The pharmacology of fluparoxan: a selective α2‐adrenoceptor antagonist

British Journal of Pharmacology

Volumn 102, Issue 4, 1991, Pages 887-895

  Halliday, C A ^a   Jones, B J ^a   Skingle, M ^a   Walsh, D M ^a   Wise, H ^a   Tyers, M B ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

fluparoxan; GR 50360; idazoxan; 2 Adrenoceptor antagonist

Indexed keywords

2 DIPROPYLAMINO 8 HYDROXYTETRALIN; ALPHA 2 ADRENERGIC RECEPTOR; ALPHA 2 ADRENERGIC RECEPTOR BLOCKING AGENT; AMITRIPTYLINE; ATROPINE; BRIMONIDINE; BUTACLAMOL; CLONIDINE; CYANOPINDOLOL; DESIPRAMINE; DOPAMINE; FLUPAROXAN; HISTAMINE; IDAZOXAN; ISOPRENALINE; KETANSERIN; METHOXAMINE; METHYLSCOPOLAMINE; MUSCARINE; NEUROTRANSMITTER RECEPTOR; OUABAIN; PARGYLINE; PHENYLEPHRINE; PIRENZEPINE; PROPRANOLOL; RADIOLIGAND; SEROTONIN; SPIPERONE; YOHIMBINE;

ANALGESIA; ANIMAL EXPERIMENT; ANIMAL TISSUE; ANOCOCCYGEUS MUSCLE; ARTICLE; BODY TEMPERATURE; BRADYCARDIA; CONTROLLED STUDY; DOG; GUINEA PIG; HYPOTHERMIA; ILEUM; INTRAVENOUS DRUG ADMINISTRATION; MALE; MOUSE; NONHUMAN; ORAL DRUG ADMINISTRATION; PRIORITY JOURNAL; RABBIT; RAT; SEDATION; SMOOTH MUSCLE CONTRACTILITY; VAS DEFERENS;

ADRENERGIC ALPHA-AGONISTS; ADRENERGIC ALPHA-ANTAGONISTS; ANALGESICS; ANIMAL; AORTA; BODY TEMPERATURE; CLONIDINE; EQUILIBRIUM; GUINEA PIGS; HEART RATE; ILEUM; IN VITRO; MALE; MUSCLE, SMOOTH; NOREPINEPHRINE; PIPEROXAN; PYRROLES; QUINOXALINES; RABBITS; RATS; RATS, INBRED STRAINS; RECEPTORS, ADRENERGIC, ALPHA; RECEPTORS, DOPAMINE; RECEPTORS, HISTAMINE; RECEPTORS, MUSCARINIC; RECEPTORS, SEROTONIN; VAS DEFERENS;

EID: 0025825190     PISSN: 00071188     EISSN: 14765381     Source Type: Journal    
DOI: 10.1111/j.1476-5381.1991.tb12272.x     Document Type: Article

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