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International Journal of Peptide and Protein Research

Volumn 39, Issue 2, 1992, Pages 131-136

Synthesis and biological activities of linear and cyclic enkephalin analogues containing a Ψ (E,CH=CH) or Ψ (CH2CH2) isosteric replacement

(11) TOURWE D a COUDER, J a CEUSTERS, M a MEERT, D a BURKS, T F b KRAMER, T H b DAVIS, P b KNAPP, R b YAMAMURA, H I b LEYSEN, J E c VAN BINST, G a

a VRIJE UNIVERSITEIT BRUSSEL (Belgium)

b UNIVERSITY OF ARIZONA (United States)

c JANSSEN RESEARCH FOUNDATION (Belgium)

Author keywords

double bond isosteres; enantioselective synthesis; enkephalin analogues; single bond isosteres; structure activity

Indexed keywords

CYCLOPEPTIDE; ENKEPHALIN DERIVATIVE; ENKEPHALIN[2 DEXTRO ALANINE 5 DEXTRO LEUCINE]; ENKEPHALIN[2,5 DEXTRO PENICILLAMINE];

ANIMAL TISSUE; ARTICLE; ILEUM; MOUSE; NONHUMAN; PEPTIDE SYNTHESIS; SMOOTH MUSCLE CONTRACTION; STRUCTURE ACTIVITY RELATION; SWINE; VAS DEFERENS;

AMINO ACID SEQUENCE; ANIMAL; ENKEPHALINS; GUINEA PIGS; IN VITRO; MAGNETIC RESONANCE SPECTROSCOPY; MALE; MICE; MOLECULAR SEQUENCE DATA; MOLECULAR STRUCTURE; MUSCLE CONTRACTION; PEPTIDES, CYCLIC; RATS; RECEPTORS, OPIOID; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0026549869 PISSN: 03678377 EISSN: 13993011 Source Type: Journal
DOI: 10.1111/j.1399-3011.1992.tb00782.x Document Type: Article

Times cited : (19)

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