2-Phenylindenes: Development of a New Mammary Tumor Inhibiting Antiestrogen by Combination of Estrogenic Side Effect Lowering Structural Elements

Journal of Medicinal Chemistry

Volumn 29, Issue 1, 1986, Pages 75-79

  Schneider, Martin R ^a   Ball, Hartwig ^a  

^a UNIVERSITY OF REGENSBURG   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIESTROGEN; ANTINEOPLASTIC AGENT; DIETHYLSTILBESTROL; ESTRADIOL; ESTROGEN; ESTRONE; NEW DRUG; RADIOISOTOPE;

2 PHENYLINDENE DERIVATIVE; 5,6 DIACETOXY 2 (3,4 DIACETOXYPHENYL) 3 ETHYL 1 METHYL 3H INDENE; ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; BREAST; BREAST CANCER; CANCER CHEMOTHERAPY; CATTLE; CELL STRAIN MXT; DOSE RESPONSE; DRUG ANALYSIS; DRUG ANTAGONISM; DRUG COMPARISON; DRUG EFFICACY; DRUG IDENTIFICATION; DRUG RECEPTOR BINDING; DRUG RESPONSE; DRUG SCREENING; DRUG SYNTHESIS; ESTRADIOL H 3; FEMALE GENITAL SYSTEM; MOUSE; NONHUMAN; PHARMACOKINETICS; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION; SUBCUTANEOUS DRUG ADMINISTRATION; THERAPY; UTERUS WEIGHT;

ANIMAL; BINDING, COMPETITIVE; BIOLOGICAL ASSAY; CATTLE; CHEMISTRY; COMPARATIVE STUDY; ESTRADIOL; ESTROGEN ANTAGONISTS; ESTRONE; FEMALE; INDENES; MAMMARY NEOPLASMS, EXPERIMENTAL; MICE; ORGAN WEIGHT; RECEPTORS, ESTRADIOL; STILBENES; STRUCTURE-ACTIVITY RELATIONSHIP; SUPPORT, NON-U.S. GOV'T; UTERUS;

EID: 0022607083     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm00151a012     Document Type: Article

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