2,4-Diamino-6,7-dimethoxyquinoline Derivatives as α1-Adrenoceptor Antagonists and Antihypertensive Agents

Journal of Medicinal Chemistry

Volumn 31, Issue 5, 1988, Pages 1031-1035

  Campbell, Simon F ^a   David Hardstone, J ^a   Palmer, Michael J ^a  

^a PFIZER GLOBAL RESEARCH AND DEVELOPMENT   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ALPHA 1 ADRENERGIC RECEPTOR; PRAZOSIN; QUINOLINE DERIVATIVE; RADIOISOTOPE;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; DRUG RECEPTOR BINDING; HYPERTENSION; NONHUMAN; ORAL DRUG ADMINISTRATION; RAT;

ADRENERGIC ALPHA-ANTAGONISTS; ANIMAL; ANTIHYPERTENSIVE AGENTS; BINDING, COMPETITIVE; BRAIN; CHEMISTRY; IN VITRO; QUINOLINES; RADIOLIGAND ASSAY; RATS; RATS, INBRED SHR; RECEPTORS, ADRENERGIC, ALPHA; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0023936336     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm00400a025     Document Type: Article

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