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Volumn 84, Issue 23, 1992, Pages 1811-1816

High-dose oral tamoxifen, a potential multidrug-resistance-reversal agent: Phase I trial in combination with vinblastine

Author keywords

[No Author keywords available]

Indexed keywords

NORTAMOXIFEN; TAMOXIFEN; VINBLASTINE;

EID: 0026445750     PISSN: 00278874     EISSN: None     Source Type: Journal    
DOI: 10.1093/jnci/84.23.1811     Document Type: Article
Times cited : (223)

References (41)
  • 1
    • 0014767029 scopus 로고
    • Cellular resistance to actinomycin D in Chinese hamster cells in vitro: Cross-resistance, radioautographic, and cytogenetic studies
    • Biedler JL, Riehm H: Cellular resistance to actinomycin D in Chinese hamster cells in vitro: Cross-resistance, radioautographic, and cytogenetic studies. Cancer Res 30:1174-1184, 1970
    • (1970) Cancer Res , vol.30 , pp. 1174-1184
    • Biedler, J.L.1    Riehm, H.2
  • 2
    • 0015963429 scopus 로고
    • Reduced permeability in CHO cells as a mechanism of resistance to colchicine
    • Ling V, Thompson L: Reduced permeability in CHO cells as a mechanism of resistance to colchicine. J Cell Physiol 83:103-116, 1973
    • (1973) J Cell Physiol , vol.83 , pp. 103-116
    • Ling, V.1    Thompson, L.2
  • 3
    • 0017225040 scopus 로고
    • Pleio-tropic phenotype of colchicine-resistant CHO cells: Cross resistance and collateral sensitivity
    • Bech-Hansen NT, Till JE, Ling V: Pleio-tropic phenotype of colchicine-resistant CHO cells: Cross resistance and collateral sensitivity. J Cell Physiol 88:23-31, 1976
    • (1976) J Cell Physiol , vol.88 , pp. 23-31
    • Bech-Hansen, N.T.1    Till, J.E.2    Ling, V.3
  • 4
    • 0015893137 scopus 로고
    • Active outward transport of daunomycin in Ehrlich ascites tumor cells
    • Dano K: Active outward transport of daunomycin in Ehrlich ascites tumor cells. Biochim Biophys Acta 323:466-483, 1973
    • (1973) Biochim Biophys Acta , vol.32 , pp. 466-483
    • Dano, K.1
  • 5
    • 0020578356 scopus 로고
    • Cell surface P-glycoprotein associated with mul-tidrug resistance in mammalian cell lines
    • Kartner N, Riordan JR, Ling V: Cell surface P-glycoprotein associated with mul-tidrug resistance in mammalian cell lines. Science 221:1285-1288, 1983
    • (1983) Science , vol.22 , pp. 1285-1288
    • Kartner, N.1    Riordan, J.R.2    Ling, V.3
  • 6
    • 0008632564 scopus 로고
    • Expression of a full-length cDNA for the human MDR 1: Gene confers resistance to colchicine, doxorubicin and vinblastine
    • Ueda K, Cardarelli C, Gottesman MM, et al: Expression of a full-length cDNA for the human MDR 1: Gene confers resistance to colchicine, doxorubicin and vinblastine. Proc Natl Acad Sci U S A 84:3004-3008, 1987
    • (1987) Proc Natl Acad Sci U S A , vol.84 , pp. 3004-3008
    • Ueda, K.1    Cardarelli, C.2    Gottesman, M.M.3
  • 7
    • 0024506222 scopus 로고
    • Drug-resistance in multiple myeloma and non-Hodgkin’s lymphoma: Detection of P-glycoprotein and potential circumvention by addition of verapamil to chemotherapy
    • Dalton WS, Grogan TM, Meltzer PS, et al: Drug-resistance in multiple myeloma and non-Hodgkin’s lymphoma: Detection of P-glycoprotein and potential circumvention by addition of verapamil to chemotherapy. J Clin Oncol 7:415-424, 1989
    • (1989) J Clin Oncol , vol.7 , pp. 415-424
    • Dalton, W.S.1    Grogan, T.M.2    Meltzer, P.S.3
  • 8
    • 0023499815 scopus 로고
    • Intrinsic drug resistance in human kidney cancer is associated with expression of a human multidrug-resistance gene
    • Fojo AT, Shen D-W, Mickley LA, et al: Intrinsic drug resistance in human kidney cancer is associated with expression of a human multidrug-resistance gene. J Clin Oncol 5:1922-1927, 1987
