A versatile approach to 2,3-disubstituted indoles through the palladium-catalysed cyclization of o-alkynyltrifluoroacetanilides with vinyl triflates and aryl halides.

Tetrahedron Letters

Volumn 33, Issue 27, 1992, Pages 3915-3918

  Antonio, Arcadi ^a   Sandro, Cacchi ^b   Fabio, Marinelli ^a  

^a UNIVERSITY OF L'AQUILA   (Italy)

^b SAPIENZA UNIVERSITY OF ROME   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

INDOLE DERIVATIVE; PALLADIUM;

ARTICLE; CHEMICAL PROCEDURES; PRIORITY JOURNAL; REACTION ANALYSIS; SYNTHESIS;

EID: 0026769043     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(00)74818-0     Document Type: Article

References (16)

1. Transition Metals in the Synthesis and Functionalization of Indoles [New Synthesis Methods (72)]
2. Condensed Heteroaromatic Ring Systems; XVII:1Palladium-Catalyzed Cyclization of β-(2-Halophenyl)amino Substituted α,β-Unsaturated Ketones and Esters to 2,3-Disubstituted Indoles