Solid phase synthesis of peptides containing the CH2NH peptide bond isostere

Peptides

Volumn 8, Issue 1, 1987, Pages 119-121

  Sasaki, Yusuke ^a   Coy, David H ^a  

^a TULANE UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

Peptide bond isostere; Peptide synthesis; Somatostatin analogs

Indexed keywords

SOMATOSTATIN ANALOG;

NONHUMAN; PEPTIDE SYNTHESIS; PRIORITY JOURNAL; SOLID PHASE CHEMISTRY;

ALKYLATION; AMINES; OXIDATION-REDUCTION; PEPTIDES; SUPPORT, U.S. GOV'T, P.H.S.;

EID: 0023150034     PISSN: 01969781     EISSN: None     Source Type: Journal    
DOI: 10.1016/0196-9781(87)90174-4     Document Type: Article

References (9)

1. The cyanohydridoborate anion as a selective reducing agent
2. An efficient synthesis of optically active α-(t-butoxycarbonylamino)-aldehydes from α-amino acids
3. Color test for detection of free terminal amino groups in the solid-phase synthesis of peptides
4. Synthesis and biological activities of some pseudo-peptide analogues of tetragastrin: the importance of the peptide backbone
5. Synthesis and biological actions of prosomatostatin
6. Octapeptide analogs of somatostatin exhibiting greatly enhanced in vivo and in vitro inhibition of growth hormone secretion
7. Synthesis of pseudo-peptide analogues of the C-terminal tetrapeptide of gastrin and evaluation of their biological activity on acid secretion
8. Peptide backbone modifications: A structure-activity analysis of peptides containing amide bond surrogates
9. Potent new inhibitors of human renin