    • (1987) J Clin Oncol , vol.5 , pp. 1922-1927
    • Fojo, A.T.1    Shen, D.-W.2    Mickley, L.A.3
  • 9
    • 0024538797 scopus 로고
    • Prediction of doxorubicin resistance in vitro in myeloma, lymphoma, and breast cancer by P-glycoprotein staining
    • Salmon SE, Grogan TM, Miller T, et al: Prediction of doxorubicin resistance in vitro in myeloma, lymphoma, and breast cancer by P-glycoprotein staining. J Natl Cancer Inst 81:696-701, 1989
    • (1989) J Natl Cancer Inst , vol.81 , pp. 696-701
    • Salmon, S.E.1    Grogan, T.M.2    Miller, T.3
  • 10
    • 0024548599 scopus 로고
    • Expression of a multidrug resistance gene in human cancers
    • Goldstein LJ, Galski H, Fojo A, et al: Expression of a multidrug resistance gene in human cancers. J Natl Cancer Inst 81: 116-124, 1989
    • (1989) J Natl Cancer Inst , vol.81 , pp. 116-124
    • Goldstein, L.J.1    Galski, H.2    Fojo, A.3
  • 11
    • 0021916585 scopus 로고
    • Detection of P-glycoprotein in ovarian cancer: A molecular marker associated with multidrug resistance
    • Bell DR, Gerlach JH, Kartner N, et al: Detection of P-glycoprotein in ovarian cancer: A molecular marker associated with multidrug resistance. J Clin Oncol 3:311-315, 1985
    • (1985) J Clin Oncol , vol.3 , pp. 311-315
    • Bell, D.R.1    Gerlach, J.H.2    Kartner, N.3
  • 12
    • 0023629183 scopus 로고
    • Amiodarone is more efficient than verapamil in reversing resistance to an-thracyclines in tumour cells
    • Chauffert B, Rey D, Coudert B, et al: Amiodarone is more efficient than verapamil in reversing resistance to an-thracyclines in tumour cells. Br J Cancer 56:119-122, 1987
    • (1987) Br J Cancer , vol.56 , pp. 119-122
    • Chauffert, B.1    Rey, D.2    Coudert, B.3
  • 13
    • 0023110246 scopus 로고
    • In vitro and in vivo enhancement of vincristine antitumor activity on B16 melanoma cells by calcium antagonist flunarizine
    • Bellelli A, Camboni C, DeLuca G, et al: In vitro and in vivo enhancement of vincristine antitumor activity on B16 melanoma cells by calcium antagonist flunarizine. Oncology 44:17-23, 1987
    • (1987) Oncology , vol.44 , pp. 17-23
    • Bellelli, A.1    Camboni, C.2    Deluca, G.3
  • 14
    • 0023871288 scopus 로고
    • The effects of verapamil and a tiapamil analogue, DMDP, on adriamycin-induced cytotoxicity in P388 adriamycin-resistant and -sensitive leukemia in vitro and in vivo
    • Radel S, Bankusli I, Mayhew E, et al: The effects of verapamil and a tiapamil analogue, DMDP, on adriamycin-induced cytotoxicity in P388 adriamycin-resistant and -sensitive leukemia in vitro and in vivo. Cancer Chemother Pharmacol 21:25-30, 1988
    • (1988) Cancer Chemother Pharmacol , vol.21 , pp. 25-30
    • Radel, S.1    Bankusli, I.2    Mayhew, E.3
  • 15
    • 0023237840 scopus 로고
    • Verapamil and adriamycin in the treatment of drug-resistant ovarian cancer patients
    • Ozols RF, Cunnion RE, Klecker RW Jr, et al: Verapamil and adriamycin in the treatment of drug-resistant ovarian cancer patients. J Clin Oncol 5:641-647, 1987
    • (1987) J Clin Oncol , vol.5 , pp. 641-647
    • Ozols, R.F.1    Cunnion, R.E.2    Klecker, R.W.3
  • 16
    • 0019430432 scopus 로고
    • Overcoming of vincristine resistance in P388 leukemia in vivo and in vitro through enhanced cytotoxicity of vincristine and vinblastine by verapamil
    • Tsuruo T, Iida H, Tsukagoshi S, et al: Overcoming of vincristine resistance in P388 leukemia in vivo and in vitro through enhanced cytotoxicity of vincristine and vinblastine by verapamil. Cancer Res 41:1967-1972, 1981
