Inhibition of [3H]resiniferatoxin binding to rat dorsal root ganglion membranes as a novel approach in evaluating compounds with capsaicin-like activity

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 344, Issue 5, 1991, Pages 551-556

  Szallasi, Arpad ^a   Szolczanyi, Janos ^b   Szallasi, Zoltan ^a   Blumberg, Peter M ^a  

^a NATIONAL CANCER INSTITUTE   (United States)

^b UNIVERSITY OF PÉCS   (Hungary)

Author keywords

3H Resiniferatoxin binding; Capsaicin analogs; Resiniferatoxin analogs

Indexed keywords

CAPSAICIN; DITERPENE; DRUG DERIVATIVE; RESINIFERATOXIN; TINYATOXIN; 1 HOMOVANILLOYLPIPERIDINE; 12 DEOXYPHORBOL 13 PHENYLACETATE 20 HOMOVANILLATE; CAPSAICIN DERIVATIVE; DRUG RECEPTOR; N CYCLODODECYLHOMOVANILLAMIDE; N DECYLHOMOVANILLAMIDE; N DODECYLHOMOVANILLAMIDE; N HEXADECYLHOMOVANILLAMIDE; N VERATRYL 2 DECENAMIDE; RADIOISOTOPE; UNCLASSIFIED DRUG;

ANIMAL; ARTICLE; BINDING SITE; CELL MEMBRANE; DRUG INTERACTION; FEMALE; METABOLISM; MOUSE; RAT; RAT STRAIN; SPINAL GANGLION; STRUCTURE ACTIVITY RELATION; ANIMAL EXPERIMENT; ANIMAL TISSUE; BINDING COMPETITION; CONTROLLED STUDY; DRUG CONCENTRATION; HYPOTHERMIA; INFLAMMATION; NONHUMAN; PAIN; PRIORITY JOURNAL; SUBCUTANEOUS DRUG ADMINISTRATION; TOPICAL DRUG ADMINISTRATION;

ANIMAL; BINDING SITES; CAPSAICIN; CELL MEMBRANE; DITERPENES; DRUG INTERACTIONS; FEMALE; GANGLIA, SPINAL; MICE; RATS; RATS, INBRED STRAINS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0025918618     PISSN: 00281298     EISSN: 14321912     Source Type: Journal    
DOI: 10.1007/BF00170651     Document Type: Article

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