Novel α2-adrenoceptor antagonists show selectivity for α2A- and α2B-adrenoceptor subtypes

European Journal of Pharmacology

Volumn 168, Issue 3, 1989, Pages 381-386

  Young, Paul ^a   Berge, John ^a   Chapman, Helen ^a   Cawthorne, Michael A ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

2 (1 METHYL 2 ISOINDOLINYLMETHYL) 2 IMIDAZOLINE; 2 (5 CHLORO 2 ISOINDOLINYLMETHYL) 2 IMIDAZOLINE; 2 (5 CHLOROISOINDOLINYLMETHYL) 2 IMIDAZOLINE; 2 ISOINDOLINYLMETHYL 2 IMIDAZOLINE DERIVATIVE; 2,3,9,13B TETRAHYDRO 1,2 DIMETHYL 1H IMIDAZO[3,4 F]MORPHANTHRIDINE; ALPHA 2 ADRENERGIC RECEPTOR; OXYMETAZOLINE; PHENTOLAMINE; PRAZOSIN; RADIOISOTOPE; RAUWOLSCINE; RECEPTOR SUBTYPE; UNCLASSIFIED DRUG;

ANIMAL CELL; BRAIN CORTEX; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; HUMAN; HUMAN CELL; LUNG; MALE; NONHUMAN; NORMAL HUMAN; PRIORITY JOURNAL; RAT; RECEPTOR AFFINITY; THROMBOCYTE MEMBRANE; VOLUNTEER;

ADRENERGIC ALPHA-ANTAGONISTS; ANIMAL; ANIMALS, NEWBORN; BINDING, COMPETITIVE; BLOOD PLATELETS; CEREBRAL CORTEX; IN VITRO; KINETICS; LUNG; MALE; OXYMETAZOLINE; PRAZOSIN; RATS; RATS, INBRED STRAINS; RECEPTORS, ADRENERGIC, ALPHA; YOHIMBINE;

EID: 0024422263     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/0014-2999(89)90801-7     Document Type: Article

References (13)

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