    • (1981) Cancer Res , vol.41 , pp. 1967-1972
    • Tsuruo, T.1    Iida, H.2    Tsukagoshi, S.3
  • 17
    • 0023691409 scopus 로고
    • Verapamil reversal of doxorubicin resistance in multidrug-resistant human myeloma cells and association with drug accumulation and DNA damage
    • Bellamy WT, Dalton WS, Kailey JM, et al: Verapamil reversal of doxorubicin resistance in multidrug-resistant human myeloma cells and association with drug accumulation and DNA damage. Cancer Res 48:6365-6370, 1988
    • (1988) Cancer Res , vol.48 , pp. 6365-6370
    • Bellamy, W.T.1    Dalton, W.S.2    Kailey, J.M.3
  • 18
    • 0023234519 scopus 로고
    • Certain calcium channel blockers bind specifically to multidrug-resistant human KB carcinoma membrane vesicles and inhibit drug binding to P-glycoprotein
    • Cornwell MM, Pastan I, Gottesman MM: Certain calcium channel blockers bind specifically to multidrug-resistant human KB carcinoma membrane vesicles and inhibit drug binding to P-glycoprotein. J Biol Chem 262:2166-2170, 1987
    • (1987) J Biol Chem , vol.26 , pp. 2166-2170
    • Cornwell, M.M.1    Pastan, I.2    Gottesman, M.M.3
  • 19
    • 0021924824 scopus 로고
    • A phase I study of vinblastine and verapamil given by concurrent iv infusion
    • Benson AB III, Trump DL, Koeller JM, et al: A phase I study of vinblastine and verapamil given by concurrent iv infusion. Cancer Treat Rep 69:795-799, 1985
    • (1985) Cancer Treat Rep , vol.69 , pp. 795-799
    • Benson, A.1    Trump, D.L.2    Koeller, J.M.3
  • 20
    • 0021259334 scopus 로고
    • Reversal of adriamycin resistance by verapamil in human ovarian cancer
    • Rogan AM, Hamilton TC, Young RC, et al: Reversal of adriamycin resistance by verapamil in human ovarian cancer. Science 224:994-996, 1984
    • (1984) Science , vol.22 , pp. 994-996
    • Rogan, A.M.1    Hamilton, T.C.2    Young, R.C.3
  • 21
    • 0026426153 scopus 로고
    • Systemic toxic effects associated with high-dose verapamil infusion and chemotherapy administration
    • Pennock GD, Dalton WS, Roeske WR, et al: Systemic toxic effects associated with high-dose verapamil infusion and chemotherapy administration. J Natl Cancer Inst 83:105-110, 1991
    • (1991) J Natl Cancer Inst , vol.83 , pp. 105-110
    • Pennock, G.D.1    Dalton, W.S.2    Roeske, W.R.3
  • 22
    • 0021162802 scopus 로고
    • Reversal of acquired resistance to doxorubicin in P388 murine leukemia cells by tamoxifen and other triparanol analogues
    • Ramu A, Glaubiger D, Fuks F: Reversal of acquired resistance to doxorubicin in P388 murine leukemia cells by tamoxifen and other triparanol analogues. Cancer Res 44:4392-4395, 1984
    • (1984) Cancer Res , vol.44 , pp. 4392-4395
    • Ramu, A.1    Glaubiger, D.2    Fuks, F.3
  • 23
    • 0025959561 scopus 로고
    • Effects of tamoxifen on cell lines displaying the multi-drug resistant phenotype
    • Berman E, Adams M, Duigou-Osterndorf R, et al: Effects of tamoxifen on cell lines displaying the multi-drug resistant phenotype. Blood 7:818-825, 1991
    • (1991) Blood , vol.7 , pp. 818-825
    • Berman, E.1    Adams, M.2    Duigou-Osterndorf, R.3
  • 24
    • 0343460160 scopus 로고
    • Intermittent high dose tamoxifen (HDT) with oral etoposide (EPO): Phase I and II clinical studies
    • Cantwell B, Carmichael J, Millward M, et al: Intermittent high dose tamoxifen (HDT) with oral etoposide (EPO): Phase I and II clinical studies. Proc ASCO 8:65, 1989
    • (1989) Proc ASCO , vol.8 , pp. 65
    • Cantwell, B.1    Carmichael, J.2    Millward, M.3
  • 25
    • 0011903190 scopus 로고
    • Tamoxifen potentiates the cytotoxicity of vinblastine by increasing intracellular drug accumulation
