Synthesis and Activity of Optical Isomers of Nipradilol1)

Chemical and Pharmaceutical Bulletin

Volumn 35, Issue 9, 1987, Pages 3691-3698

  Shiratsuchi, Masami ^a   Kawamura, Kiyoshi ^a   Akashi, Toshihiro ^a   Ishihama, Hiroshi ^a   Nakamura, Masaki ^a   Takenaka, Fumio ^a  

^a KOWA COMPANY LTD   (Japan)

Author keywords

benzopyran; nipradilol; optical isomer; synthesis; vasodilating activity; blocking activity; blocking activity

Indexed keywords

NIPRADILOL; PROPRANOLOL;

ANIMAL CELL; BETA ADRENERGIC RECEPTOR BLOCKING; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; NONHUMAN; STRUCTURE ACTIVITY RELATION; VASODILATATION;

ADRENERGIC ALPHA-ANTAGONISTS; ANIMAL; DOGS; GUINEA PIGS; IN VITRO; PROPANOLAMINES; STEREOISOMERISM;

EID: 0023550191     PISSN: 00092363     EISSN: 13475223     Source Type: Journal    
DOI: 10.1248/cpb.35.3691     Document Type: Article

References (13)

1. This work was presented at the 7th Symposium on Medicinal Chemistry, Pharmaceutical Society of Japan, Gifu, 1985.
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