SOMATOSTATIN;

ANIMAL TISSUE; ARTICLE; BRAIN CORTEX; BRAIN SYNAPTOSOME; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG ANTAGONISM; MALE; NEUROTRANSMITTER RELEASE; NONHUMAN; PRIORITY JOURNAL; RAT;

ANIMAL; BACLOFEN; BENZYLAMINES; CEREBRAL CORTEX; GAMMA-AMINOBUTYRIC ACID; GLUTAMATES; GLUTAMIC ACID; IN VITRO; MALE; ORGANOPHOSPHORUS COMPOUNDS; RATS; RATS, WISTAR; RECEPTORS, GABA-A; SOMATOSTATIN; SUPPORT, NON-U.S. GOV'T;

EID: 0027162802     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/0014-2999(93)90268-M     Document Type: Article

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