Approaches to the synthesis of endothiopeptides: Synthesis of a thioamide-containing C-terminal bombesin nonapeptide

Tetrahedron

Volumn 48, Issue 40, 1992, Pages 8601-8614

  Jurayj, Jurjus ^a   Cushman, Mark ^a  

^a PURDUE UNIVERSITY   (United States)

Author keywords

bombesin.; Dithioester; endothiopeptide; epimerization; thioacylation; thioamide

Indexed keywords

BOMBESIN DERIVATIVE;

ARTICLE; PEPTIDE SYNTHESIS;

EID: 0026714007     PISSN: 00404020     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4020(01)89436-9     Document Type: Article

References (41)

1. Studies on amino acids and peptides. Part 6. Methods for introducing thioamide bonds into the peptide backbone: synthesis of the four monothio analogues of leucine enkephalin
2. 2,4-Bis(4-methylpheylthio)-1,3,2?5,4?5-dithiadiphosphetan-2,4-dithion: Ein neues Reagens zur Schwefelung vonN,N-disubstituierten Amiden
3. �ber die Verwendung von Dicyclohexylcarbodiimid/3-Hydroxy-4-oxo-3,4-dihydro-chinazolin f�r die Synthese des C-terminalen Hexapeptidamids von Substanz P
4. Peptide Coupling Reagents; VIII. A High Yield Preparation of Phenyl Esters of Amino Acids using Benzotriazolyloxytris[dimethylamino]phosphonium Hexafluorophosphate (BOP Reagent)
5. New Aspects of Dithio and Thiono Esters
6. Peptide Coupling Reagents VI1. A Novel, Cheaper Preparation of Benzotriazolyloxytris[dimethylamino]phosphonium Hexafluorophosphate (BOP Reagent)
7. Polypeptides. Part IV. Syntheses of human gastrin (HI)