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Volumn 50, Issue 1-3, 1987, Pages 147-161

In vitro and in vivo studies demonstrating potent and selective estrogen inhibition with the nonsteroidal aromatase inhibitor CGS 16949A

Author keywords

[No Author keywords available]

Indexed keywords

AMINOGLUTETHIMIDE; ANDROSTENEDIONE; AROMATASE; AROMATASE INHIBITOR; ESTROGEN; FADROZOLE; RADIOISOTOPE; TESTOSTERONE;

EID: 0023517368     PISSN: 0039128X     EISSN: None     Source Type: Journal    
DOI: 10.1016/0039-128X(83)90068-5     Document Type: Article
Times cited : (212)

References (24)
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    • Thompson1    Siiteri2
  • 2
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    • Graves1    Salhanick2
  • 5
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  • 7
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    • Samojlik1    Veldhuis2    Wells3    Santen4
  • 9
    • 0018868660 scopus 로고
    • Modifications of enzymatic activity and difference spectra of cytochrome P-450 from various sources by cholesterol side-chain cleavage inhibitors
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    • Graves1    Uzgiris2    Salhanick3
  • 10
    • 0016293443 scopus 로고
    • Utilization of oxygen and reduced nicotinamide adenine dinucleotide phosphate by human placental microsomes during aromatization of androstenedione
    • (1974) J Biol Chem , vol.249 , pp. 5364-5372
    • Thompson1    Siiteri2
  • 11
    • 0018760737 scopus 로고
    • Enzymological studies of rat luteinized ovaries in relation to acute reduction of aromatizable androgen formation and stimulated production of progestins
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    • Suzuki1    Tamaoki2
  • 15
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    • Kinetic properties of human placental aromatase
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  • 17
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    • Evidence of the direct aromatization of testosterone and different aromatization sites for testosterone and androstenedione in human placental microsomes
    • (1974) Biochemistry , vol.13 , pp. 1925-1931
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  • 18
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    • Substrate specificity of the placental microsomal aromatase
    • (1980) Steroids , vol.36 , pp. 507-519
    • Gibb1    Lavoie2
  • 19
    • 0017367812 scopus 로고
    • Aromatization of androstenedione, 19-hydroxy-androstenedione, and 19-oxo-androstenedione at a common catalytic site in human placental microsomes
    • (1977) Biochemistry , vol.16 , pp. 140-145
    • Kelly1    Judd2    Stolee3
  • 24
    • 0019199963 scopus 로고
    • Postovulatory decrease in estrogen production is caused by the diminished supply of aromatizable androgen to ovarian aromatase
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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.