Analogues of Caffeine and Theophylline: Effect of Structural Alterations on Affinity at Adenosine Receptors

Journal of Medicinal Chemistry

Volumn 29, Issue 7, 1986, Pages 1305-1308

  Daly, J W ^a   Padgett, W L ^a   Shamim, M T ^a  

^a Laboratory of Bioorganic Chemistry ^*  (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

2 CHLOROADENOSINE; ADENOSINE A1 RECEPTOR; ADENOSINE A2 RECEPTOR; CAFFEINE; CAFFEINE DERIVATIVE; RADIOISOTOPE; THEOPHYLLINE; THEOPHYLLINE DERIVATIVE; XANTHINE DERIVATIVE;

6 N CYCLOHEXYLADENOSINE H 3; 7 PROPARGYL 1,3 DIPROPYLXANTHINE; ADENINE H 3; ANIMAL CELL; BIOLOGICAL MODEL; BRAIN; CENTRAL NERVOUS SYSTEM; DRUG ANALYSIS; DRUG ANTAGONISM; DRUG COMPARISON; DRUG IDENTIFICATION; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG SYNTHESIS; GUINEA PIG; NONHUMAN; PHARMACOKINETICS; RAT; STRUCTURE ACTIVITY RELATION;

ANIMAL; CAFFEINE; CELL MEMBRANE; CEREBRAL CORTEX; COMPARATIVE STUDY; INDICATORS AND REAGENTS; RATS; RECEPTORS, PURINERGIC; SPECTRUM ANALYSIS, MASS; STRUCTURE-ACTIVITY RELATIONSHIP; SUPPORT, NON-U.S. GOV'T; THEOPHYLLINE; XANTHINES;

EID: 0022544144     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm00157a035     Document Type: Article

References (7)

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