    • Fine RL, Sachs CW, Albers M, et al: Tamoxifen potentiates the cytotoxicity of vinblastine by increasing intracellular drug accumulation. Proc Am Assoc Cancer Res 32:375, 1991
    • (1991) Proc am Assoc Cancer Res , vol.32 , pp. 375
    • Fine, R.L.1    Sachs, C.W.2    Albers, M.3
  • 26
    • 0024459880 scopus 로고
    • Toremifene: Pharmacologic and pharmacokinetic basis of reversing multidrug resistance
    • DeGregorio MW, Ford JM, Benz CC, et al: Toremifene: Pharmacologic and pharmacokinetic basis of reversing multidrug resistance. J Clin Oncol 7:1359-1364, 1989
    • (1989) J Clin Oncol , vol.7 , pp. 1359-1364
    • Degregorio, M.W.1    Ford, J.M.2    Benz, C.C.3
  • 27
    • 0020676409 scopus 로고
    • Determination of tamoxifen and metabolites in human serum by high performance liquid chromatography with post-column fluorescence activation
    • Brown RR, Bain R, Jordan VC: Determination of tamoxifen and metabolites in human serum by high performance liquid chromatography with post-column fluorescence activation. J Chromatogr 272:351-358, 1983
    • (1983) J Chromatogr , vol.27 , pp. 351-358
    • Brown, R.R.1    Bain, R.2    Jordan, V.C.3
  • 28
    • 0019179910 scopus 로고
    • Clinical pharmacology of tamoxifen in patients with breast cancer: Comparison of traditional and loading dose schedules
    • Fabian C, Sternson L, Barnett M: Clinical pharmacology of tamoxifen in patients with breast cancer: Comparison of traditional and loading dose schedules. Cancer Treat Rep 64:765-773, 1980
    • (1980) Cancer Treat Rep , vol.64 , pp. 765-773
    • Fabian, C.1    Sternson, L.2    Barnett, M.3
  • 29
    • 0017028360 scopus 로고
    • Evaluation of tamoxifen dose in advanced breast cancer: A progress report
    • Tormey DC, Simon RM, Lippman ME, et al: Evaluation of tamoxifen dose in advanced breast cancer: A progress report. Cancer Treat Rep 60:1451-1459, 1976
    • (1976) Cancer Treat Rep , vol.60 , pp. 1451-1459
    • Tormey, D.C.1    Simon, R.M.2    Lippman, M.E.3
  • 30
    • 0023462787 scopus 로고
    • Controlled clinical trial of doxorubicin and tamoxifen versus doxorubicin alone in hepatocellular carcinoma
    • Melia WM, Johnson PJ, Williams R: Controlled clinical trial of doxorubicin and tamoxifen versus doxorubicin alone in hepatocellular carcinoma. Cancer Treat Rep 71:1213-1216, 1987
    • (1987) Cancer Treat Rep , vol.71 , pp. 1213-1216
    • Melia, W.M.1    Johnson, P.J.2    Williams, R.3
  • 31
    • 0022495689 scopus 로고
    • Cyclosporin A corrects daunorubicin resistance in Ehrlich ascites carcinoma
    • Slater LM, Sweet P, Stupecky M, et al: Cyclosporin A corrects daunorubicin resistance in Ehrlich ascites carcinoma. Br J Cancer 54:235-238, 1986
    • (1986) Br J Cancer , vol.54 , pp. 235-238
    • Slater, L.M.1    Sweet, P.2    Stupecky, M.3
  • 32
    • 26844556332 scopus 로고
    • Verapamil (V) and quinine (Q) chemo-sensitize myeloma cells to doxorubicin (DOX) and vincristine (VCR) in vitro and are capable of reversing clinical relapses in multiple myeloma (MM)
    • Salmon SE, Lehnert M, Grogan T, et al: Verapamil (V) and quinine (Q) chemo-sensitize myeloma cells to doxorubicin (DOX) and vincristine (VCR) in vitro and are capable of reversing clinical relapses in multiple myeloma (MM). Blood [Suppl] 74:197, 1989
    • (1989) Blood [Suppl] , vol.74 , pp. 197
    • Salmon, S.E.1    Lehnert, M.2    Grogan, T.3
  • 33
    • 0344102285 scopus 로고
    • The use of R-verapamil (R-VPM) is superior to racemic VPM in breaking multidrag resistance (MDR) of malignant cells
    • Keilhauer C, Emling F, Raschack M, et al: The use of R-verapamil (R-VPM) is superior to racemic VPM in breaking multidrag resistance (MDR) of malignant cells. Proc Am Assoc Cancer Res 30:503, 1989
