Synthesis and Antitumor Activity of 9-[(Carbamoyloxy)alkyl]anthracyclines: A Novel Class of Anthracycline Derivatives

Journal of Medicinal Chemistry

Volumn 33, Issue 9, 1990, Pages 2380-2384

  Adams, Nigei ^a   Blake, Colin ^a   Broadhurst, Michael J ^a   Bushnell, David J ^a   Hassall, Cedric H ^a   Hartmann, Hans R ^a   Keech, Elizabeth ^a   Stratton, Alan R ^a   Thomas, Gareth J ^a  

^a ROCHE PRODUCTS LTD   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

9 DEACETYL 4 DEMETHOXY 9 (PHENYLCARBAMOYLOXYMETHYL) 4' EPIDAUNORUBICIN; DAUNORUBICIN; DOXORUBICIN; IDARUBICIN; IDARUBICIN DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; DRUG SCREENING; DRUG SYNTHESIS; INTRAPERITONEAL DRUG ADMINISTRATION; LEUKEMIA L 1210; LEUKOPENIA; MOUSE; NONHUMAN; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

ANIMAL; ANTIBIOTICS, ANTHRACYCLINE; CARBAMATES; CHEMISTRY; FEMALE; LEUKEMIA L1210; MICE; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0025184823     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm00171a011     Document Type: Article

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