Hydrolysis of 3H-bambuterol, a carbamate prodrug of terbutaline, in blood from humans and laboratory animals in vitro

Biochemical Pharmacology

Volumn 37, Issue 20, 1988, Pages 3867-3876

  Tunek, Anders ^a   Levin, Eva ^a   Svensson, Leif Å ^a  

^a Research and Development Department   (Sweden)

Author keywords

[No Author keywords available]

Indexed keywords

BAMBUTEROL; CARBAMIC ACID DERIVATIVE; CHOLINESTERASE; DRUG DERIVATIVE; PHYSOSTIGMINE; PRODRUG; TERBUTALINE; DRUG METABOLITE; RADIOISOTOPE;

ADULT; ANIMAL; ARTICLE; BLOOD; FEMALE; HUMAN; HYDROLYSIS; IN VITRO STUDY; KINETICS; MALE; MOUSE; RABBIT; RAT; RAT STRAIN; ANIMAL CELL; BLOOD LEVEL; DRUG METABOLISM; HUMAN CELL; LIQUID CHROMATOGRAPHY; NONHUMAN; PRIORITY JOURNAL;

ADULT; ANIMAL; BUTYRYLCHOLINESTERASE; CARBAMATES; FEMALE; HUMAN; HYDROLYSIS; IN VITRO; KINETICS; MALE; MICE; PHYSOSTIGMINE; PRODRUGS; RABBITS; RATS; RATS, INBRED STRAINS; TERBUTALINE;

EID: 0023820851     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/0006-2952(88)90068-8     Document Type: Article

References (12)

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9. Mode of action of anticholinesterases
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11. Pharmacokinetic properties of bambuterol in solution and tablet-basis for once-daily dosage in asthma. III World Conference on Clinical Pharmacology and Therapeutics