    • (1989) Proc am Assoc Cancer Res , vol.30 , pp. 503
    • Keilhauer, C.1    Emling, F.2    Raschack, M.3
  • 34
    • 0008879750 scopus 로고
    • Phase I trial of multidrug resistance modulation with cyclosporin A
    • Samuels B, Ratain M, Mick R, et al: Phase I trial of multidrug resistance modulation with cyclosporin A. Proc Am Assoc Cancer Res 32:195, 1991
    • (1991) Proc am Assoc Cancer Res , vol.32 , pp. 195
    • Samuels, B.1    Ratain, M.2    Mick, R.3
  • 35
    • 0000829338 scopus 로고
    • Bilirubin: A physiological substrate for the multidrug transporter
    • Gosland MP, Brophy NA, Duran GE, et al: Bilirubin: A physiological substrate for the multidrug transporter. Proc Am Assoc Cancer Res 32:426, 1991
    • (1991) Proc am Assoc Cancer Res , vol.32 , pp. 426
    • Gosland, M.P.1    Brophy, N.A.2    Duran, G.E.3
  • 36
    • 0019813814 scopus 로고
    • Determination of tamoxifen and biologically active metabolites in human breast tumours and plasma
    • Daniel P, Gaskell SJ, Bishop H, et al: Determination of tamoxifen and biologically active metabolites in human breast tumours and plasma. Eur J Cancer Clin Oncol 17:1183-1189, 1981
    • (1981) Eur J Cancer Clin Oncol , vol.17 , pp. 1183-1189
    • Daniel, P.1    Gaskell, S.J.2    Bishop, H.3
  • 37
    • 0023501880 scopus 로고
    • Serum tamoxifen concentrations in the athymic nude mouse after three methods of administration
    • DeGregorio MW, Wilbur BJ, Coronado E, et al: Serum tamoxifen concentrations in the athymic nude mouse after three methods of administration. Cancer Chem-other Pharmacol 20:316-318, 1987
    • (1987) Cancer Chem-Other Pharmacol , vol.20 , pp. 316-318
    • Degregorio, M.W.1    Wilbur, B.J.2    Coronado, E.3
  • 38
    • 84969066360 scopus 로고
    • Modulation of vinblastine [VB] cytotoxicity by dipyridamole [DP] versus tamoxifen [TAM]: An in vivo preclinical study by subrenal capsule assay [SRCA] of human renal carcinoma [HRCC]
    • Keane TE, Rosner G, Walther PJ: Modulation of vinblastine [VB] cytotoxicity by dipyridamole [DP] versus tamoxifen [TAM]: An in vivo preclinical study by subrenal capsule assay [SRCA] of human renal carcinoma [HRCC]. Proc Am Assoc Cancer Res 31:376, 1990
    • (1990) Proc am Assoc Cancer Res , vol.31 , pp. 376
    • Keane, T.E.1    Rosner, G.2    Walther, P.J.3
  • 39
    • 0022591252 scopus 로고
    • Triphenylethylenes: A new class of protein kinase C inhibitors
    • O’Brian CA, Liskamp RM, Soloman DH, et al: Triphenylethylenes: A new class of protein kinase C inhibitors. JNCI 76:1243-1246, 1986
    • (1986) JNCI , vol.76 , pp. 1243-1246
    • O’Brian, C.A.1    Liskamp, R.M.2    Soloman, D.H.3
  • 40
    • 0023129529 scopus 로고
    • Calcium channel antagonist properties of antineoplastic antiestrogen. Tamoxifen in the PC12 neurosecretory cell line
    • Greenberg DA, Carpenter CL, Messing RO: Calcium channel antagonist properties of antineoplastic antiestrogen. Tamoxifen in the PC12 neurosecretory cell line. Cancer Res 47:70-74, 1987
    • (1987) Cancer Res , vol.47 , pp. 70-74
    • Greenberg, D.A.1    Carpenter, C.L.2    Messing, R.O.3
  • 41
    • 0023447098 scopus 로고
    • Cellular localization of the multidrug-resistance gene product P-glycoprotein in normal human tissues
    • Thiebaut F, Tsuruo T, Hamada H, et al: Cellular localization of the multidrug-resistance gene product P-glycoprotein in normal human tissues. Proc Natl Acad Sci USA 84:7735-7738, 1987
    • (1987) Proc Natl Acad Sci USA , vol.84 , pp. 7735-7738
    • Thiebaut, F.1    Tsuruo, T.2    Hamada, H.3


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